Target Details
| UniProt AC | P24530 |
|---|---|
| Gene Symbol | EDNRB |
| Protein Name | Endothelin receptor type B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 507
- Clinical molecules 0
- Avg pChEMBL 7.11
KEGG Pathways (6)
Associated Diseases (4)
Active Molecules (507)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RUXNEULYFPIVIB
|
6.1 | IC50 | 2 | — | |
VRCKDEMDFQJSQX
|
6.1 | IC50 | 2 | — | |
XGEPLEYWMXVDFS
|
6.1 | IC50 | 2 | — | |
DJUNTHAWPBMJGJ
|
6.1 | IC50 | 2 | — | |
DTRNHYYWARQBED
|
6.1 | IC50 | 2 | — | |
NHKDLOQLHLFRRT
|
6.1 | IC50 | 2 | — | |
QDRPQGXYQQITQV
|
6.1 | Ki | 2 | — | |
XBXUZKKIOMHQDF
|
6.1 | IC50 | 2 | — | |
YQOHFDDJNGNMBZ
|
6.1 | IC50 | 2 | — | |
JNAFKCJWVUJAQU
|
6.1 | Ki | 2 | — | |
NBEGSXJDADJYHX
|
6.1 | IC50 | 2 | — | |
OXHAHXSAOMBNOX
|
6.1 | IC50 | 2 | — | |
PUMKVXYNDYQHJI
|
6.1 | IC50 | 2 | — | |
MODHKIOUVGRQCC
|
6.1 | IC50 | 2 | — | |
QGMUOSXKQHPOGD
|
6.1 | Ki | 2 | — | |
AXFKGEZDVMCYEO
|
6.1 | Ki | 2 | — | |
BRSITRUZDCGGKH
|
6.1 | IC50 | 2 | — | |
FPZOGKSKYWZFIO
|
6.1 | IC50 | 2 | — | |
OZBAKTZMSBVKFA
|
6.1 | IC50 | 2 | — | |
PIJUSICWAKBTEZ
|
6.1 | IC50 | 2 | — | |
ZHWQNJCSTDEVGM
|
6.1 | IC50 | 2 | — | |
ARCCNAPMMHWOCU
|
6.1 | IC50 | 2 | — | |
HXUVUUFEMYJLDB
|
6.1 | IC50 | 2 | — | |
LQWGCVIETCFLOP
|
6.1 | IC50 | 2 | — | |
OVPKPOGJHFVIFR
|
6.1 | IC50 | 2 | — | |
RDFPZCGBCKZXNO
|
6.1 | IC50 | 2 | — | |
JXZLHWXGEORAOB
|
6.1 | IC50 | 2 | — | |
KJNXTLHIZCKQRF
|
6.1 | IC50 | 2 | — | |
OGGZHZAVIHOULX
|
6.1 | IC50 | 2 | — | |
BMROGBGRQLVZIB
|
6.0 | IC50 | 2 | — | |
FIMDOJGUQJFHTD
|
6.0 | IC50 | 2 | — | |
PTGZJENBFJFKND
|
6.0 | IC50 | 2 | — | |
FKUFTGMFORIVAP
|
6.0 | IC50 | 2 | — | |
JZVDVZMUHGSKGI
|
6.0 | IC50 | 2 | — | |
NNXCMHJFFYTMCA
|
6.0 | IC50 | 2 | — | |
WLIQAZXJDQKSEC
|
6.0 | IC50 | 2 | — | |
ZXSBLFBQTHAAHA
|
6.0 | IC50 | 2 | — | |
KPISXONXINCUAB
|
6.0 | IC50 | 2 | — | |
KZOKREKJZZEWAD
|
6.0 | IC50 | 2 | — | |
LQXABJNKFHBROP
|
6.0 | IC50 | 2 | — | |
VTCDHOQFPYTIFV
|
6.0 | IC50 | 2 | — | |
FEJVSJIALLTFRP
|
6.0 | Ki | 2 | — | |
JOFLWUQNEHCQRX
|
6.0 | IC50 | 2 | — | |
NRDKXLWFPVYSKL
|
6.0 | IC50 | 2 | — | |
RLZUSDGCLWDQGG
|
6.0 | IC50 | 2 | — | |
XVGVBINHYILTRX
|
6.0 | Ki | 2 | — | |
DKULOVKANLVDEA
|
6.0 | IC50 | 2 | — | |
FTHTWZGSLVJZJB
|
6.0 | Ki | 2 | — | |
PBTTZSSLQDEUPI
|
6.0 | IC50 | 2 | — | |
VHHUBYWYNJXLPT
|
6.0 | Ki | 2 | — |