Target Details
| UniProt AC | P25025 |
|---|---|
| Gene Symbol | CXCR2 |
| Protein Name | C-X-C chemokine receptor type 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 224
- Clinical molecules 0
- Avg pChEMBL 7.63
KEGG Pathways (7)
Associated Diseases (1)
Active Molecules (224)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UDJPTWYRKLFZEK
|
8.3 | Ki | 2 | — | |
UJPYCQPUOFQYIE
|
8.3 | Ki | 2 | — | |
UNUGDTFIICVXIP
|
8.3 | IC50 | 2 | — | |
VBCZYGZLNUHVPO
|
8.3 | Ki | 2 | — | |
XPVZCYDESBRJFA
|
8.3 | IC50 | 2 | — | |
YVZGSKYWJOEQBN
|
8.3 | Ki | 2 | — | |
ZYESTBRTKPGMTF
|
8.3 | Ki | 2 | — | |
FVNZKJFLVPSOMX
|
8.3 | IC50 | 2 | — | |
KQDRVXQXKZXMHP
|
8.3 | IC50 | 2 | — | |
ACYREHAZQPOKBX
|
8.3 | IC50 | 2 | — | |
XNPQHVAEYPMNED
|
8.3 | IC50 | 2 | — | |
NFCNTLMYLMTDEB
|
8.2 | IC50 | 2 | — | |
RXIUEIPPLAFSDF
|
8.2 | IC50 | 2 | — | |
GEWHNBHOBDABRZ
|
8.2 | IC50 | 2 | — | |
ULCDGLYZEHBIFT
|
8.2 | IC50 | 2 | — | |
VVCVHUHCUBCBGN
|
8.2 | Ki | 2 | — | |
LZWZAAXBIRFFQO
|
8.2 | IC50 | 2 | — | |
QPGNAJBQDXRPEA
|
8.2 | IC50 | 2 | — | |
XNPQHVAEYPMNED
|
8.2 | IC50 | 2 | — | |
DTKBCDNYQAWTDG
|
8.2 | IC50 | 2 | — | |
ILEJORXRDPNPIM
|
8.2 | IC50 | 2 | — | |
CSVHKWZKMWYMAX
|
8.2 | IC50 | 2 | — | |
GAXCFOGLVNGOBY
|
8.2 | Ki | 2 | — | |
WEGWRFJDASFVFU
|
8.2 | IC50 | 2 | — | |
XDIAMTWURDXGAQ
|
8.2 | Ki | 2 | — | |
HPCHAHFHNCQQJC
|
8.1 | IC50 | 2 | — | |
VYOMLNMMWYPDOS
|
8.1 | IC50 | 2 | — | |
DDMTYZBTPDHBMN
|
8.1 | Ki | 2 | — | |
XOVUJMYKTAPPTR
|
8.1 | IC50 | 2 | — | |
KAVIMWXSTVLBFP
|
8.1 | IC50 | 2 | — | |
KIUIYAHJRLTVRF
|
8.1 | IC50 | 2 | — | |
GAZMRTOTNDECNS
|
8.1 | IC50 | 2 | — | |
VYOMLNMMWYPDOS
|
8.1 | IC50 | 2 | — | |
DNQSYCVLRVJIIH
|
8.1 | IC50 | 2 | — | |
FKEAPOKGKRZRRW
|
8.1 | IC50 | 2 | — | |
GOXKLDRNSZHYPN
|
8.1 | Ki | 2 | — | |
WPWBLYBMUDAPNW
|
8.1 | IC50 | 2 | — | |
XMCIQQDUJUKYBJ
|
8.1 | Ki | 2 | — | |
ONXDSBZQWUWHRA
|
8.0 | IC50 | 2 | — | |
PUFZIIVLLJVRDL
|
8.0 | IC50 | 2 | — | |
YYNIZWVXZWEFEA
|
8.0 | IC50 | 2 | — | |
HKRHEFYVMVBQCG
|
8.0 | Ki | 2 | — | |
OPXPMFMLALQTGS
|
8.0 | Ki | 2 | — | |
XFJBABVMOSLUTO
|
8.0 | IC50 | 2 | — | |
BDLSEEFGQREQHH
|
8.0 | Ki | 2 | — | |
HGTGVULEPQRUEB
|
8.0 | IC50 | 2 | — | |
HJQGYKRAMBLSHY
|
8.0 | Ki | 2 | — | |
PASCQQQYSMLKAC
|
8.0 | Ki | 2 | — | |
HNQKLXTUDLBLDQ
|
7.9 | IC50 | 2 | — | |
DABXGLPZDQYKGO
|
7.9 | Ki | 2 | — |