Target Details
| UniProt AC | P24530 |
|---|---|
| Gene Symbol | EDNRB |
| Protein Name | Endothelin receptor type B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 507
- Clinical molecules 0
- Avg pChEMBL 7.11
KEGG Pathways (6)
Associated Diseases (4)
Active Molecules (507)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FYULQKSAMXDPLJ
|
8.5 | Ki | 2 | — | |
LUQZWCBOERIKEO
|
8.5 | IC50 | 2 | — | |
LZBDEPUGFFURHL
|
8.4 | IC50 | 2 | — | |
AEDJOIBTFWFFLB
|
8.4 | IC50 | 2 | — | |
FYQSINZSEYBXAC
|
8.4 | Kd | 2 | — | |
HDWHUKBOFNHSSO
|
8.4 | IC50 | 2 | — | |
JPBZOZDHBRRLBM
|
8.4 | IC50 | 2 | — | |
CLSJNXXMIVKULC
|
8.3 | Ki | 2 | — | |
FZJJZYJWWWMPOB
|
8.3 | IC50 | 2 | — | |
GQPZSZRJZWLIAV
|
8.3 | IC50 | 2 | — | |
MXLGWPUNPPHJQC
|
8.3 | IC50 | 2 | — | |
JPPYWKVKLSBQJM
|
8.3 | Ki | 2 | — | |
HAZBSXKXEZHGFW
|
8.2 | IC50 | 2 | — | |
HPSVGPXJVPTNPI
|
8.2 | IC50 | 2 | — | |
VRQCDTCXZAZNSU
|
8.2 | IC50 | 2 | — | |
NMXUCISAFBDZIZ
|
8.2 | IC50 | 2 | — | |
OTMGLEOGWQJHIQ
|
8.2 | IC50 | 2 | — | |
AUSMSARLDRBCDW
|
8.2 | IC50 | 2 | — | |
CLSJNXXMIVKULC
|
8.2 | Ki | 2 | — | |
NSROWKBSRVFCCQ
|
8.1 | IC50 | 2 | — | |
GCISLFODTRCVKS
|
8.1 | IC50 | 2 | — | |
BFGUYLRYXCFHGG
|
8.1 | IC50 | 2 | — | |
FHOLSLVTQPRBKJ
|
8.0 | IC50 | 2 | — | |
PHWXUGHIIBDVKD
|
8.0 | IC50 | 2 | — | |
KEGRAIQJSRYPGR
|
8.0 | IC50 | 2 | — | |
AQEWYBHXBBBFNY
|
8.0 | IC50 | 2 | — | |
CICVRMZHTUTILV
|
8.0 | IC50 | 2 | — | |
LTFMLNPARFSYNA
|
8.0 | IC50 | 2 | — | |
OXPNVLRJIHCUBM
|
8.0 | IC50 | 2 | — | |
YAWNVAQKVARTGQ
|
7.9 | IC50 | 2 | — | |
MIOQPXBHUMVZRF
|
7.9 | IC50 | 2 | — | |
HZWIXRSMTHDZGL
|
7.9 | IC50 | 2 | — | |
NKONTEUZTOHVNH
|
7.9 | IC50 | 2 | — | |
WFGXYWSSRLHSJI
|
7.9 | IC50 | 2 | — | |
FCGUSVKFZTVUQB
|
7.8 | IC50 | 2 | — | |
GJLMSZJTTPBCHM
|
7.8 | IC50 | 2 | — | |
OYGNCRBWGRCEDM
|
7.8 | IC50 | 2 | — | |
XBXKAPLYGJALOL
|
7.8 | IC50 | 2 | — | |
OOUHAJURRQCGRG
|
7.8 | Ki | 2 | — | |
HQIPFADRUMZDIT
|
7.8 | IC50 | 2 | — | |
UUAVCCWBNUITBB
|
7.8 | Ki | 2 | — | |
SQHUBOCKWBVIDO
|
7.8 | IC50 | 2 | — | |
YFGVPMLVIXUCGP
|
7.8 | IC50 | 2 | — | |
ASUNSLBCCFVKJD
|
7.8 | IC50 | 2 | — | |
OSRCBCUYZBTKBZ
|
7.8 | IC50 | 2 | — | |
UUAVCCWBNUITBB
|
7.8 | Ki | 2 | — | |
VWXMUZZYWKEWJY
|
7.8 | Ki | 2 | — | |
LZMBWESXCWUQBJ
|
7.8 | IC50 | 2 | — | |
JHOHFSMURHXTHA
|
7.8 | IC50 | 2 | — | |
AXVBSGVXXMZTEC
|
7.7 | IC50 | 2 | — |