Target Details
| UniProt AC | P25024 |
|---|---|
| Gene Symbol | CXCR1 |
| Protein Name | C-X-C chemokine receptor type 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 198
- Clinical molecules 0
- Avg pChEMBL 7.05
KEGG Pathways (6)
Associated Diseases (1)
Active Molecules (198)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
STUJFSIJLYQOCY
|
6.4 | IC50 | 2 | — | |
CMANXHXTSWTYRG
|
6.4 | IC50 | 2 | — | |
MNULHNJDCIVGAO
|
6.4 | Kd | 2 | — | |
AXLRSENOHOPWNY
|
6.4 | Ki | 2 | — | |
CBIODTKCFBGXHU
|
6.4 | IC50 | 2 | — | |
LPLKAXWKZWWASO
|
6.4 | IC50 | 2 | — | |
MCQSWTLKUIEWQM
|
6.4 | Ki | 2 | — | |
WOBYQWNRYZGWRU
|
6.4 | IC50 | 2 | — | |
TVANIYMHXPLFFL
|
6.4 | IC50 | 2 | — | |
NEZMHIVTYRWBEX
|
6.4 | IC50 | 2 | — | |
VOAPNZIKRKHEHR
|
6.4 | IC50 | 2 | — | |
PDQPKFKGQOJWGZ
|
6.4 | IC50 | 2 | — | |
UKBAGMZMGJKUER
|
6.3 | IC50 | 2 | — | |
XSINIJBRURGTOY
|
6.3 | IC50 | 2 | — | |
PPCFLIBERCNFID
|
6.3 | IC50 | 2 | — | |
XEJUWHPWBDYKSK
|
6.3 | IC50 | 2 | — | |
KBLOFZHBIDLNIS
|
6.3 | IC50 | 2 | — | |
NTWHZYBSKKHULS
|
6.3 | IC50 | 2 | — | |
ONXDSBZQWUWHRA
|
6.3 | IC50 | 2 | — | |
OISJPBYRKOJZRI
|
6.3 | IC50 | 2 | — | |
OISJPBYRKOJZRI
|
6.3 | IC50 | 2 | — | |
DTKBCDNYQAWTDG
|
6.2 | IC50 | 2 | — | |
MRHPZVNAGXMSIH
|
6.2 | IC50 | 2 | — | |
GULGFHPSYNQMBP
|
6.2 | IC50 | 2 | — | |
SIUQYAWDXLUCLD
|
6.2 | IC50 | 4 | — | |
DGGJPUBUCAEEHT
|
6.2 | IC50 | 2 | — | |
PASCQQQYSMLKAC
|
6.2 | Ki | 2 | — | |
QUKXEAVCHJVKEA
|
6.2 | IC50 | 2 | — | |
XETXTFIIXKTWPQ
|
6.2 | IC50 | 2 | — | |
SIUQYAWDXLUCLD
|
6.2 | IC50 | 2 | — | |
ASWBTVXNCFSFOM
|
6.2 | IC50 | 2 | — | |
KCIRBTXGALUYHT
|
6.2 | IC50 | 2 | — | |
QMQGUUOGRMUXFL
|
6.2 | IC50 | 2 | — | |
PUFZIIVLLJVRDL
|
6.2 | IC50 | 2 | — | |
SJWVRSVJDTUULR
|
6.2 | IC50 | 2 | — | |
AHAOUMFJVVZFDM
|
6.1 | IC50 | 2 | — | |
IYZWLQHDOCJREA
|
6.1 | IC50 | 2 | — | |
ACYREHAZQPOKBX
|
6.1 | IC50 | 2 | — | |
GAZMRTOTNDECNS
|
6.1 | IC50 | 2 | — | |
HGTGVULEPQRUEB
|
6.1 | IC50 | 2 | — | |
OISJPBYRKOJZRI
|
6.1 | IC50 | 2 | — | |
XOVUJMYKTAPPTR
|
6.1 | IC50 | 2 | — | |
PCXDKTNTSYUMHN
|
6.1 | IC50 | 2 | — | |
NLXWGGVLQFIGKR
|
6.1 | IC50 | 2 | — | |
VZRIHFZJVIOJBE
|
6.1 | IC50 | 2 | — | |
JVOHPOBSHINFNU
|
6.0 | IC50 | 2 | — | |
RZXVFVRPSNXVEC
|
6.0 | IC50 | 2 | — | |
PFVOSGMAMDBGFG
|
6.0 | IC50 | 2 | — |