Target Details
| UniProt AC | P24530 |
|---|---|
| Gene Symbol | EDNRB |
| Protein Name | Endothelin receptor type B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 507
- Clinical molecules 0
- Avg pChEMBL 7.11
KEGG Pathways (6)
Associated Diseases (4)
Active Molecules (507)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JGAUQCSCABMOTB
|
6.7 | IC50 | 2 | — | |
SIPPOBLYWAIKGU
|
6.7 | IC50 | 2 | — | |
BSMQWDCPKODFQI
|
6.7 | IC50 | 2 | — | |
FYDHNMUVDRWWCO
|
6.7 | IC50 | 2 | — | |
HRAQSWKGRRUBDJ
|
6.7 | IC50 | 2 | — | |
IBNKZYKCCCSKLB
|
6.7 | IC50 | 2 | — | |
UJGUMHQLVYROSG
|
6.7 | IC50 | 2 | — | |
XJSUBSFOTRRUES
|
6.7 | IC50 | 2 | — | |
ZWTAXWXITAZUQP
|
6.7 | IC50 | 2 | — | |
DEOGRJUDPLWPSR
|
6.7 | IC50 | 2 | — | |
ZXXCWRYARSIMPM
|
6.7 | Ki | 2 | — | |
BEGQGXHBEYDHFL
|
6.7 | IC50 | 2 | — | |
FDVBFLHJYUCEKU
|
6.7 | IC50 | 2 | — | |
ZLSUWQHIYSFEQP
|
6.7 | IC50 | 2 | — | |
SXEVCCXWQGAXSQ
|
6.7 | IC50 | 2 | — | |
NNGHGYQUGDQKJY
|
6.6 | IC50 | 2 | — | |
QWDHLTWAAVZDIR
|
6.6 | Ki | 2 | — | |
RBIUYHJGRUEIPU
|
6.6 | IC50 | 2 | — | |
WYPXYGWFNRNTHH
|
6.6 | IC50 | 2 | — | |
SWIPVSPLUXWKTL
|
6.6 | IC50 | 2 | — | |
BYCLKBXHEZQIHD
|
6.6 | IC50 | 2 | — | |
FQXLGGFHDJJJJO
|
6.6 | IC50 | 2 | — | |
SQHRONMOLLICCQ
|
6.6 | IC50 | 2 | — | |
UTGRGVUJLJJKSH
|
6.6 | IC50 | 2 | — | |
WUYGPPAFDHJCRQ
|
6.6 | IC50 | 2 | — | |
XUMJJSAQQCTKAO
|
6.6 | IC50 | 3 | — | |
PGAMLYVKCIXYNX
|
6.6 | IC50 | 2 | — | |
BYBPPGGQNVVISN
|
6.6 | IC50 | 2 | — | |
XMLFZKYJSPXNGH
|
6.6 | IC50 | 2 | — | |
QSFFFSPNGBKTGJ
|
6.6 | IC50 | 2 | — | |
ABTJDYUDDLHWCG
|
6.6 | IC50 | 2 | — | |
AVUMTAXWDOUGCR
|
6.6 | IC50 | 2 | — | |
YJGADOCQUFXVMH
|
6.6 | IC50 | 2 | — | |
XPBBDUYWSIZCNR
|
6.6 | Ki | 2 | — | |
AAQHGXPJHYKNDF
|
6.5 | IC50 | 2 | — | |
NQDCDWVUSPOECA
|
6.5 | IC50 | 2 | — | |
KSGHGYRWLMKYNA
|
6.5 | IC50 | 2 | — | |
XNGPPJRUZXMHOV
|
6.5 | IC50 | 2 | — | |
XSSAXXJNGRXQCR
|
6.5 | IC50 | 2 | — | |
YLJHCAFDKWQJPI
|
6.5 | IC50 | 2 | — | |
BUZZXSDSIRQVKH
|
6.5 | IC50 | 2 | — | |
KZSPAFPPOAOZPK
|
6.5 | IC50 | 2 | — | |
NWZLYDCUPZYBAX
|
6.5 | IC50 | 2 | — | |
AOOKNPITEDSSNB
|
6.5 | Ki | 2 | — | |
BOZMVLDNYMRJIR
|
6.5 | IC50 | 2 | — | |
TYLZGSIGPRVNQJ
|
6.5 | IC50 | 2 | — | |
LNPRLVTXUXFAEN
|
6.5 | Ki | 2 | — | |
OGTVYDGVOOLHDI
|
6.5 | IC50 | 2 | — | |
ZHXNJGISXVIIND
|
6.5 | Ki | 2 | — | |
CHLXSJALJVYDID
|
6.5 | IC50 | 2 | — |