Target Details
| UniProt AC | P24530 |
|---|---|
| Gene Symbol | EDNRB |
| Protein Name | Endothelin receptor type B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 507
- Clinical molecules 0
- Avg pChEMBL 7.11
KEGG Pathways (6)
Associated Diseases (4)
Active Molecules (507)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FJHPXCQTPSEFDQ
|
7.2 | IC50 | 2 | — | |
ICAHNKLYQDWFQQ
|
7.2 | IC50 | 2 | — | |
PYSZMARKHQLZJY
|
7.2 | IC50 | 2 | — | |
GBDHMDQPXDYBRO
|
7.2 | IC50 | 2 | — | |
KRSWVPASAJDUGK
|
7.2 | IC50 | 2 | — | |
MHZFPYMEACEGKL
|
7.2 | IC50 | 2 | — | |
TZPUDTSXRNOQNK
|
7.2 | Ki | 2 | — | |
XCDYCRJUBJSYLD
|
7.2 | IC50 | 2 | — | |
GEAANMFRDZRIIE
|
7.1 | IC50 | 2 | — | |
AAKCZJIYTMOXJF
|
7.1 | IC50 | 2 | — | |
KKGSEDUFHOPCFO
|
7.1 | IC50 | 2 | — | |
PUEQTWGTNQUURY
|
7.1 | IC50 | 2 | — | |
CBJKZXKXUSTFHL
|
7.1 | IC50 | 2 | — | |
FRQPGCPVRMZTNE
|
7.1 | IC50 | 2 | — | |
PFRXWKQQCRIVDP
|
7.1 | IC50 | 2 | — | |
WERWDDKHJRXHAF
|
7.1 | IC50 | 2 | — | |
WCPSMXYWDQGMJD
|
7.1 | IC50 | 2 | — | |
APXDEEHRWJDGMC
|
7.1 | IC50 | 2 | — | |
KNUFDNSKLOOTIB
|
7.1 | IC50 | 2 | — | |
LDYLIYKANSSERK
|
7.1 | IC50 | 2 | — | |
UHXUKJPNFOYGKB
|
7.1 | IC50 | 2 | — | |
YTNUBEUYCFIHBS
|
7.1 | IC50 | 2 | — | |
GDAGOGOXJLUVGB
|
7.1 | IC50 | 2 | — | |
LYOPDHNZJQBGAC
|
7.1 | IC50 | 2 | — | |
CJGRNBWHDOSFES
|
7.1 | Ki | 2 | — | |
DEYKKRWFIMYKJM
|
7.1 | IC50 | 2 | — | |
GYPOJYXMDPSAQP
|
7.1 | IC50 | 2 | — | |
MOTJMGVDPWRKOC
|
7.1 | IC50 | 2 | — | |
QWIJRDPSRHJFIY
|
7.1 | IC50 | 2 | — | |
XIIITWQEAPOZLF
|
7.1 | IC50 | 2 | — | |
HDHCADXZMJNZJH
|
7.0 | IC50 | 2 | — | |
VEMZPXZQLOLLKQ
|
7.0 | IC50 | 2 | — | |
VNLAEVZRIYGZCY
|
7.0 | IC50 | 2 | — | |
BSLISXSHQLGIIZ
|
7.0 | IC50 | 2 | — | |
PMUCOFCFESYTCH
|
7.0 | Ki | 2 | — | |
UMVOCHGUCRDMRD
|
7.0 | IC50 | 2 | — | |
ACMPQUAKYNONQE
|
7.0 | IC50 | 2 | — | |
DIAOYWORMSQRFB
|
7.0 | IC50 | 2 | — | |
IKSWGOKQGJQKIW
|
7.0 | IC50 | 2 | — | |
NONLTBWVEZEZFY
|
7.0 | IC50 | 2 | — | |
YPBPZJHPGUUGME
|
7.0 | IC50 | 2 | — | |
RQNOIZBVICJIJP
|
7.0 | IC50 | 2 | — | |
UPQGVXBBBKNPNZ
|
7.0 | IC50 | 2 | — | |
PYYAHQASPOJSMT
|
7.0 | IC50 | 2 | — | |
TUTZGEFUGWQBKP
|
7.0 | IC50 | 2 | — | |
XNUQKPOLJGKCNN
|
7.0 | IC50 | 2 | — | |
GLCKXJLCYIJMRB
|
7.0 | Ki | 2 | — | |
NHVWTLKWIKMKNS
|
7.0 | IC50 | 2 | — | |
YCVDVWIZRUNCFR
|
7.0 | IC50 | 2 | — | |
JNFNRBRGVCBLHK
|
6.9 | Ki | 2 | — |