Target Details
| UniProt AC | P25024 |
|---|---|
| Gene Symbol | CXCR1 |
| Protein Name | C-X-C chemokine receptor type 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 198
- Clinical molecules 0
- Avg pChEMBL 7.05
KEGG Pathways (6)
Associated Diseases (1)
Active Molecules (198)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HEFNNWSXXWATRW
|
7.0 | IC50 | 3 | — | |
QIBUUCFTHGXSFM
|
7.0 | IC50 | 2 | — | |
BIVKRDOOTZFPRA
|
7.0 | IC50 | 2 | — | |
ZHOSAEFOHKXJDJ
|
6.9 | IC50 | 5 | — | |
YWEPAFKNLSBBBU
|
6.9 | IC50 | 3 | — | |
HJQGYKRAMBLSHY
|
6.9 | Ki | 2 | — | |
HKRHEFYVMVBQCG
|
6.9 | Ki | 2 | — | |
XFJBABVMOSLUTO
|
6.9 | IC50 | 2 | — | |
XMCIQQDUJUKYBJ
|
6.9 | Ki | 2 | — | |
XNPQHVAEYPMNED
|
6.9 | IC50 | 2 | — | |
ARPPAIXHGDGLEQ
|
6.8 | IC50 | 2 | — | |
ZPVPYCVHNDXDMK
|
6.8 | IC50 | 2 | — | |
LZWZAAXBIRFFQO
|
6.8 | IC50 | 2 | — | |
WCBDQNUHQNEQLF
|
6.8 | IC50 | 2 | — | |
NFCNTLMYLMTDEB
|
6.8 | IC50 | 2 | — | |
HDQNDRCZSVEGSG
|
6.8 | IC50 | 2 | — | |
VYOMLNMMWYPDOS
|
6.8 | IC50 | 2 | — | |
XNPQHVAEYPMNED
|
6.8 | IC50 | 2 | — | |
FVNZKJFLVPSOMX
|
6.7 | IC50 | 2 | — | |
RSYRCNGIYXIWNH
|
6.7 | IC50 | 2 | — | |
MSJKBTMMJKJYHB
|
6.7 | IC50 | 2 | — | |
SSBIYBNARHHMGE
|
6.7 | Ki | 2 | — | |
WEGWRFJDASFVFU
|
6.7 | IC50 | 2 | — | |
OTUJIXWHVZRCBM
|
6.7 | IC50 | 2 | — | |
DRBFDAYBUUMUHY
|
6.7 | IC50 | 2 | — | |
VZNLCSKTOPAQML
|
6.7 | IC50 | 2 | — | |
KBLOFZHBIDLNIS
|
6.7 | IC50 | 2 | — | |
DNQSYCVLRVJIIH
|
6.7 | IC50 | 2 | — | |
KAVIMWXSTVLBFP
|
6.7 | IC50 | 2 | — | |
YFTUGOHVHFFSHQ
|
6.7 | IC50 | 2 | — | |
ZMLPGOTZQCYELQ
|
6.7 | IC50 | 2 | — | |
UNUGDTFIICVXIP
|
6.7 | IC50 | 2 | — | |
VYOMLNMMWYPDOS
|
6.7 | IC50 | 2 | — | |
JBBKREGWJICILL
|
6.6 | IC50 | 2 | — | |
SGLBQNTUAMMYTP
|
6.6 | IC50 | 2 | — | |
XBPBJDFJAWKYCK
|
6.6 | IC50 | 2 | — | |
BGHMYZUFTBKLKU
|
6.6 | IC50 | 2 | — | |
GYUXYROXDXSLDH
|
6.6 | IC50 | 2 | — | |
VWSXKWXISJLOQM
|
6.6 | IC50 | 6 | — | |
GYUXYROXDXSLDH
|
6.6 | IC50 | 2 | — | |
PYRYGTVIJGRYHE
|
6.5 | Ki | 2 | — | |
KIUIYAHJRLTVRF
|
6.5 | IC50 | 2 | — | |
WPWBLYBMUDAPNW
|
6.5 | IC50 | 2 | — | |
DXPCTOZNUCZJPC
|
6.5 | Ki | 2 | — | |
YYNIZWVXZWEFEA
|
6.5 | IC50 | 2 | — | |
MMVFNAGMKWQAKS
|
6.5 | IC50 | 4 | — | |
MXCRXBCGEWUMNZ
|
6.5 | IC50 | 2 | — | |
ZHAAHVPYFDDLLE
|
6.5 | IC50 | 2 | — | |
QMTVQFUSOXHPSA
|
6.5 | IC50 | 2 | — | |
HPCHAHFHNCQQJC
|
6.5 | IC50 | 2 | — |