Target Details
UniProt ACP25025
Gene SymbolCXCR2
Protein NameC-X-C chemokine receptor type 2
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 224
  • Clinical molecules 0
  • Avg pChEMBL 7.63
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (224)
InChIKey pChEMBL Type Targets Clinical
DDLPYOCJHQSVSZ 10.0 IC50 2
KYIGOCCCBXRHNJ 9.6 IC50 43
QIFFSXAXKXBABE 9.2 Ki 2
SHHCDMLDQIVBPV 9.1 Ki 2
QZECRCLSIGFCIO 9.1 IC50 2
WDHCGTYXANMGHV 9.0 Ki 2
DGKQQEVYYPCMNE 8.9 IC50 2
UOURTTOYLTUYKY 8.7 IC50 2
DYCPTIVMRFRWPY 8.7 Ki 2
FPOWMMYKRZVTRO 8.7 Ki 2
HEBGAKBUHZNNIN 8.7 Ki 2
QQQUUPHVVBLGTA 8.7 Ki 2
UNUGDTFIICVXIP 8.6 IC50 2
RSYRCNGIYXIWNH 8.6 IC50 2
JYHUHCFVWDEFFY 8.5 Ki 2
WRZQOIBQWPDIJN 8.5 Ki 2
NFCNTLMYLMTDEB 8.5 IC50 2
PDQPKFKGQOJWGZ 8.5 IC50 2
LINCELSOWBPXFG 8.4 IC50 2
JBJWLRHFBRZPOP 8.4 IC50 2
LGKVILKPRCDSRP 8.4 IC50 2
MYFOCPUZNAPZSE 8.4 IC50 2
ZPVPYCVHNDXDMK 8.4 IC50 2
BRNMYMQVVHGBOR 8.4 Ki 2
DCVPTCRKYYMBDG 8.4 Ki 2
IACZVCYFISPAOZ 8.4 Ki 2
IRTVRKUICFESKI 8.4 IC50 2
OTUJIXWHVZRCBM 8.4 IC50 2
PXRGDKPMOBTHFQ 8.4 Ki 2
PYRYGTVIJGRYHE 8.4 Ki 2
SENJTLMDCKVBAA 8.4 Ki 2
UYLPYMZAFWHRJL 8.4 Ki 2
DPHCMAJDWUKUPJ 8.4 Ki 2
NLXWGGVLQFIGKR 8.4 IC50 2
PISGUALHIYOOTC 8.4 IC50 2
AXLRSENOHOPWNY 8.3 Ki 2
LGKVILKPRCDSRP 8.3 IC50 2
RXIUEIPPLAFSDF 8.3 IC50 2
GYUXYROXDXSLDH 8.3 IC50 2
XSINIJBRURGTOY 8.3 IC50 2
XZECPGNWHKHNIN 8.3 Ki 2
GYUXYROXDXSLDH 8.3 IC50 2
DRBFDAYBUUMUHY 8.3 IC50 2
ARPPAIXHGDGLEQ 8.3 IC50 2
JAQGOALYPJHHST 8.3 Ki 2
JBJWLRHFBRZPOP 8.3 IC50 2
KMESOOYCTQWBIE 8.3 Ki 2
QMTVQFUSOXHPSA 8.3 Ki 2
RDLJCEZYIYATCE 8.3 Ki 2
SDCMXLFUIGWAOW 8.3 Ki 2
2D structure