Target Details
| UniProt AC | P24385 |
|---|---|
| Gene Symbol | CCND1 |
| Protein Name | G1/S-specific cyclin-D1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02984 (Cyclin_C) PF00134 (Cyclin_N) |
Summary
- Multi-target molecules 1,643
- Clinical molecules 278
- Avg pChEMBL 7.73
KEGG Pathways (49)
- AGE-RAGE signaling pathway in diabetic complications
- AMPK signaling pathway
- Acute myeloid leukemia
- Alcoholic liver disease
- Apelin signaling pathway
- Bladder cancer
- Breast cancer
- Cell cycle
- Cellular senescence
- Chemical carcinogenesis - receptor activation
- Chronic myeloid leukemia
- Colorectal cancer
- Cushing syndrome
- Endocrine resistance
- Endometrial cancer
- Epstein-Barr virus infection
- Focal adhesion
- FoxO signaling pathway
- Gastric cancer
- Glioma
- Hedgehog signaling pathway
- Hepatitis C
- Hepatocellular carcinoma
- Hippo signaling pathway
- Human T-cell leukemia virus 1 infection
- Human cytomegalovirus infection
- Human papillomavirus infection
- Integrin signaling
- JAK-STAT signaling pathway
- Kaposi sarcoma-associated herpesvirus infection
- Measles
- Melanoma
- MicroRNAs in cancer
- Non-small cell lung cancer
- Oxytocin signaling pathway
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Prolactin signaling pathway
- Prostate cancer
- Proteoglycans in cancer
- Small cell lung cancer
- Thyroid cancer
- Thyroid hormone signaling pathway
- Tight junction
- Viral carcinogenesis
- Viral myocarditis
- Wnt signaling pathway
- p53 signaling pathway
Associated Diseases (9)
Active Molecules (1,643)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QELIOBZBBHRBAA
|
8.6 | Ki | 4 | — | |
TWBXLKWAYLBJOV
|
8.6 | IC50 | 3 | — | |
WWYNWGGCJJEZAV
|
8.6 | Ki | 4 | — | |
NXHNUMBGXRTEFE
|
8.6 | Ki | 4 | — | |
PKXRYTDXRPPJDM
|
8.6 | Ki | 4 | — | |
ZBJPNNCODVAXRF
|
8.6 | Ki | 4 | — | |
ZBYFYISKUULBLB
|
8.6 | Ki | 4 | — | |
BSGQHAMZJBZCDP
|
8.6 | IC50 | 3 | — | |
GWZYVJHBZJZRJD
|
8.6 | IC50 | 2 | — | |
NVPGIFLCJMRJOV
|
8.6 | IC50 | 2 | — | |
FVTBNLXYEQBKLR
|
8.6 | IC50 | 2 | — | |
MCGKCTAGXKRXDO
|
8.6 | Ki | 4 | — | |
FIFYTWABWYHZIS
|
8.6 | Ki | 4 | — | |
FIHHRMZWXIZLJV
|
8.6 | Ki | 4 | — | |
GEHWYWMDTGSDFR
|
8.6 | Ki | 4 | — | |
HGINWKMFVVFJSI
|
8.6 | Ki | 4 | — | |
KOOSKJVCROTXBQ
|
8.6 | IC50 | 3 | — | |
QVWFFHVKVHIONZ
|
8.6 | Ki | 4 | — | |
XZKHOZLKTBKGNZ
|
8.6 | Ki | 4 | — | |
WFMBBNNZNAMTGD
|
8.6 | Ki | 7 | — | |
XFCBYRQZMFSMHZ
|
8.6 | Ki | 4 | — | |
XLSYZSRXVVCHLS
|
8.6 | IC50 | 48 | — | |
YNJJUSMMVIXAQM
|
8.6 | IC50 | 3 | — | |
DVAPMYJVUZJNDK
|
8.5 | Ki | 8 | — | |
HKSZLNNOFSGOKW
|
8.5 | IC50 | 49 | Yes | |
UZGLLJQDQDOFFE
|
8.5 | IC50 | 2 | — | |
AEFFENQISAXIKE
|
8.5 | IC50 | 9 | — | |
AMPDZRFNHCTPTF
|
8.5 | Ki | 10 | — | |
AZXYPCBAGCXZPP
|
8.5 | IC50 | 4 | — | |
BBUVDDPUURMFOX
|
8.5 | IC50 | 3 | — | |
CGZPQEKNAAVWHA
|
8.5 | Ki | 4 | — | |
CQMZJAORBQTGTR
|
8.5 | IC50 | 4 | — | |
CZPQAZKLLINYQE
|
8.5 | IC50 | 2 | — | |
DUHXDQPGUINDGD
|
8.5 | IC50 | 3 | — | |
GBVXPZRKGCHAIL
|
8.5 | IC50 | 6 | — | |
GTQSNWXKTIFPBY
|
8.5 | IC50 | 5 | — | |
HOKDQPMWTBQYHL
|
8.5 | IC50 | 8 | — | |
HOWIXJOUKWURJN
|
8.5 | IC50 | 2 | — | |
ICVHMFOFVOYFPB
|
8.5 | IC50 | 3 | — | |
IEPYZPJZYINELK
|
8.5 | IC50 | 5 | — | |
JYLSDMOABXIYSW
|
8.5 | IC50 | 3 | — | |
MGLCYKLRRMBDTH
|
8.5 | IC50 | 3 | — | |
NWIPTENCWQPQTO
|
8.5 | Ki | 4 | Yes | |
POFVJRKJJBFPII
|
8.5 | Ki | 8 | — | |
QFGDMFUYBQHULK
|
8.5 | IC50 | 3 | — | |
SHEPFXMPLORKLW
|
8.5 | Ki | 8 | — | |
TUVPQAXSMZXTMF
|
8.5 | IC50 | 2 | — | |
USXJKWQIDCWKGZ
|
8.5 | Ki | 10 | — | |
VCQXPLQAUTUUTC
|
8.5 | IC50 | 3 | — | |
VFNJLPYDAYDGKC
|
8.5 | IC50 | 5 | — |