Target Details
| UniProt AC | P24530 |
|---|---|
| Gene Symbol | EDNRB |
| Protein Name | Endothelin receptor type B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 507
- Clinical molecules 0
- Avg pChEMBL 7.11
KEGG Pathways (6)
Associated Diseases (4)
Active Molecules (507)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MOTJMGVDPWRKOC
|
6.9 | IC50 | 2 | — | |
BZSLFEJGVQKVKX
|
6.9 | IC50 | 2 | — | |
GAZYTXSFOKMUAC
|
6.9 | IC50 | 2 | — | |
NDGMTIKKHLLDIV
|
6.9 | IC50 | 2 | — | |
NNLKMQXTQXTMET
|
6.9 | IC50 | 2 | — | |
DNIIBGYNGASUDE
|
6.9 | IC50 | 2 | — | |
MRZPJCAABGPJED
|
6.9 | IC50 | 2 | — | |
TWGYPFLCDZVWJV
|
6.9 | IC50 | 2 | — | |
HAHANBGRLRTDGL
|
6.9 | IC50 | 2 | — | |
KVMLOIHJNDCBKI
|
6.9 | IC50 | 2 | — | |
RIFDNBGSPYSLKK
|
6.9 | Ki | 2 | — | |
UIYNSXMUJGBENK
|
6.9 | IC50 | 2 | — | |
OFCTYBMKKTVKCR
|
6.9 | Ki | 2 | — | |
ILKUULNNGMUWFG
|
6.8 | IC50 | 2 | — | |
BTPMMVWQHRCMQR
|
6.8 | IC50 | 2 | — | |
XPOWMKNHKCJZNA
|
6.8 | IC50 | 2 | — | |
XPUJKHFCHQYTEQ
|
6.8 | IC50 | 2 | — | |
MNRPBSOBVCAVNX
|
6.8 | IC50 | 2 | — | |
HKMVKDPUVNFFAO
|
6.8 | Ki | 2 | — | |
ZMUVTNWMWOXWGB
|
6.8 | IC50 | 2 | — | |
BWMGPBPXTCNARL
|
6.8 | Ki | 2 | — | |
FAYAMAAFPRXGJT
|
6.8 | IC50 | 2 | — | |
KYDWTWOSIICWFQ
|
6.8 | Ki | 2 | — | |
PWHUJWODHSRAIM
|
6.8 | IC50 | 2 | — | |
ARFNEXZBRRNUKE
|
6.8 | IC50 | 2 | — | |
QYVHDIUYFHTCJX
|
6.8 | IC50 | 2 | — | |
FDDMPZZHBROSPE
|
6.8 | IC50 | 2 | — | |
OCZIRSIFHBBDKN
|
6.8 | Ki | 2 | — | |
QLKHVLXMFAFDAZ
|
6.8 | IC50 | 2 | — | |
YDIGUOCUKLHGNZ
|
6.8 | IC50 | 2 | — | |
LFWCJABOXHSRGC
|
6.8 | IC50 | 2 | — | |
FINMPMBYTTVLPJ
|
6.7 | IC50 | 2 | — | |
FVWWHXXCNJDXHS
|
6.7 | IC50 | 2 | — | |
GQTAIGFWINAVHA
|
6.7 | IC50 | 2 | — | |
HEEXATKNWQMTKJ
|
6.7 | IC50 | 2 | — | |
WITCSGJQNAEGBT
|
6.7 | IC50 | 2 | — | |
JOMWRKGBRATICM
|
6.7 | IC50 | 2 | — | |
SENIALTXHXJCNY
|
6.7 | IC50 | 2 | — | |
ZGXRPHUWXAFFDA
|
6.7 | IC50 | 2 | — | |
MOXPGMJEOXCNPF
|
6.7 | IC50 | 2 | — | |
OUJTZYPIHDYQMC
|
6.7 | IC50 | 2 | — | |
OUJTZYPIHDYQMC
|
6.7 | Ki | 2 | — | |
PIWOCJNYDKRQRS
|
6.7 | IC50 | 2 | — | |
VQUBCMKIGJZUME
|
6.7 | Ki | 2 | — | |
BATSJXIVNKJCKQ
|
6.7 | IC50 | 2 | — | |
DAZOXLCENQFWSQ
|
6.7 | IC50 | 2 | — | |
GJPICJJJRGTNOD
|
6.7 | IC50 | 2 | — | |
KNCYVPWSDRUANJ
|
6.7 | IC50 | 2 | — | |
VVOGFCYZFAKNMH
|
6.7 | IC50 | 2 | — | |
GADXZXTXFHEOKH
|
6.7 | IC50 | 2 | — |