Target Details
| UniProt AC | P24530 |
|---|---|
| Gene Symbol | EDNRB |
| Protein Name | Endothelin receptor type B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 507
- Clinical molecules 0
- Avg pChEMBL 7.11
KEGG Pathways (6)
Associated Diseases (4)
Active Molecules (507)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OTPDSJIKVVZMFC
|
6.3 | IC50 | 2 | — | |
ZQMGLMDAJMDRHF
|
6.3 | IC50 | 2 | — | |
HLYUXTAHAPGOGF
|
6.3 | IC50 | 2 | — | |
KAAWXPGZQHJMQL
|
6.3 | IC50 | 2 | — | |
VIVHYWNEMYNSTR
|
6.3 | IC50 | 2 | — | |
XPPNYNZMOQSBAA
|
6.3 | Ki | 2 | — | |
YPXSZXRASAVIKK
|
6.3 | IC50 | 2 | — | |
DKRMKDLKTIKQIE
|
6.2 | IC50 | 2 | — | |
FWIARXJRYJCABB
|
6.2 | IC50 | 2 | — | |
JKNAAXSOIGHTLX
|
6.2 | IC50 | 2 | — | |
KSWCYNIYGNMXLW
|
6.2 | IC50 | 2 | — | |
QLOACGMSZNOMDZ
|
6.2 | IC50 | 2 | — | |
SDXSGUVLSFVWRF
|
6.2 | IC50 | 2 | — | |
AIVZWVQMNJFOIL
|
6.2 | IC50 | 2 | — | |
AQDCZLZCKZWUCZ
|
6.2 | IC50 | 2 | — | |
IDINHRPVYGDPHV
|
6.2 | IC50 | 2 | — | |
KMOYVJSVLLXFQU
|
6.2 | Ki | 2 | — | |
RPBOIJRVAJKCSF
|
6.2 | IC50 | 2 | — | |
YCDUZUIVJLJHQL
|
6.2 | IC50 | 2 | — | |
CKAWNKDSMUUPOR
|
6.2 | IC50 | 2 | — | |
HAHANBGRLRTDGL
|
6.2 | Ki | 2 | — | |
YOMSYVFQYBPECD
|
6.2 | IC50 | 2 | — | |
DYHGVCADLVCJGZ
|
6.2 | IC50 | 2 | — | |
HOPRHFCRDCRJAB
|
6.2 | IC50 | 2 | — | |
IECXSVOMLVKXGN
|
6.2 | IC50 | 2 | — | |
YBWLTKFZAOSWSM
|
6.2 | IC50 | 2 | — | |
ZDGQZBNPWPRKMF
|
6.2 | IC50 | 2 | — | |
IUTFNAAZZLIBQX
|
6.2 | IC50 | 2 | — | |
SCOBRKBPUKEATJ
|
6.2 | IC50 | 2 | — | |
VXJUFLPIZFIKQL
|
6.2 | IC50 | 2 | — | |
CTANMDRPZQDKDO
|
6.2 | IC50 | 2 | — | |
FZNWHURKGWXPCC
|
6.2 | IC50 | 2 | — | |
QXJMSZDXBBMLGU
|
6.2 | Ki | 2 | — | |
RXNZJEAMURXNLG
|
6.2 | IC50 | 2 | — | |
MIPNODJPKTVQHX
|
6.2 | IC50 | 2 | — | |
PQJLYRULHJYQDW
|
6.2 | IC50 | 2 | — | |
TVTJICVMTXUAKS
|
6.2 | IC50 | 2 | — | |
PGAMLYVKCIXYNX
|
6.2 | IC50 | 2 | — | |
PGDSQHCYBSJOHQ
|
6.2 | IC50 | 2 | — | |
WAOUMQDGIOSVAF
|
6.2 | IC50 | 2 | — | |
GINOPQFPTRYBHX
|
6.2 | IC50 | 2 | — | |
NIGCNIFGPYTDPJ
|
6.2 | IC50 | 2 | — | |
QRKZNZMLWQPCPE
|
6.2 | IC50 | 2 | — | |
UZLLGNWABVRSKB
|
6.2 | IC50 | 2 | — | |
ADKWUFCPMCLUKI
|
6.2 | IC50 | 2 | — | |
ASYDIUHFIWWNJR
|
6.2 | IC50 | 2 | — | |
JGCMJLQTOLPTCY
|
6.2 | IC50 | 2 | — | |
OZRQEMUTNMRJTM
|
6.1 | IC50 | 2 | — | |
HMDVOILXHRHOGL
|
6.1 | IC50 | 2 | — | |
NVONIBWWXNXALH
|
6.1 | IC50 | 2 | — |