Target Details
| UniProt AC | P24557 |
|---|---|
| Gene Symbol | TBXAS1 |
| Protein Name | Thromboxane-A synthase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00067 (p450) |
Summary
- Multi-target molecules 191
- Clinical molecules 8
- Avg pChEMBL 7.38
KEGG Pathways (3)
Associated Diseases (1)
Active Molecules (191)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VDSYMHSEFRKHET
|
7.9 | IC50 | 2 | — | |
SHRNOBNPOTZEAM
|
7.9 | IC50 | 2 | — | |
VNFPBHJOKIVQEB
|
7.8 | IC50 | 20 | Yes | |
RERMKDAOFJRCJU
|
7.8 | IC50 | 2 | — | |
AEMOPCLSCUUOFI
|
7.7 | IC50 | 2 | — | |
LMSWDFLNAYPJJD
|
7.7 | IC50 | 2 | — | |
SOUOKSHPPGIZRL
|
7.7 | IC50 | 2 | — | |
VGBBXLWOWUXXFE
|
7.7 | IC50 | 2 | — | |
DGYJMRJVVGLCDV
|
7.7 | IC50 | 2 | — | |
DKVCJHBRBBPIGM
|
7.7 | IC50 | 2 | — | |
QNSOXESEHPFNCD
|
7.7 | IC50 | 2 | — | |
CDTZYZWEPCKHSB
|
7.7 | IC50 | 2 | — | |
LQZKCALSANZAMX
|
7.7 | IC50 | 2 | — | |
LQZKCALSANZAMX
|
7.7 | IC50 | 2 | — | |
NMJYFIAGWNELHF
|
7.7 | IC50 | 2 | — | |
RGGXEZXJJJANGJ
|
7.7 | IC50 | 2 | — | |
RGGXEZXJJJANGJ
|
7.7 | IC50 | 2 | — | |
LMSWDFLNAYPJJD
|
7.6 | IC50 | 2 | — | |
BHULVFAMAJBLNZ
|
7.6 | IC50 | 2 | — | |
NUPJOHLAKYWZHZ
|
7.6 | IC50 | 2 | — | |
QOIVFTOIMRANMQ
|
7.6 | IC50 | 2 | — | |
QOIVFTOIMRANMQ
|
7.6 | IC50 | 2 | — | |
GZYRADOPCAPBPA
|
7.6 | IC50 | 2 | — | |
ATTDTTWNDPANQN
|
7.6 | IC50 | 2 | — | |
JEILTEAKGWGOSO
|
7.6 | IC50 | 2 | — | |
JEILTEAKGWGOSO
|
7.6 | IC50 | 2 | — | |
SWLNUQSMWKYMJE
|
7.6 | IC50 | 2 | — | |
SWLNUQSMWKYMJE
|
7.6 | IC50 | 2 | — | |
WSGAKKPWXZPETA
|
7.6 | IC50 | 2 | — | |
UEBOELMCZQDCEI
|
7.6 | IC50 | 2 | — | |
UEBOELMCZQDCEI
|
7.6 | IC50 | 2 | — | |
CNJDBFHUIFFSQK
|
7.6 | IC50 | 2 | — | |
IONAQTGMWFXHIX
|
7.5 | IC50 | 3 | — | |
LEZWWPYKPKIXLL
|
7.5 | IC50 | 20 | — | |
UASKRIFPIWYGAQ
|
7.5 | IC50 | 2 | — | |
PMZRHVZFESEBFJ
|
7.5 | IC50 | 2 | — | |
RXLLZZVKOZGWDX
|
7.5 | IC50 | 2 | — | |
JILQVWNDRFJPRF
|
7.5 | IC50 | 2 | — | |
NMJYFIAGWNELHF
|
7.5 | IC50 | 2 | — | |
PJZSRUKFPMOTFE
|
7.5 | IC50 | 2 | — | |
POPJWIHAKVJLHO
|
7.5 | IC50 | 2 | — | |
AERMYTSNNRHMDS
|
7.5 | IC50 | 2 | — | |
XJKMOZFCIYEDDT
|
7.5 | IC50 | 2 | — | |
AQQCPDIIPNDMEK
|
7.5 | IC50 | 2 | — | |
WMXZEBHSAJEWND
|
7.4 | IC50 | 2 | — | |
FMGMZPGNRHRJQC
|
7.4 | IC50 | 2 | — | |
NEJDMJAJYOXVJF
|
7.4 | IC50 | 2 | — | |
HEMGORMJZTVDGN
|
7.4 | IC50 | 2 | — | |
WHLKEJMJCAGFRW
|
7.4 | IC50 | 2 | — | |
AVFPODQCTNAKHD
|
7.4 | IC50 | 2 | — |