Target Details
UniProt ACP25021
Gene SymbolHRH2
Protein NameHistamine H2 receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 120
  • Clinical molecules 9
  • Avg pChEMBL 7.06
Top Co-occurrence Targets
Active Molecules (120)
InChIKey pChEMBL Type Targets Clinical
GKDBTHSYQZTDAJ 9.1 IC50 13
ZMOPTLXEYOVARP 8.8 Ki 14 Yes
FFKSIHLRCNTALR 8.7 Ki 3
ABDWUBPDHWDFCV 8.3 Ki 2
ZRQMUCDHVVOENY 8.3 Ki 17
VSWBSWWIRNCQIJ 8.2 Ki 4
VSWBSWWIRNCQIJ 8.2 Ki 23
IWBMAAUPHUCYCI 8.2 Kd 20
OVYZCEIGUJNWKN 8.1 Kd 4
GWAMGWDJCYIREE 8.1 Kd 20
IOSVPGDHSQVBED 8.1 Kd 6
LDXAOQSIBXRCIN 8.1 Kd 6
RXDHWPCPLSUTCP 8.1 Kd 4
PKALTNFRHBJDRH 8.1 Kd 6
QVAKGXNPTKFJST 8.0 Kd 6
FASDKYOPVNHBLU 7.9 Kd 9
HKCHNLZUCRQSTO 7.9 Kd 4
JASKXIBVQDMBJJ 7.9 Kd 4
LMBAXHGIFALPQJ 7.9 Kd 4
NNBLASKQLZCYBL 7.9 Kd 4
ZKKBZRDZTBXDKE 7.9 Kd 4
CDGJSIMJNZNZFE 7.9 Kd 6
OJYUKAHOHYUAHF 7.9 Kd 6
KCCBFGKNVMTXIQ 7.8 Kd 6
KGGHECZDYBMALC 7.8 Kd 6
QTIAXUAWMLBIGP 7.7 Ki 3
XQOLXGFKFIWXQP 7.7 Kd 6
HPJNWYRQLUNOIA 7.7 Kd 4
WEGLOYDTDILXDA 7.7 Ki 22
WKXIZVSDLMORMY 7.6 Ki 2
MODBIBJHAWXYOZ 7.6 Kd 20
MWNWERUECAJGJC 7.5 Kd 6
CKIPXVNSJRXNTQ 7.5 Ki 3
MZDWSPIRGJHBII 7.5 Ki 2
YPAOZTCVMTXDID 7.4 Kd 4
YVJCOHIKEMZVAO 7.4 Kd 4
GVGOZYJHWUIVHV 7.4 Ki 2
PMBDKZARCOUAFU 7.4 Ki 3
XUFQPHANEAPEMJ 7.4 IC50 11
USBWQDPYNKDRSV 7.4 Kd 4
BQYXPJXIOSEURA 7.3 Kd 4
QTIAXUAWMLBIGP 7.3 Ki 3
YYXYUTGQFNFTGX 7.3 Kd 4
FARKBYHYALPKMO 7.3 Kd 4
KIRWEWNKOWMEBM 7.3 Kd 4
ZYFQYFZOSKEOGJ 7.3 Kd 4
LKPZDFCAQDGUKZ 7.2 Kd 4
SRELLSOOXBJTLE 7.2 Kd 4
TYUKINNXLNULMD 7.2 Ki 4
CDZGYTJJJXXWBS 7.2 Kd 4
2D structure