Target Details
| UniProt AC | P24941 |
|---|---|
| Gene Symbol | CDK2 |
| Protein Name | Cyclin-dependent kinase 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 5,432
- Clinical molecules 978
- Avg pChEMBL 7.43
KEGG Pathways (19)
- Cell cycle
- Cellular senescence
- Cushing syndrome
- Epstein-Barr virus infection
- FoxO signaling pathway
- Gastric cancer
- Hepatitis B
- Hepatitis C
- Human T-cell leukemia virus 1 infection
- Human papillomavirus infection
- Measles
- Oocyte meiosis
- PI3K-Akt signaling pathway
- Pathways in cancer
- Progesterone-mediated oocyte maturation
- Prostate cancer
- Small cell lung cancer
- Viral carcinogenesis
- p53 signaling pathway
Active Molecules (5,432)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XLZHLULRODUOPS
|
6.5 | IC50 | 5 | — | |
XUCUUZVZPFEPFA
|
6.5 | IC50 | 3 | — | |
ZAVTUNDLFXKBOM
|
6.5 | IC50 | 3 | — | |
ANAAVHLLZPPWCU
|
6.5 | IC50 | 6 | — | |
GOXVDXLRXMYVPC
|
6.5 | IC50 | 2 | — | |
GSYUZRLLPWNNAL
|
6.5 | IC50 | 6 | — | |
JNZTWAOEOYBNNP
|
6.5 | IC50 | 5 | — | |
MADUTGUALSLNOW
|
6.5 | IC50 | 4 | — | |
NJPIZAROFOGVAA
|
6.5 | IC50 | 3 | — | |
NQVNNPOALMGCQC
|
6.5 | IC50 | 3 | — | |
QLQYWGHSSLXLOS
|
6.5 | IC50 | 5 | — | |
QLTMJJAAHXGJMD
|
6.5 | Ki | 10 | — | |
URDPTNPMRNZRHJ
|
6.5 | IC50 | 5 | — | |
ZWWTZNLYKPWLQS
|
6.5 | IC50 | 2 | — | |
BTSZMJKDZCBEGX
|
6.4 | pIC50 | 5 | Yes | |
DGKDQGNOYZSJDK
|
6.4 | IC50 | 2 | — | |
FTMBNJPJFUAMIW
|
6.4 | IC50 | 4 | — | |
GKWZHZVUJVOVJN
|
6.4 | pIC50 | 2 | Yes | |
HGEJNHUGVPFHIF
|
6.4 | Kd | 3 | — | |
IVKYJVDFJKEXIH
|
6.4 | IC50 | 6 | — | |
JYWSISJKMHOMBG
|
6.4 | IC50 | 3 | — | |
LVNMUXRXRACMFH
|
6.4 | IC50 | 3 | — | |
LWYOYMDGSBDNLO
|
6.4 | IC50 | 3 | — | |
LYDJRRHXAUQPTD
|
6.4 | IC50 | 2 | — | |
MYUXGKKMSXZYMX
|
6.4 | IC50 | 2 | — | |
PWTPFCZIUPMVTG
|
6.4 | IC50 | 5 | — | |
QRXPIPWIGBYIFY
|
6.4 | pIC50 | 2 | Yes | |
QTBZFGYORPEJEV
|
6.4 | IC50 | 3 | — | |
RJPUDBUEIKLQCU
|
6.4 | IC50 | 2 | — | |
UIUYDZQKYIIPIT
|
6.4 | pIC50 | 2 | Yes | |
VILFMZCEQNTADR
|
6.4 | IC50 | 2 | — | |
WUFVFWHZRSJNAV
|
6.4 | pIC50 | 4 | Yes | |
WVSIOWNEXQMNSF
|
6.4 | IC50 | 6 | — | |
YGGYBJSDWZSAAU
|
6.4 | IC50 | 5 | — | |
ZQAZHQLWCKQXTD
|
6.4 | pIC50 | 2 | Yes | |
ZTSRCWHLXVMIPQ
|
6.4 | IC50 | 3 | — | |
BBUVDDPUURMFOX
|
6.4 | IC50 | 4 | — | |
CFBXWHPXNROFFK
|
6.4 | IC50 | 4 | — | |
CGECJCJUHCZZGO
|
6.4 | IC50 | 9 | — | |
FPGLJBDFRLADTG
|
6.4 | Ki | 2 | — | |
GWRVGNYOXQHPMF
|
6.4 | Ki | 5 | — | |
HCPRSMOENBWIIA
|
6.4 | IC50 | 3 | — | |
JRZGFHZNTXYGPL
|
6.4 | pIC50 | 3 | Yes | |
KPUBBCGAMBGWSV
|
6.4 | pIC50 | 2 | Yes | |
LAQCQSKKZIRXFW
|
6.4 | IC50 | 9 | — | |
QQOSANNDIZSJOV
|
6.4 | IC50 | 2 | — | |
UQAHWAQRLXARGK
|
6.4 | IC50 | 3 | — | |
UVVGSZJKQAELIC
|
6.4 | IC50 | 4 | — | |
VKUXBRRQHBTQPW
|
6.4 | IC50 | 3 | — | |
XVRFIUSGDOJQMI
|
6.4 | IC50 | 3 | — |