Target Details
| UniProt AC | P24530 |
|---|---|
| Gene Symbol | EDNRB |
| Protein Name | Endothelin receptor type B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 507
- Clinical molecules 0
- Avg pChEMBL 7.11
KEGG Pathways (6)
Associated Diseases (4)
Active Molecules (507)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GWVRRZASHHOARI
|
7.5 | IC50 | 2 | — | |
HTKNCJNRSZJTJH
|
7.5 | IC50 | 2 | — | |
LFVLYJPEMPWXGS
|
7.5 | IC50 | 2 | — | |
XIKMSNPORKHQQQ
|
7.5 | IC50 | 2 | — | |
HMBISNTYKZVPJD
|
7.5 | Ki | 2 | — | |
MAJFWFWHJWCHLH
|
7.4 | IC50 | 2 | — | |
BQFWUVDRXODPBL
|
7.4 | IC50 | 2 | — | |
OQVTWUJKWGKZHT
|
7.4 | Ki | 2 | — | |
UTSWGARHIRATMS
|
7.4 | Ki | 2 | — | |
YNFUBOJUAKNKLF
|
7.4 | IC50 | 2 | — | |
ITRTVLHSTSAZIL
|
7.4 | IC50 | 2 | — | |
JOBIZVVLDQEHKD
|
7.4 | IC50 | 2 | — | |
PBFKMRLPTUCFLU
|
7.4 | IC50 | 2 | — | |
WQULYHKGCLHTBZ
|
7.4 | IC50 | 2 | — | |
DWNNWTCEZHVDLU
|
7.4 | IC50 | 2 | — | |
IDRPGYTWDRQQOE
|
7.4 | IC50 | 2 | — | |
RZTQQRCQEYQARM
|
7.4 | IC50 | 2 | — | |
PZBFMEKBVYTVOD
|
7.4 | IC50 | 2 | — | |
SRYQEUIBRIIYSG
|
7.4 | IC50 | 2 | — | |
IGUNGSMXNZWMPG
|
7.3 | IC50 | 2 | — | |
MRBWXOFHOJHYOZ
|
7.3 | IC50 | 2 | — | |
XAJNNLNUOAQGQO
|
7.3 | IC50 | 2 | — | |
LZPJHRAWMATYTH
|
7.3 | IC50 | 2 | — | |
QCHYZDXDWZKACW
|
7.3 | IC50 | 2 | — | |
WLXMNQFBLVMITG
|
7.3 | IC50 | 2 | — | |
DUZPNAKTFLDXQA
|
7.3 | IC50 | 2 | — | |
KIJALYSAGLYTQO
|
7.3 | IC50 | 2 | — | |
QGSBCBLFBNGHAE
|
7.3 | IC50 | 2 | — | |
BKUCZUUARYQRPP
|
7.3 | IC50 | 2 | — | |
BOQQYCYLUTYLGS
|
7.3 | IC50 | 2 | — | |
FYPZYGLVQHCNCC
|
7.3 | IC50 | 2 | — | |
NXZDWYHCLMUTOJ
|
7.3 | IC50 | 2 | — | |
DWRQMVBEIBBSTC
|
7.3 | IC50 | 2 | — | |
CQHSRRONBVIJRO
|
7.3 | IC50 | 2 | — | |
KBHRSNOQJNLUNL
|
7.3 | IC50 | 2 | — | |
ITICTHRGYDERJA
|
7.3 | IC50 | 2 | — | |
VJGDGBUWSOZGFC
|
7.3 | Ki | 2 | — | |
BKGYGEADRLJUHK
|
7.2 | IC50 | 2 | — | |
GHIWIAMAJCWXDD
|
7.2 | Ki | 2 | — | |
JOZGLYQYYYGZBS
|
7.2 | IC50 | 2 | — | |
NTQWAQFOJQQOTK
|
7.2 | IC50 | 3 | — | |
WQLXYQSKSGEIPU
|
7.2 | IC50 | 4 | — | |
FVNKNOUQLKAPJI
|
7.2 | IC50 | 2 | — | |
SBPQWNOPLSRSMS
|
7.2 | Ki | 2 | — | |
XYKNJZNFEGDDIP
|
7.2 | IC50 | 2 | — | |
YGGFLIPTDYLEIC
|
7.2 | IC50 | 2 | — | |
YZQQVZQBQWFHTP
|
7.2 | IC50 | 2 | — | |
ZYPQETRCACBJNS
|
7.2 | IC50 | 2 | — | |
DTXFUEYWZXGNEF
|
7.2 | IC50 | 2 | — | |
PQGJCQZVHZMJFI
|
7.2 | IC50 | 2 | — |