Target Details
UniProt ACP25021
Gene SymbolHRH2
Protein NameHistamine H2 receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 120
  • Clinical molecules 9
  • Avg pChEMBL 7.06
Top Co-occurrence Targets
Active Molecules (120)
InChIKey pChEMBL Type Targets Clinical
DDBBPVWZBRHZDD 7.2 Kd 4
IZCLJDQWYJTBAN 7.2 Ki 3
UWTPDHDYCBTOMN 7.2 Kd 4
VMXUWOKSQNHOCA 7.2 Kd 4
BIJXMFDKONGOAN 7.2 Kd 4
ONVSJLPIADFJKR 7.2 Kd 4
SAEILUJHGHNPAN 7.2 Kd 4
UAFKZBOQJUSIDU 7.2 Kd 4
VFGWQQNKIVMZLG 7.2 Ki 3
GOPXEUGGDXDMDT 7.2 Ki 3
BIZMGZSJEDDVNF 7.1 Ki 3
XNSQSOGNTZGMDA 7.1 Kd 4
UGRVOYIHHOLSHQ 7.1 Ki 3
YVENIGOVHPMTDH 7.1 Ki 23
DVSMVUMYJDOPJQ 7.1 Ki 16
RHRPOJKRNUHOJA 7.1 Kd 4
PCFGLLVVPCPPIG 7.0 Kd 4
BFCDFTHTSVTWOG 7.0 IC50 11
BKRGVLQUQGGVSM 6.9 Ki 26 Yes
GUTIIYCXIXRNPB 6.9 Ki 2
AQIXAKUUQRKLND 6.8 Ki 2
KYIGOCCCBXRHNJ 6.8 IC50 43
WEGLOYDTDILXDA 6.8 Ki 22
BNXNWRSVYQHTOH 6.8 Ki 12
YQNWZWMKLDQSAC 6.7 Ki 15
JJCFRYNCJDLXIK 6.7 IC50 25 Yes
QXYZJXCNTMMWEO 6.7 Ki 15
FOLXSEMOHDUPCN 6.6 Ki 15
LTBDUUVNJFIMTM 6.6 Kd 2
NTYJJOPFIAHURM 6.6 Ki 4
SGUZNMAAJVIZHU 6.6 Ki 14
GKTQBPYMIGXPKG 6.5 Ki 21 Yes
GKTQBPYMIGXPKG 6.5 Ki 18
UFIMBHYPDHTMKA 6.4 Ki 4
YNNUSGIPVFPVBX 6.4 IC50 24 Yes
GALCSZPFCCZIBC 6.4 IC50 20 Yes
QSLMDECMDJKHMQ 6.4 IC50 20
TWMXGXSGGIIQDM 6.4 Ki 5
UBNDBTRGSCEYOS 6.4 Ki 7
SHKOYYABTMCHBH 6.3 Ki 3
VDCBDIRJDJYCIZ 6.3 Ki 5
KOIIIBWVKNCMBP 6.3 Ki 2
GOFKTWKLJPDQCU 6.3 Ki 5
HVGNYVOUQOKFLU 6.3 Ki 5
MZVVLAMPOFUDJD 6.3 Ki 5
ZJBSNCPQNNTTRY 6.3 Ki 2
CJGNMVAAMQAWEF 6.3 Ki 16
FVVJBQFXISQDKF 6.3 Ki 3
QBWLTDPVSJCLIE 6.3 Ki 15
MHNSOBBJZCWUGS 6.2 Ki 17
2D structure