Target Details
| UniProt AC | P25024 |
|---|---|
| Gene Symbol | CXCR1 |
| Protein Name | C-X-C chemokine receptor type 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 198
- Clinical molecules 0
- Avg pChEMBL 7.05
KEGG Pathways (6)
Associated Diseases (1)
Active Molecules (198)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DYCPTIVMRFRWPY
|
7.5 | Ki | 2 | — | |
QPGNAJBQDXRPEA
|
7.5 | IC50 | 2 | — | |
WYWJXUDCXPYMIQ
|
7.5 | Ki | 2 | — | |
XDIAMTWURDXGAQ
|
7.5 | Ki | 2 | — | |
BGXSRDRXCPKCLB
|
7.4 | IC50 | 2 | — | |
KBLOFZHBIDLNIS
|
7.4 | IC50 | 5 | — | |
RXIUEIPPLAFSDF
|
7.4 | IC50 | 2 | — | |
HNQKLXTUDLBLDQ
|
7.4 | IC50 | 2 | — | |
UXUIKTKXWYNOMQ
|
7.4 | Ki | 2 | — | |
ILEJORXRDPNPIM
|
7.4 | IC50 | 2 | — | |
IPLGVPPLWIAZSG
|
7.4 | Ki | 2 | — | |
UTDWJMBRBOKFJV
|
7.4 | IC50 | 2 | — | |
OQCIAVOJSLDHHC
|
7.4 | Ki | 2 | — | |
JBBKREGWJICILL
|
7.4 | IC50 | 5 | — | |
SHLGVUBRPWNMLF
|
7.4 | IC50 | 2 | — | |
FNGBYTBDUQDISM
|
7.4 | IC50 | 2 | — | |
GAXCFOGLVNGOBY
|
7.4 | Ki | 2 | — | |
QPFHUUXBBCZCOF
|
7.3 | IC50 | 2 | — | |
XZECPGNWHKHNIN
|
7.3 | Ki | 2 | — | |
YTTGJPIBJUDFQG
|
7.3 | IC50 | 2 | — | |
DKYWVDODHFEZIM
|
7.3 | IC50 | 4 | — | |
FPOWMMYKRZVTRO
|
7.3 | Ki | 2 | — | |
GEWHNBHOBDABRZ
|
7.3 | IC50 | 2 | — | |
KMOKWTXCNPBSHR
|
7.3 | IC50 | 2 | — | |
DLHXKIOUORFOQU
|
7.3 | IC50 | 2 | — | |
FIBJPCXODZVPBQ
|
7.3 | Ki | 2 | — | |
JYHUHCFVWDEFFY
|
7.3 | Ki | 2 | — | |
VBCZYGZLNUHVPO
|
7.3 | Ki | 2 | — | |
LINCELSOWBPXFG
|
7.3 | IC50 | 2 | — | |
XPVZCYDESBRJFA
|
7.3 | IC50 | 2 | — | |
BDLSEEFGQREQHH
|
7.2 | Ki | 2 | — | |
LGKVILKPRCDSRP
|
7.2 | IC50 | 2 | — | |
JBJWLRHFBRZPOP
|
7.2 | IC50 | 2 | — | |
KCVWGCOBGFLUEB
|
7.1 | IC50 | 5 | — | |
GMNNTQPTKYJUKQ
|
7.1 | IC50 | 2 | — | |
KQDRVXQXKZXMHP
|
7.1 | IC50 | 2 | — | |
LQUGDEWJKLEGOJ
|
7.1 | IC50 | 2 | — | |
UUNDOBHSENXEFU
|
7.0 | IC50 | 2 | — | |
APDVPDFSMORZLD
|
7.0 | IC50 | 2 | — | |
UNUGDTFIICVXIP
|
7.0 | IC50 | 2 | — | |
CSVHKWZKMWYMAX
|
7.0 | IC50 | 2 | — | |
HEFNNWSXXWATRW
|
7.0 | IC50 | 5 | — | |
LGKVILKPRCDSRP
|
7.0 | IC50 | 2 | — | |
QEOSQTDOWDCAEV
|
7.0 | Kd | 2 | — | |
RXIUEIPPLAFSDF
|
7.0 | IC50 | 2 | — | |
SDCMXLFUIGWAOW
|
7.0 | Ki | 2 | — | |
JAQGOALYPJHHST
|
7.0 | Ki | 2 | — | |
NFCNTLMYLMTDEB
|
7.0 | IC50 | 2 | — | |
ULCDGLYZEHBIFT
|
7.0 | IC50 | 2 | — | |
HDQNDRCZSVEGSG
|
7.0 | IC50 | 5 | — |