Target Details
UniProt ACP25024
Gene SymbolCXCR1
Protein NameC-X-C chemokine receptor type 1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 198
  • Clinical molecules 0
  • Avg pChEMBL 7.05
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (198)
InChIKey pChEMBL Type Targets Clinical
DDLPYOCJHQSVSZ 10.0 IC50 2
QZECRCLSIGFCIO 9.4 Kd 2
KQDRVXQXKZXMHP 9.0 IC50 2
UOURTTOYLTUYKY 8.7 IC50 2
KRRJDGLUFFFYHX 8.5 IC50 2
DGKQQEVYYPCMNE 8.3 IC50 2
PXRGDKPMOBTHFQ 8.3 Ki 2
HEBGAKBUHZNNIN 8.2 Ki 2
NICQNGMZJXZBJM 8.2 Ki 2
OPXPMFMLALQTGS 8.2 Ki 2
IRTVRKUICFESKI 8.2 IC50 2
WDHCGTYXANMGHV 8.2 Ki 2
MWABJGSIPHBDDC 8.1 Ki 2
QIFFSXAXKXBABE 8.1 Ki 2
YVZGSKYWJOEQBN 8.1 Ki 2
SENJTLMDCKVBAA 8.1 Ki 2
UJPYCQPUOFQYIE 8.1 Ki 2
DCVPTCRKYYMBDG 8.0 Ki 2
IACZVCYFISPAOZ 8.0 Ki 2
WRZQOIBQWPDIJN 8.0 Ki 2
MYFOCPUZNAPZSE 8.0 IC50 2
UYLPYMZAFWHRJL 8.0 Ki 2
DCOPUUMXTXDBNB 7.9 IC50 5
LUNAFTMLJLEOEQ 7.9 Ki 2
BRNMYMQVVHGBOR 7.8 Ki 2
GOXKLDRNSZHYPN 7.8 Ki 2
SCSNKXZAGMCAGA 7.8 Ki 2
PSPSMPJFVZTXSD 7.8 Ki 2
UNPQYPMTWSIZRR 7.8 Ki 2
VVCVHUHCUBCBGN 7.8 Ki 2
WWSNTFDUUVNWIC 7.8 Ki 2
DGPHJNJINCRCKW 7.7 IC50 5
HCGUUQDQSYMJAU 7.7 IC50 2
RDLJCEZYIYATCE 7.7 Ki 2
PISGUALHIYOOTC 7.7 IC50 2
XZVGETAASKRSBI 7.7 Ki 2
CODGMHXCDXLYFF 7.7 IC50 2
KMESOOYCTQWBIE 7.7 Ki 2
MQBZVUNNWUIPMK 7.7 IC50 3
DDMTYZBTPDHBMN 7.6 Ki 2
ZYESTBRTKPGMTF 7.6 Ki 2
QQQUUPHVVBLGTA 7.6 Ki 2
JBJWLRHFBRZPOP 7.6 IC50 2
DABXGLPZDQYKGO 7.5 Ki 2
FKEAPOKGKRZRRW 7.5 IC50 2
SHHCDMLDQIVBPV 7.5 Ki 2
SPLGZZDGUQTEHE 7.5 IC50 5
UDJPTWYRKLFZEK 7.5 Ki 2
AEDMWJARWOMJKQ 7.5 IC50 2
DKYWVDODHFEZIM 7.5 IC50 3
2D structure