Target Details
| UniProt AC | P23975 |
|---|---|
| Gene Symbol | SLC6A2 |
| Protein Name | Sodium-dependent noradrenaline transporter |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00209 (SNF) |
Summary
- Multi-target molecules 2,491
- Clinical molecules 106
- Avg pChEMBL 7.28
KEGG Pathways (2)
Associated Diseases (1)
Active Molecules (2,491)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VZYAMIGSWLJHCX
|
10.2 | IC50 | 3 | — | |
DRKVKHDMRAXUGE
|
10.1 | Ki | 3 | — | |
PZYPYVNKHXTQCH
|
10.1 | IC50 | 2 | — | |
WFSYXANMSWQZLY
|
10.1 | IC50 | 3 | — | |
HIDQBTRNELCGFN
|
10.0 | IC50 | 3 | — | |
UEZGSCSNHZZABE
|
9.9 | IC50 | 3 | — | |
QNFARVIAWDUFFL
|
9.7 | IC50 | 2 | — | |
JNLXUEPMJIMNHM
|
9.6 | Ki | 3 | — | |
PYIBCEOJEPANCH
|
9.6 | Ki | 3 | — | |
YLQFFYJKBKUKLF
|
9.5 | Ki | 3 | — | |
DPINDTNFGDXWLU
|
9.5 | IC50 | 3 | — | |
VZKPRNYGLKTGQY
|
9.5 | IC50 | 2 | — | |
ONSLZFSSJGOMSK
|
9.4 | Ki | 3 | — | |
KUJKCGJIUCGPED
|
9.4 | Ki | 3 | — | |
URVPSAOJVKMKND
|
9.4 | IC50 | 3 | — | |
WDFMVSDPRALOJK
|
9.4 | IC50 | 3 | — | |
DPINDTNFGDXWLU
|
9.3 | IC50 | 3 | — | |
GIKANUDLIOICAL
|
9.3 | IC50 | 4 | — | |
HIKRIVCRSDESKA
|
9.3 | IC50 | 3 | — | |
IBZJKEOJOGAMGJ
|
9.3 | Ki | 11 | Yes | |
QDZIBQWKRRRXAL
|
9.3 | IC50 | 3 | — | |
RRGCJEHCXSKPFY
|
9.3 | IC50 | 2 | — | |
UUSPTDRDECONSP
|
9.3 | IC50 | 3 | — | |
DHKBDZKBBAEQNU
|
9.2 | IC50 | 3 | — | |
GXWUVPPXUBCALT
|
9.2 | Ki | 3 | — | |
KIMRUTAJTDBFHO
|
9.2 | Ki | 4 | — | |
KMNJYBBPXRFSBY
|
9.2 | Ki | 3 | — | |
ORUPHFRKUPILCN
|
9.2 | Ki | 4 | — | |
PJIMUTYPWDGKIC
|
9.2 | Ki | 3 | — | |
VNJFIBFHISUZRV
|
9.2 | Ki | 4 | — | |
PAIAJJFPYBWMBV
|
9.2 | IC50 | 2 | — | |
UCAUHLPHMUPKJI
|
9.2 | Ki | 3 | — | |
VWKLNUPRXXIKKE
|
9.1 | Ki | 2 | — | |
JYATVHIJHCVTMN
|
9.1 | IC50 | 3 | — | |
IJNSXDVGJQEXPC
|
9.1 | IC50 | 3 | — | |
MCHVXQNUHBOZIA
|
9.1 | IC50 | 3 | — | |
QLILSXLCYHMHMR
|
9.1 | IC50 | 3 | — | |
RSAGNBIVUSOUTP
|
9.1 | IC50 | 3 | — | |
VMITZEMDDZVHBZ
|
9.1 | IC50 | 3 | — | |
YHCLEHAMAKETBI
|
9.1 | IC50 | 3 | — | |
YMQUDJCSTPMZTF
|
9.1 | Ki | 3 | — | |
YBVYVIFNGYOFSX
|
9.1 | IC50 | 3 | — | |
MZGJHBJKODTIQM
|
9.0 | Ki | 2 | — | |
CIVPMJLKYXGWQT
|
9.0 | Ki | 3 | — | |
IJNSXDVGJQEXPC
|
9.0 | IC50 | 3 | — | |
IRFOFLZPBFIIGA
|
9.0 | IC50 | 3 | — | |
JTLPJEXKDFZLAY
|
9.0 | Ki | 2 | — | |
OSXVIZKTSFAUPG
|
9.0 | Ki | 4 | — | |
QCGAHDLRCVBZHH
|
9.0 | Ki | 3 | — | |
RJEHJYSUUDYRCE
|
9.0 | IC50 | 2 | — |