Target Details
| UniProt AC | P24557 |
|---|---|
| Gene Symbol | TBXAS1 |
| Protein Name | Thromboxane-A synthase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00067 (p450) |
Summary
- Multi-target molecules 191
- Clinical molecules 8
- Avg pChEMBL 7.38
KEGG Pathways (3)
Associated Diseases (1)
Active Molecules (191)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CDEOOMRKYGZADT
|
7.4 | IC50 | 2 | — | |
FZZMVSWCYIOLSW
|
7.4 | IC50 | 2 | — | |
CHFCDPZHINDKME
|
7.4 | IC50 | 2 | — | |
UYIFEFLIAAUJOU
|
7.3 | IC50 | 2 | — | |
PTVHLCSHLNBWFT
|
7.3 | IC50 | 2 | — | |
JTCXJAJLGOTNRH
|
7.3 | IC50 | 2 | — | |
LACPPBQCKQXQIH
|
7.3 | IC50 | 2 | — | |
UTAFETDONDFNBQ
|
7.3 | IC50 | 2 | — | |
BXVLOKOSLGIICL
|
7.3 | IC50 | 2 | — | |
DJPVNHLABTYAMF
|
7.3 | IC50 | 2 | — | |
IDSQFTJASXFWNN
|
7.3 | IC50 | 2 | — | |
JEJFHDDECMACOD
|
7.3 | IC50 | 2 | — | |
MBFUMLZEULKFON
|
7.3 | IC50 | 2 | — | |
VWNGGSJYQAOKAV
|
7.3 | IC50 | 2 | — | |
WHSSOYNNHOWWJE
|
7.3 | IC50 | 2 | — | |
GUTGDFJEUBLDBQ
|
7.2 | IC50 | 2 | — | |
OCWOTYUFXGGBAW
|
7.2 | IC50 | 2 | — | |
FACJEJPQFUXMOA
|
7.2 | IC50 | 2 | — | |
JFHKOMDCQBVNHI
|
7.2 | IC50 | 2 | — | |
JMPFSEBWVLAJKM
|
7.2 | IC50 | 8 | Yes | |
NMJYFIAGWNELHF
|
7.2 | IC50 | 2 | — | |
NCDNCNXCDXHOMX
|
7.1 | IC50 | 12 | — | |
LTCQRNQPODCPAS
|
7.1 | IC50 | 2 | — | |
LTCQRNQPODCPAS
|
7.1 | IC50 | 2 | — | |
HQAGYVZFEKMBFE
|
7.0 | IC50 | 2 | — | |
AGAXMMPHPXHEAW
|
7.0 | IC50 | 2 | — | |
BBQILAZFNVDEMU
|
7.0 | IC50 | 2 | — | |
CGIGDMFJXJATDK
|
7.0 | IC50 | 11 | Yes | |
CPHBHPJSMLOFHV
|
7.0 | IC50 | 2 | — | |
IIXGCBPDCHNSLC
|
7.0 | IC50 | 2 | — | |
LQUYEBKTHLMNKY
|
7.0 | IC50 | 2 | — | |
MIIIWVNAZRSKJI
|
7.0 | IC50 | 2 | — | |
OIMUMJMHBPPFFI
|
7.0 | IC50 | 2 | — | |
WDGUBDMXGCFGIL
|
7.0 | IC50 | 2 | — | |
WPBWMPUZDXLQIX
|
7.0 | IC50 | 2 | — | |
KMESAVNRPDKZCQ
|
6.9 | IC50 | 2 | — | |
HPJSHFVQFXNALY
|
6.8 | IC50 | 2 | — | |
NTKWRAAWKFNECW
|
6.8 | IC50 | 2 | — | |
ZNRZNAHHOIANAO
|
6.8 | IC50 | 2 | — | |
AFNXATANNDIXLG
|
6.7 | IC50 | 11 | — | |
HTEXFAJUBRSJDG
|
6.7 | IC50 | 2 | — | |
HTEXFAJUBRSJDG
|
6.7 | IC50 | 2 | — | |
KTUFNOKKBVMGRW
|
6.7 | IC50 | 38 | Yes | |
LKFAYNBLUNPUHN
|
6.7 | IC50 | 2 | — | |
OYMNICOOAXOYPP
|
6.7 | IC50 | 2 | — | |
PUECHKOKBSMEOQ
|
6.7 | IC50 | 2 | — | |
RUAOGLCGDIBHJR
|
6.7 | IC50 | 2 | — | |
WSFCJPZVQFMTRY
|
6.7 | IC50 | 2 | — | |
FNTPEBIGZTYDQK
|
6.7 | IC50 | 2 | — | |
AKUSUAZJHUIURR
|
6.6 | IC50 | 2 | — |