Target Details
| UniProt AC | P24530 |
|---|---|
| Gene Symbol | EDNRB |
| Protein Name | Endothelin receptor type B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 507
- Clinical molecules 0
- Avg pChEMBL 7.11
KEGG Pathways (6)
Associated Diseases (4)
Active Molecules (507)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VUAQGALNRBYHNG
|
6.5 | IC50 | 2 | — | |
YNKZURRWQXRKDP
|
6.5 | IC50 | 2 | — | |
IISLJISTBMPEAA
|
6.5 | IC50 | 2 | — | |
VAXUKYCSAUELNZ
|
6.5 | IC50 | 2 | — | |
KWXXXHXCVVFIMQ
|
6.5 | Ki | 2 | — | |
NEOVBIIJKPUROI
|
6.5 | Ki | 2 | — | |
RXNZJEAMURXNLG
|
6.5 | IC50 | 2 | — | |
FPJPMEXULUCUCB
|
6.4 | Ki | 2 | — | |
HTNBCWLAXCOARB
|
6.4 | IC50 | 2 | — | |
FEJVSJIALLTFRP
|
6.4 | Ki | 2 | — | |
GMNFTSXERCOCMB
|
6.4 | IC50 | 2 | — | |
MHNJEAOUFUNYKE
|
6.4 | IC50 | 2 | — | |
TWNPZFARHUKPBV
|
6.4 | Ki | 2 | — | |
JGCMEBMXRHSZKX
|
6.4 | IC50 | 3 | — | |
JPRDUKLJMTUKCJ
|
6.4 | IC50 | 2 | — | |
SGMHXYMWOLAIMX
|
6.4 | IC50 | 2 | — | |
AEDZVHIKLJEHDR
|
6.4 | IC50 | 2 | — | |
GWBCKOWLDKFIHO
|
6.4 | IC50 | 2 | — | |
UEHPBBFVUYURNP
|
6.4 | IC50 | 2 | — | |
AIJJGHXRGHAKEG
|
6.4 | IC50 | 2 | — | |
JDIFCWUHBJXZLK
|
6.4 | IC50 | 2 | — | |
KRTXDXIJWFIGGJ
|
6.4 | IC50 | 2 | — | |
MRISGPUEHMXCRJ
|
6.4 | IC50 | 2 | — | |
TWBVBLFAEWNYQQ
|
6.4 | IC50 | 2 | — | |
VACPWIZSMORWDJ
|
6.4 | IC50 | 2 | — | |
CFOMGVYXSNFELK
|
6.4 | IC50 | 2 | — | |
BIHSQJMJRJBBHK
|
6.4 | IC50 | 2 | — | |
GKCAKABSOVLWHG
|
6.4 | IC50 | 2 | — | |
JGEXEIBPRHWMSL
|
6.3 | IC50 | 2 | — | |
NRCLKFNYCQXXAL
|
6.3 | IC50 | 2 | — | |
SCMXLDCMGHKGGU
|
6.3 | IC50 | 2 | — | |
CMPCSJBKUBWQGQ
|
6.3 | IC50 | 2 | — | |
RJXHHVXIVAHBHS
|
6.3 | IC50 | 2 | — | |
UGJAKYVVBJWFEZ
|
6.3 | IC50 | 2 | — | |
UJPMGYUNKDMJEA
|
6.3 | IC50 | 2 | — | |
VIQIKJNRAFJKTQ
|
6.3 | IC50 | 2 | — | |
WBTXDANWVHPDGU
|
6.3 | IC50 | 2 | — | |
IGKCOJUPPUGBIE
|
6.3 | IC50 | 2 | — | |
WSNWXTKIOPWVDW
|
6.3 | IC50 | 2 | — | |
XYZWCNYWABHTRK
|
6.3 | IC50 | 2 | — | |
BJSXTKDRYZUWEL
|
6.3 | Ki | 2 | — | |
HEGRKFSINVTUKI
|
6.3 | IC50 | 2 | — | |
PWIPORDFWDZCJG
|
6.3 | IC50 | 2 | — | |
PYNCHZOAMKYGTR
|
6.3 | IC50 | 2 | — | |
MCHCGWZNXSZKJY
|
6.3 | Ki | 2 | — | |
RULBFQDDCRBSBY
|
6.3 | IC50 | 2 | — | |
IDRSXRPOEONBKT
|
6.3 | IC50 | 2 | — | |
LSQXFROVPNDBMN
|
6.3 | IC50 | 2 | — | |
QZLAMPMKCJHEKL
|
6.3 | IC50 | 2 | — | |
GBYVJKRBUNPVLB
|
6.3 | IC50 | 2 | — |