Target Details
| UniProt AC | P23443 |
|---|---|
| Gene Symbol | RPS6KB1 |
| Protein Name | Ribosomal protein S6 kinase beta-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 1,180
- Clinical molecules 27
- Avg pChEMBL 7.62
KEGG Pathways (31)
- AMPK signaling pathway
- Acute myeloid leukemia
- Apelin signaling pathway
- Autophagy - animal
- Breast cancer
- Chemical carcinogenesis - receptor activation
- Choline metabolism in cancer
- Colorectal cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocrine resistance
- ErbB signaling pathway
- Fc gamma R-mediated phagocytosis
- Gastric cancer
- HIF-1 signaling pathway
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human immunodeficiency virus 1 infection
- Human papillomavirus infection
- Insulin resistance
- Insulin signaling pathway
- Longevity regulating pathway
- Longevity regulating pathway - multiple species
- PD-L1 expression and PD-1 checkpoint pathway in cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Proteoglycans in cancer
- Shigellosis
- TGF-beta signaling pathway
- Thermogenesis
- mTOR signaling pathway
Active Molecules (1,180)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZIVRJCGAZHOIHR
|
8.2 | IC50 | 2 | — | |
CVCLGNCOASWGPB
|
8.2 | IC50 | 2 | — | |
CXSQMXRQOZZFLD
|
8.2 | IC50 | 18 | — | |
CZIVUSJISIAXJB
|
8.2 | IC50 | 18 | — | |
FFJNCCISXWZBSC
|
8.2 | IC50 | 2 | — | |
PABLVBARXHFRFL
|
8.2 | Kd | 5 | — | |
XONRTPBYDAFIRW
|
8.2 | IC50 | 9 | — | |
ASWOCBCCZIYUHK
|
8.1 | IC50 | 2 | — | |
GWUYLDMVDQHMJN
|
8.1 | IC50 | 2 | — | |
XWAKIYAMWRQWDT
|
8.1 | IC50 | 4 | — | |
FVJQXZUWHGTQIX
|
8.1 | IC50 | 2 | — | |
HITVHYHCWXALKZ
|
8.1 | IC50 | 2 | — | |
PZOKYBNWYFILSM
|
8.1 | IC50 | 2 | — | |
MHGPJIHGGLSWFD
|
8.1 | IC50 | 8 | — | |
MTUDBXWJNZCYKU
|
8.1 | IC50 | 2 | — | |
QUGOKCFHVXBZFZ
|
8.1 | IC50 | 2 | — | |
BHSOPYVVEZFHDB
|
8.1 | Ki | 25 | Yes | |
GSXRCPJTNIGKSZ
|
8.1 | Ki | 43 | — | |
LYADGAGFYYXXIO
|
8.1 | IC50 | 82 | — | |
VXYDJXMHISGSDA
|
8.1 | Ki | 59 | — | |
WBOJNPOFWWQXBX
|
8.1 | IC50 | 4 | — | |
XYRCIBHDJSUCBV
|
8.1 | IC50 | 2 | — | |
CXSMTMCUUMPVML
|
8.1 | IC50 | 2 | — | |
NSHZNQHXFGNGRZ
|
8.1 | IC50 | 2 | — | |
OWCPNEJTTGLSQC
|
8.1 | IC50 | 4 | — | |
SXBOBECESAKPQZ
|
8.1 | IC50 | 2 | — | |
ZGVJCAMSCAQSAM
|
8.1 | IC50 | 2 | — | |
ZTCGLAMYEAGAAN
|
8.1 | IC50 | 2 | — | |
OPIDKMDIFBLRSY
|
8.1 | IC50 | 2 | — | |
FNVHPAHIBFFSHW
|
8.1 | IC50 | 2 | — | |
GGFFWRSIWQPPJE
|
8.1 | IC50 | 2 | — | |
HCBIHPMBVAMDAB
|
8.1 | IC50 | 3 | — | |
QHCQKCYWPJSUQX
|
8.1 | IC50 | 2 | — | |
GKXOHJMEBCPQIB
|
8.1 | IC50 | 2 | — | |
IXXXRLXHQHLRSJ
|
8.1 | IC50 | 3 | — | |
NUAVXRQHCVNICO
|
8.1 | IC50 | 2 | — | |
OHUFXMWOWSOHFW
|
8.1 | IC50 | 2 | — | |
OQISTSSMSVJSIA
|
8.1 | IC50 | 2 | — | |
SXDPQGRNHSLZPC
|
8.1 | IC50 | 18 | — | |
ZKQGSMFEXARYCS
|
8.1 | IC50 | 3 | — | |
GTUAZZUFAUMXII
|
8.0 | IC50 | 2 | — | |
NCEKGJMLNJWDDU
|
8.0 | IC50 | 2 | — | |
RFRCSMPUQCLUQP
|
8.0 | IC50 | 2 | — | |
INIPMXIFCLHYIN
|
8.0 | IC50 | 2 | — | |
JSWLTWQQWLTHEL
|
8.0 | IC50 | 2 | — | |
MMJLTRRVKQFACD
|
8.0 | IC50 | 2 | — | |
RGLSQZGEAOHRTM
|
8.0 | IC50 | 3 | — | |
SEZZPLMFRCCWJD
|
8.0 | IC50 | 2 | — | |
JVFZWHNQUXTCCX
|
8.0 | IC50 | 2 | — | |
JWYNPNNKXPDNQR
|
8.0 | IC50 | 2 | — |