Target Details
| UniProt AC | P24723 |
|---|---|
| Gene Symbol | PRKCH |
| Protein Name | Protein kinase C eta type |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF00168 (C2) PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 348
- Clinical molecules 144
- Avg pChEMBL 7.36
KEGG Pathways (2)
Active Molecules (348)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WTXAWDOYPWWUJL
|
10.1 | IC50 | 11 | — | |
REAZZDPREXHWNV
|
10.0 | Ki | 7 | — | |
SSXCVTWCXHGTLK
|
9.9 | IC50 | 11 | — | |
KTGVSZYYHHRRGW
|
9.8 | IC50 | 11 | — | |
VIESIZQAHOPEBR
|
9.8 | IC50 | 11 | — | |
NVYBXIDWOJVGQI
|
9.8 | IC50 | 11 | — | |
APVOCXHEVZBCGS
|
9.7 | IC50 | 11 | — | |
XSJFPSCYMJFDNI
|
9.7 | Ki | 7 | — | |
DHTLXMRCLSUJPP
|
9.7 | IC50 | 11 | — | |
DASVAQCTVIQROX
|
9.5 | Ki | 8 | Yes | |
RHJPBGWFGOAEID
|
9.4 | Ki | 8 | Yes | |
VVRRZOFLLJAMIK
|
9.4 | IC50 | 11 | — | |
SWKUTOXEFLDOID
|
9.3 | Ki | 7 | — | |
IRGJDPZJEUYSKS
|
9.2 | IC50 | 7 | — | |
IRGJDPZJEUYSKS
|
9.2 | IC50 | 9 | — | |
IRGJDPZJEUYSKS
|
9.2 | IC50 | 6 | — | |
BQJRUJTZSGYBEZ
|
9.1 | Kd | 13 | Yes | |
IRGJDPZJEUYSKS
|
9.0 | IC50 | 9 | — | |
WAKGEHXTOOFEAE
|
9.0 | IC50 | 27 | — | |
FANQQVWXAKUWNI
|
8.8 | IC50 | 6 | — | |
NVSJOASGKCGXBZ
|
8.8 | IC50 | 16 | Yes | |
UZCZCOMLMMSRLY
|
8.7 | IC50 | 6 | — | |
CKJRKRPDNLRZPQ
|
8.7 | IC50 | 6 | — | |
CKJRKRPDNLRZPQ
|
8.7 | IC50 | 7 | — | |
FCVHMDURXUOCFY
|
8.7 | IC50 | 6 | — | |
QYBVZIIWBRIXMX
|
8.7 | IC50 | 12 | Yes | |
YUJAAMQBNNAQRP
|
8.7 | IC50 | 6 | — | |
JZLFYMHIISZQCZ
|
8.7 | IC50 | 12 | Yes | |
QZCYXWFWSDBJGL
|
8.6 | Ki | 8 | Yes | |
HEZSSKBBLQBTMF
|
8.6 | Ki | 4 | — | |
KGPGFQWBCSZGEL
|
8.6 | Kd | 59 | Yes | |
BPNNZZBLGSVSAA
|
8.5 | IC50 | 6 | — | |
BPNNZZBLGSVSAA
|
8.5 | IC50 | 7 | — | |
BPNNZZBLGSVSAA
|
8.5 | IC50 | 6 | — | |
BPNNZZBLGSVSAA
|
8.5 | IC50 | 7 | — | |
FCVHMDURXUOCFY
|
8.5 | IC50 | 7 | — | |
OWJIKBAZUBPKGN
|
8.5 | IC50 | 6 | — | |
OWJIKBAZUBPKGN
|
8.5 | IC50 | 7 | — | |
STEGBXHZVWLLAP
|
8.5 | IC50 | 6 | — | |
WOFBHAKTZOZODW
|
8.5 | IC50 | 6 | — | |
URLJNGHIJZMXTK
|
8.5 | IC50 | 6 | — | |
HXWARSZQGAFXJM
|
8.5 | Ki | 7 | — | |
FWEDWNSLCBHVQT
|
8.4 | IC50 | 5 | — | |
IVGCXWIFBNPPBW
|
8.4 | IC50 | 6 | — | |
OWJIKBAZUBPKGN
|
8.4 | IC50 | 6 | — | |
OWJIKBAZUBPKGN
|
8.4 | IC50 | 7 | — | |
VLUGUCDUHZVABE
|
8.4 | IC50 | 6 | — | |
YIZRPXUMLQCIMQ
|
8.4 | IC50 | 9 | — | |
YIZRPXUMLQCIMQ
|
8.4 | IC50 | 7 | — | |
YIZRPXUMLQCIMQ
|
8.4 | IC50 | 9 | — |