Target Details
| UniProt AC | P23743 |
|---|---|
| Gene Symbol | DGKA |
| Protein Name | Diacylglycerol kinase alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF14513 (DAG_kinase_N) PF00609 (DAGK_acc) PF00781 (DAGK_cat) |
Summary
- Multi-target molecules 602
- Clinical molecules 0
- Avg pChEMBL 6.95
KEGG Pathways (6)
Active Molecules (602)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BYKFYOKJPGUNAA
|
9.0 | IC50 | 2 | — | |
BJQUZQCQURWIFF
|
8.7 | IC50 | 2 | — | |
CSGAEEBCVJCSNT
|
8.7 | IC50 | 2 | — | |
LPRUJAUVHPQLBZ
|
8.7 | IC50 | 2 | — | |
VTSHKKONDMPIMA
|
8.7 | IC50 | 2 | — | |
GTWMNNUMVLGAGX
|
8.7 | IC50 | 2 | — | |
BAODLKSFSNLJNA
|
8.6 | IC50 | 2 | — | |
BUPUSOPATJEBTJ
|
8.5 | IC50 | 2 | — | |
KNEROOXXUFWGJG
|
8.5 | IC50 | 2 | — | |
OGWDRSCFXBZVLF
|
8.5 | IC50 | 2 | — | |
VZOODQRZMWZABR
|
8.5 | IC50 | 2 | — | |
XUOSUEUNXZNGLU
|
8.5 | IC50 | 2 | — | |
ZUIBYMTVKIBSFU
|
8.5 | IC50 | 2 | — | |
VTSHKKONDMPIMA
|
8.4 | IC50 | 2 | — | |
NLCGWOCDNDMESP
|
8.4 | IC50 | 2 | — | |
OIJJUDSQJFRQJO
|
8.4 | IC50 | 2 | — | |
SGMHRVADCWKYNE
|
8.4 | IC50 | 2 | — | |
XEBIGJPRBYBJCT
|
8.4 | IC50 | 2 | — | |
CHHDXZMBRMBJND
|
8.4 | IC50 | 2 | — | |
CMQUMOFRQVSJBY
|
8.4 | IC50 | 2 | — | |
OIYGURYNTMBMFX
|
8.4 | IC50 | 2 | — | |
GZSZUNRIGWPCEU
|
8.4 | IC50 | 2 | — | |
ULMQKFGWNBCDOA
|
8.3 | IC50 | 2 | — | |
WWYRRIXMRBOBPV
|
8.3 | IC50 | 2 | — | |
XAHMIJCNFUSTMT
|
8.3 | IC50 | 5 | — | |
YVKUPUFXGMVIPV
|
8.3 | IC50 | 2 | — | |
ITXYZZWMUWXKLB
|
8.3 | IC50 | 2 | — | |
IFLUOHYLAOOPPM
|
8.2 | IC50 | 2 | — | |
IFLUOHYLAOOPPM
|
8.2 | IC50 | 2 | — | |
LPRUJAUVHPQLBZ
|
8.2 | IC50 | 2 | — | |
OIJJUDSQJFRQJO
|
8.2 | IC50 | 2 | — | |
RYANVYSVCYNQFK
|
8.2 | IC50 | 2 | — | |
UBVHJAFAZDBCMD
|
8.2 | IC50 | 2 | — | |
HRSQHAKCQPOBGZ
|
8.1 | IC50 | 2 | — | |
RPWBAOPOLGTNMO
|
8.1 | IC50 | 2 | — | |
HXVZPMYQYLPZTN
|
8.1 | IC50 | 2 | — | |
JJADZKTWJXFGBO
|
8.1 | IC50 | 2 | — | |
BBOXBKOMCYZQAX
|
8.1 | IC50 | 2 | — | |
CZZLNVIJCVVDRT
|
8.1 | IC50 | 2 | — | |
GYBMYFBRAOIKDJ
|
8.1 | IC50 | 2 | — | |
OIJJUDSQJFRQJO
|
8.1 | IC50 | 2 | — | |
PLBSSVSZEMKBGC
|
8.1 | IC50 | 2 | — | |
RGINEJGBRUOJFR
|
8.1 | IC50 | 2 | — | |
RUWKUJCWKWQZPL
|
8.1 | IC50 | 2 | — | |
ZRUJIFQLHPPENZ
|
8.0 | IC50 | 2 | — | |
LRPZCKXZLKOFCR
|
8.0 | IC50 | 2 | — | |
MRMLFXOFRQVANT
|
8.0 | IC50 | 2 | — | |
OGWDRSCFXBZVLF
|
8.0 | IC50 | 2 | — | |
PQDGLYOENNXENG
|
8.0 | IC50 | 2 | — | |
SGMHRVADCWKYNE
|
8.0 | IC50 | 2 | — |