Target Details
UniProt ACP23946
Gene SymbolCMA1
Protein NameChymase
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00089 (Trypsin)
Summary
  • Multi-target molecules 67
  • Clinical molecules 0
  • Avg pChEMBL 7.57
Top Co-occurrence Targets
Active Molecules (67)
InChIKey pChEMBL Type Targets Clinical
HQIKQQKBLGAORR 8.8 IC50 6
RERFKFYMYKTFND 8.8 Ki 5
FVFSUZHBTIUSFU 8.7 Ki 2
JBVRJKUPBUZDDJ 8.6 Ki 2
NQFWNRFKRYMGAI 8.5 Ki 2
XUJQPDQURBZEGJ 8.5 IC50 2
XUJQPDQURBZEGJ 8.5 IC50 2
JDARDSVOVYVQST 8.4 IC50 2
PGIXYPNBNAOYHW 8.4 IC50 5
FNQYNLSBEYGVCO 8.3 IC50 3
DGAACZPYHKOXDE 8.2 IC50 3
DWKQSWOPFOFIHM 8.2 Ki 2
DWKQSWOPFOFIHM 8.2 Ki 2
RSKAMAUHJHZMQX 8.2 Ki 6
PDFLMEOJDBZIJL 8.2 IC50 4
WMDQHRZMWIVOHA 8.2 Ki 2
XADHZGACMQLWMK 8.1 Ki 6
KKRGXDSPEUYYKM 8.1 IC50 6
NUNGDKUJSAHDEV 8.1 Ki 2
YGRSMPVCBHOYMS 8.0 Ki 2
SNCGFOXGVUAVRV 8.0 Ki 2
XAMQZXSJYFEDPF 8.0 Ki 2
WYMWGQYFGRDOEW 7.9 IC50 3
LUAHLAHELOSEBD 7.9 Ki 2
MRXDGVXSWIXTQL 7.9 IC50 2
YBGXUZGJYQNALN 7.9 Ki 2
DFUULODUOQISLS 7.8 Ki 2
GHWYBKPVWOOAPL 7.8 Ki 2
WISJYGPAQGRLCK 7.7 IC50 2
HCFCPJNPHOFKAO 7.7 Ki 2
AZTARPFJXYNPTC 7.7 IC50 4
ZBVDAILDYSBUAI 7.7 Ki 6
YSOMBHFITHOMPW 7.7 IC50 2
HIUQSFGYYWNUPS 7.6 Ki 2
BBAWEDCPNXPBQM 7.6 IC50 9
VUEVZBHUKRORBJ 7.6 IC50 2
BWTNDBKCQZCMSA 7.5 IC50 2
IMXJHAMVFYJETE 7.5 IC50 2
KJWGUGYELVNALG 7.5 IC50 3
LHHCSNFAOIFYRV 7.5 IC50 8
HUMKWHCZOMYLFG 7.5 Ki 2
PWVRTWWSNMKTDS 7.5 Ki 2
CEAQLKDYOYEPQY 7.4 IC50 3
YDCSNPSSWBJJIR 7.4 IC50 2
XDTTYVCUSUPDCP 7.3 Ki 2
MBGPBHRYFCMIPN 7.3 Ki 5
HPGZOBMWVCIJEN 7.2 IC50 3
YVERQXIEPUPSEH 7.2 IC50 2
XAIBYEBSDCVCAA 7.2 IC50 2
MSMUEUPZLNNJEQ 7.1 Ki 2
2D structure