Target Details
| UniProt AC | P23743 |
|---|---|
| Gene Symbol | DGKA |
| Protein Name | Diacylglycerol kinase alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF14513 (DAG_kinase_N) PF00609 (DAGK_acc) PF00781 (DAGK_cat) |
Summary
- Multi-target molecules 602
- Clinical molecules 0
- Avg pChEMBL 6.95
KEGG Pathways (6)
Active Molecules (602)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IHYGFNVKFQBGBL
|
7.1 | IC50 | 2 | — | |
LRDFZCUPPMVNOG
|
7.1 | IC50 | 2 | — | |
YZKWVJLUQQWBMW
|
7.0 | IC50 | 2 | — | |
MQFZXGIUEHCSRW
|
7.0 | IC50 | 2 | — | |
NALBGDIPGZZNPU
|
7.0 | IC50 | 2 | — | |
ROJUBHHZPCNNHB
|
7.0 | IC50 | 2 | — | |
FPFNLEITMFVBFR
|
7.0 | IC50 | 2 | — | |
YPOLDQUTKVKLAC
|
7.0 | IC50 | 2 | — | |
VAMCGULYLMVAFZ
|
7.0 | IC50 | 2 | — | |
AXHAGKHSYRVLOD
|
7.0 | IC50 | 2 | — | |
NALBGDIPGZZNPU
|
7.0 | IC50 | 2 | — | |
VSKMLJUHNWUTOR
|
7.0 | IC50 | 2 | — | |
NGFKLLURPNIYOB
|
7.0 | IC50 | 2 | — | |
ZNGFYPGJBRQQGH
|
7.0 | IC50 | 2 | — | |
DHVPUHWXIGHNFO
|
7.0 | IC50 | 2 | — | |
UUWAPVVCYGIXME
|
7.0 | IC50 | 2 | — | |
AZSUDGZSKNUIDL
|
7.0 | IC50 | 2 | — | |
BBTYAQXYBAZXSH
|
7.0 | IC50 | 2 | — | |
LDVSVGYKPLBAIF
|
7.0 | IC50 | 2 | — | |
UMWFXEDDZKUQFI
|
7.0 | IC50 | 2 | — | |
VJBDPCBYYMZIDA
|
7.0 | IC50 | 2 | — | |
BXELTHAKILJGRL
|
6.9 | IC50 | 2 | — | |
JOOLNXYMZCGYHE
|
6.9 | IC50 | 2 | — | |
TXKGQNQDLBAMGH
|
6.9 | IC50 | 2 | — | |
WHIADQDFBPMMDU
|
6.9 | IC50 | 2 | — | |
IAHVZWOOPIRCFP
|
6.9 | IC50 | 2 | — | |
LRPZCKXZLKOFCR
|
6.9 | IC50 | 2 | — | |
NNFZKMUSGYIMJR
|
6.9 | IC50 | 2 | — | |
AIVDFWPDLDQNIT
|
6.9 | IC50 | 2 | — | |
CYYJMUNSJMTJAQ
|
6.9 | IC50 | 2 | — | |
JZURNMQGKZUYTO
|
6.9 | IC50 | 2 | — | |
QRKDAQMUDNGYFH
|
6.9 | IC50 | 2 | — | |
VNTNTWQXDHPADI
|
6.9 | IC50 | 2 | — | |
XXSHBOTWQGLOOB
|
6.9 | IC50 | 2 | — | |
ZAMDRPUSGBMQPY
|
6.9 | IC50 | 2 | — | |
YUQGIFMXFXYLJM
|
6.9 | IC50 | 2 | — | |
FIDWNNPDXFYCCC
|
6.9 | IC50 | 2 | — | |
HJPYIWYWEGLCDH
|
6.9 | IC50 | 2 | — | |
NLKPDRDYJHFQDR
|
6.9 | IC50 | 2 | — | |
CCBLWZOUZOWTTD
|
6.9 | IC50 | 2 | — | |
FOUKILCVIKGIFD
|
6.9 | IC50 | 2 | — | |
GIUGPGNKCSNMTD
|
6.9 | IC50 | 2 | — | |
OYCLQKSMENELGY
|
6.9 | IC50 | 2 | — | |
PJUXVVUCSUAXJK
|
6.9 | IC50 | 2 | — | |
YWDBJKNPZWFYGQ
|
6.9 | IC50 | 2 | — | |
AIVDFWPDLDQNIT
|
6.9 | IC50 | 2 | — | |
FKWOBRNPWQEVCD
|
6.9 | IC50 | 2 | — | |
HXVZPMYQYLPZTN
|
6.9 | IC50 | 2 | — | |
OEVWBZQTSYXUMP
|
6.9 | IC50 | 2 | — | |
HZAQCPXZCYUIHK
|
6.8 | IC50 | 2 | — |