Target Details
| UniProt AC | P24158 |
|---|---|
| Gene Symbol | PRTN3 |
| Protein Name | Myeloblastin |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00089 (Trypsin) |
Summary
- Multi-target molecules 12
- Clinical molecules 0
- Avg pChEMBL 6.81
Active Molecules (12)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LRHBPVVPFQMQPP
|
8.2 | Ki | 6 | — | |
RNXBQIJUOJFKHW
|
8.2 | Ki | 2 | — | |
NHPVRNNXFZLMPU
|
7.8 | Ki | 2 | — | |
MSIGLHAWDSGRGI
|
6.7 | IC50 | 2 | — | |
LDFVFAFYMOXYNX
|
6.5 | IC50 | 2 | — | |
BTGNGJJLZOIYID
|
6.5 | IC50 | 2 | — | |
CPJZBAKYBNKFMF
|
6.4 | IC50 | 2 | — | |
DOVSNSDMRJVTMR
|
6.4 | IC50 | 2 | — | |
AOYZKUMTEYCRDS
|
6.3 | IC50 | 2 | — | |
OXSUHSQWSLABCN
|
6.3 | IC50 | 2 | — | |
OMVZRWSTCVAYPK
|
6.2 | IC50 | 2 | — | |
PSORSGLVGFXCQD
|
6.2 | IC50 | 2 | — |