Target Details
| UniProt AC | P24723 |
|---|---|
| Gene Symbol | PRKCH |
| Protein Name | Protein kinase C eta type |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF00168 (C2) PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 348
- Clinical molecules 144
- Avg pChEMBL 7.36
KEGG Pathways (2)
Active Molecules (348)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AQGHYUYFBXMRBC
|
7.8 | IC50 | 6 | — | |
FXGHOAZJQNLNFD
|
7.8 | IC50 | 13 | Yes | |
DVMQYKHCZLPSAP
|
7.7 | IC50 | 5 | — | |
UHIFMIXIMAHXIB
|
7.7 | IC50 | 6 | — | |
AZIMEXGKUWHPQV
|
7.7 | IC50 | 12 | Yes | |
CKJRKRPDNLRZPQ
|
7.7 | IC50 | 6 | — | |
CKJRKRPDNLRZPQ
|
7.7 | IC50 | 7 | — | |
FSBMWCWKNXQVMP
|
7.7 | IC50 | 12 | Yes | |
GQCWIZZVARXZGR
|
7.7 | IC50 | 6 | — | |
GQCWIZZVARXZGR
|
7.7 | IC50 | 6 | — | |
MKPSMRQVGPTYRL
|
7.7 | IC50 | 5 | — | |
MKPSMRQVGPTYRL
|
7.7 | IC50 | 6 | — | |
OWLWQUHZHTVSAN
|
7.7 | IC50 | 6 | — | |
PQWWKDOKHDWZBH
|
7.7 | IC50 | 6 | — | |
TXVBBLNFLUZGIT
|
7.7 | IC50 | 6 | — | |
ULGQQNXZFKHRIL
|
7.7 | IC50 | 3 | — | |
USEYXZSHZLLAJS
|
7.7 | IC50 | 6 | — | |
XYUFCXJZFZPEJD
|
7.7 | IC50 | 9 | — | |
XYUFCXJZFZPEJD
|
7.7 | IC50 | 23 | Yes | |
YUKJJLKBBAFYNN
|
7.7 | IC50 | 12 | Yes | |
ZOGSVRRXRLSQNC
|
7.7 | IC50 | 6 | — | |
RVIJQMOQZFCSHL
|
7.7 | Ki | 8 | Yes | |
XYUFCXJZFZPEJD
|
7.7 | IC50 | 6 | — | |
RSTWARDIGORXQU
|
7.6 | Ki | 7 | Yes | |
IDSZLHFEKAUIOL
|
7.6 | IC50 | 7 | Yes | |
MVPSDKPPZLPMBB
|
7.6 | Ki | 7 | Yes | |
QJVMNACFDUTHPM
|
7.6 | IC50 | 6 | — | |
MGQDMSJZRRHMFT
|
7.6 | IC50 | 6 | — | |
JHLONFVVTLRHIZ
|
7.6 | IC50 | 4 | — | |
KPCVAMMFCPIUIU
|
7.5 | IC50 | 12 | Yes | |
CEMBEUHBOHDWPN
|
7.5 | IC50 | 4 | — | |
CYRPAUWSHGGREB
|
7.5 | Ki | 8 | Yes | |
JOOTZGPUMCZHLH
|
7.5 | IC50 | 5 | — | |
OQICVMYHDNIADM
|
7.5 | IC50 | 6 | — | |
OVJZHEDXGAPGDA
|
7.5 | IC50 | 5 | — | |
XXDWSQPJTJZKSJ
|
7.5 | IC50 | 12 | Yes | |
ZZSBPGIGIUFJRA
|
7.5 | IC50 | 15 | Yes | |
FELQRVDTGNDOSI
|
7.5 | IC50 | 15 | Yes | |
ZEYTZKVCOZMUKL
|
7.5 | IC50 | 5 | — | |
MYOUXQLHWTWXON
|
7.5 | IC50 | 16 | Yes | |
DZIUPOCVDSYPSY
|
7.5 | IC50 | 8 | Yes | |
YDZJEODKNRAYMA
|
7.5 | IC50 | 12 | Yes | |
AJFLRCLZEMUXCH
|
7.5 | IC50 | 4 | — | |
ZMHXVAQNZDUNOG
|
7.5 | IC50 | 6 | — | |
ZYUGNHPOVKADFZ
|
7.5 | IC50 | 11 | — | |
HPBJQOWLAKYNDM
|
7.4 | IC50 | 15 | Yes | |
QMYFYCSCELQGHP
|
7.4 | IC50 | 7 | Yes | |
MVQGUYKZTHVOEH
|
7.4 | Ki | 8 | Yes | |
OSVUGUHRKMMBSE
|
7.4 | Kd | 170 | — | |
AMSOPBXQXSAAAC
|
7.4 | IC50 | 12 | Yes |