Target Details
| UniProt AC | P24557 |
|---|---|
| Gene Symbol | TBXAS1 |
| Protein Name | Thromboxane-A synthase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00067 (p450) |
Summary
- Multi-target molecules 191
- Clinical molecules 8
- Avg pChEMBL 7.38
KEGG Pathways (3)
Associated Diseases (1)
Active Molecules (191)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UICLKHCKXGFMBB
|
6.6 | IC50 | 2 | — | |
VICNFVKMEAIXSQ
|
6.6 | IC50 | 2 | — | |
XYEOSUOFNKZBKV
|
6.6 | IC50 | 2 | — | |
XYEOSUOFNKZBKV
|
6.6 | IC50 | 2 | — | |
YERVHMNPCKNRIB
|
6.6 | IC50 | 2 | — | |
BYBLEWFAAKGYCD
|
6.6 | IC50 | 16 | Yes | |
DJMSMHXCSIBVSA
|
6.5 | IC50 | 2 | — | |
AYMZVORQEONTPY
|
6.5 | IC50 | 2 | — | |
DTNBASHNJVNKBM
|
6.5 | IC50 | 2 | — | |
MMDSGIVIWHELNX
|
6.5 | IC50 | 2 | — | |
YKMLNPDQLWRQKS
|
6.5 | IC50 | 2 | — | |
YKMLNPDQLWRQKS
|
6.5 | IC50 | 2 | — | |
IMMNAXXZSBKGMT
|
6.4 | IC50 | 2 | — | |
IMMNAXXZSBKGMT
|
6.4 | IC50 | 2 | — | |
JVPRGMUQAFLVBU
|
6.4 | IC50 | 2 | — | |
PVQYCYOIOKLQMP
|
6.4 | IC50 | 2 | — | |
PVQYCYOIOKLQMP
|
6.4 | IC50 | 2 | — | |
VKYMAXGZPKUBLB
|
6.4 | IC50 | 2 | — | |
TXKRKUVUYCOYKP
|
6.4 | IC50 | 2 | — | |
TXKRKUVUYCOYKP
|
6.4 | IC50 | 2 | — | |
IUIKKXJIHSJKKO
|
6.3 | Kd | 2 | — | |
CDMGBJANTYXAIV
|
6.3 | IC50 | 34 | Yes | |
COOJSXJHFBIVLU
|
6.3 | IC50 | 2 | — | |
LGHLGTHRJNIRCA
|
6.3 | IC50 | 2 | — | |
ZHBPUNZHLIFKIH
|
6.3 | IC50 | 2 | — | |
MPGBYGNPFRLHAO
|
6.3 | IC50 | 2 | — | |
DOADCIRUVGSBTJ
|
6.2 | IC50 | 2 | — | |
KKKDZZRICRFGSD
|
6.2 | IC50 | 6 | — | |
QRJJEGAJXVEBNE
|
6.2 | IC50 | 9 | — | |
HCLFUHWPLXVRIS
|
6.2 | IC50 | 2 | — | |
VPDLANZEXFQJSQ
|
6.2 | IC50 | 2 | — | |
YKPJTNNQDJFQBF
|
6.2 | IC50 | 2 | — | |
JHKBLBMCCJQROB
|
6.2 | IC50 | 2 | — | |
XHYZCGGTDZPVPB
|
6.1 | IC50 | 2 | — | |
NZWWYUMFUATSTK
|
6.1 | IC50 | 3 | Yes | |
NKANXQFJJICGDU
|
6.0 | IC50 | 35 | Yes | |
JAANHRCZVHDEGF
|
6.0 | IC50 | 2 | — | |
JAANHRCZVHDEGF
|
6.0 | IC50 | 2 | — | |
DCNXKPFVMNEKDU
|
6.0 | IC50 | 2 | — | |
LJZXVXGFHZARCP
|
6.0 | IC50 | 2 | — | |
MVVKZSDUMIXCAZ
|
6.0 | IC50 | 2 | — |