Target Details
| UniProt AC | P24530 |
|---|---|
| Gene Symbol | EDNRB |
| Protein Name | Endothelin receptor type B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 507
- Clinical molecules 0
- Avg pChEMBL 7.11
KEGG Pathways (6)
Associated Diseases (4)
Active Molecules (507)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QPZJVKVINGMRAL
|
7.7 | IC50 | 2 | — | |
UUIMPPMXRVSIPX
|
7.7 | IC50 | 2 | — | |
VYAFCUPPLXQIIN
|
7.7 | IC50 | 2 | — | |
RQKVNFYBHIQIDV
|
7.7 | IC50 | 2 | — | |
HOULTIREPNOFQE
|
7.7 | IC50 | 2 | — | |
YLMSOIIFAYJNMX
|
7.7 | IC50 | 2 | — | |
ZPWXQORYIQFGQB
|
7.7 | IC50 | 2 | — | |
UTSKZBKTKROJBZ
|
7.7 | IC50 | 2 | — | |
FFXSFOBUYYTLRH
|
7.7 | IC50 | 2 | — | |
KANHASGBLWIAIA
|
7.7 | IC50 | 2 | — | |
MSRYVIMFULZUGC
|
7.7 | Ki | 2 | — | |
XZYQXDCTRBGYKO
|
7.7 | IC50 | 2 | — | |
HAIMYEQNXQUSSG
|
7.7 | IC50 | 2 | — | |
TUYWTLTWNJOZNY
|
7.7 | IC50 | 2 | — | |
GGEVZGHUELFPFK
|
7.7 | IC50 | 2 | — | |
JQAHCXASBUTBKC
|
7.7 | IC50 | 2 | — | |
QSPLUDJQEFUAHB
|
7.7 | IC50 | 2 | — | |
VRSKDQFILRKSHK
|
7.7 | IC50 | 2 | — | |
MWZFOVILFVOLMJ
|
7.6 | IC50 | 2 | — | |
YAWKZANKTNYRSZ
|
7.6 | IC50 | 2 | — | |
PYQNCKSTTLEMCS
|
7.6 | Ki | 2 | — | |
GEKLWHMKKGCLLE
|
7.6 | IC50 | 2 | — | |
IFLIQLQVUMXNFU
|
7.6 | Ki | 2 | — | |
JKISBSRHDYZOEO
|
7.6 | Ki | 2 | — | |
KWLKTEPEDKFNSG
|
7.6 | IC50 | 2 | — | |
MIDBNMYTUQUADA
|
7.6 | Ki | 2 | — | |
NPLNAUBFRRXHRY
|
7.6 | Ki | 2 | — | |
VKZGOHFGTOOZHY
|
7.6 | IC50 | 2 | — | |
FHRCXZSDINFQMI
|
7.6 | IC50 | 2 | — | |
HWNXCQQEFQWPHX
|
7.6 | IC50 | 2 | — | |
JNUYVBGNCBJGHQ
|
7.6 | IC50 | 2 | — | |
KJNNBRVUQZDOET
|
7.6 | Ki | 2 | — | |
KXJZFAQLRGGYSV
|
7.6 | IC50 | 2 | — | |
OOJYMKAJOJBARX
|
7.6 | IC50 | 2 | — | |
WUNUEBZYLIUGHH
|
7.6 | Ki | 2 | — | |
YQDGZNPRSNHCNL
|
7.6 | IC50 | 2 | — | |
MNJJBWIQROUNDM
|
7.6 | IC50 | 2 | — | |
IJWIKFGUGIKEKW
|
7.6 | IC50 | 2 | — | |
SEXZWLMIBXVFQM
|
7.6 | IC50 | 2 | — | |
XSAFCBSWMREXMT
|
7.5 | IC50 | 2 | — | |
DVNMKMKQUAYZDJ
|
7.5 | IC50 | 2 | — | |
OBNJEEOFTPJHQY
|
7.5 | IC50 | 2 | — | |
QPUBINGNDLKIHN
|
7.5 | IC50 | 2 | — | |
JMCMZOQWXJPCLI
|
7.5 | IC50 | 2 | — | |
MZAAFBAXCKYSNN
|
7.5 | IC50 | 2 | — | |
YJMPVDOQESXRRN
|
7.5 | IC50 | 2 | — | |
DTDRDEIFMKNNTL
|
7.5 | IC50 | 2 | — | |
MHHROYOBQSBUEV
|
7.5 | IC50 | 2 | — | |
ADOZPFPWNPYHGT
|
7.5 | IC50 | 2 | — | |
FGGUYHAUIAJAKH
|
7.5 | IC50 | 2 | — |