Target Details
UniProt ACP24530
Gene SymbolEDNRB
Protein NameEndothelin receptor type B
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 507
  • Clinical molecules 0
  • Avg pChEMBL 7.11
Top Co-occurrence Targets
Active Molecules (507)
InChIKey pChEMBL Type Targets Clinical
IUHMIOAKWHUFKU 10.0 Ki 2
YGARCWJUVOXSDS 10.0 IC50 2
CSBNIDOCJNQVQX 9.8 Ki 2
ZUBDGKVDJUIMQQ 9.8 IC50 2
UVTGPXVPTNTUDR 9.7 Ki 2
HVBUELUOUQXXRH 9.6 Ki 2
PZBNHZOXFOMEDO 9.6 Ki 2
VLHPYESMRDUJNS 9.6 Ki 2
HUDYDAYXYKCRPT 9.6 Ki 2
XBKVYIJFYBIMJN 9.6 Ki 2
MMVFGIYZPKSYRV 9.5 Ki 2
IPZKGERDMRMXJO 9.5 IC50 2
CIMUQXQFDACEAW 9.4 Ki 2
LGRQZNNALZAMDJ 9.4 Ki 2
KOWYKBJZTIDYKI 9.4 Ki 2
GJEGFKNDKHXDSQ 9.3 Ki 2
XRUKXLWYVUMZLF 9.3 Ki 2
SISHUQWGICPIJE 9.3 IC50 2
BMNFTWGABWKVKN 9.3 IC50 2
KBYIOWQONLGJJU 9.2 Ki 2
CFTTVXIBXXPWEU 9.2 Ki 2
MWHGEJXLFJLVHX 9.2 Ki 2
UNUUFLTUZOLRDF 9.2 IC50 2
WELUHUKTVXHVBY 9.1 IC50 2
RDVHLMJRZJBHMF 9.1 Ki 2
GAICYMPBDZVZOU 9.1 IC50 2
XDNAXXIOBHFZDQ 9.1 IC50 2
ZHGGJHSZAGTHLS 9.1 Ki 2
NSVNTHSZOXQBPE 9.0 IC50 2
BSUWUKYJNUNGOM 9.0 IC50 2
JYYUWMLSDGSJDK 9.0 IC50 2
XDNAXXIOBHFZDQ 9.0 IC50 2
JVWVTPZZEHLARL 8.9 IC50 2
UZDORQWMYRRLQV 8.9 IC50 2
CQHLNCPJLNXFBC 8.9 IC50 2
IFLIQLQVUMXNFU 8.9 Ki 2
KEZZZBNAPVGBEW 8.9 IC50 2
RNNCMVHNZGHSLY 8.9 IC50 2
IAHNMFPHUACREU 8.9 Ki 2
JMWQBPRIANCZRQ 8.8 IC50 2
BYIKTFONIZDLEI 8.8 IC50 2
BCRJIIJVFJJYRD 8.7 IC50 2
DASGRKPWAFYAFD 8.7 IC50 2
WOQBGOSNHKHPRH 8.7 IC50 2
ZWURMMRAUYXFRY 8.6 IC50 2
QLRLGCLZQTWZOK 8.5 Ki 2
WETZUHODUGXVKY 8.5 Ki 2
WZCUCQGZYXGPHF 8.5 Ki 2
HFWWOBMAMIJJEP 8.5 IC50 2
WYLRXEBBERTKHN 8.5 IC50 2
2D structure