Target Details
| UniProt AC | P24928 |
|---|---|
| Gene Symbol | POLR2A |
| Protein Name | DNA-directed RNA polymerase II subunit RPB1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF04997 (RNA_pol_Rpb1_1) PF00623 (RNA_pol_Rpb1_2) PF04983 (RNA_pol_Rpb1_3) PF05000 (RNA_pol_Rpb1_4) PF04998 (RNA_pol_Rpb1_5) PF04992 (RNA_pol_Rpb1_6) PF04990 (RNA_pol_Rpb1_7) PF05001 (RNA_pol_Rpb1_R) |
Summary
- Multi-target molecules 1
- Clinical molecules 0
- Avg pChEMBL 6.81
KEGG Pathways (3)
Associated Diseases (1)
Active Molecules (1)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AAAQFGUYHFJNHI
|
6.8 | IC50 | 252 | — |