Target Details
| UniProt AC | P23443 |
|---|---|
| Gene Symbol | RPS6KB1 |
| Protein Name | Ribosomal protein S6 kinase beta-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 1,180
- Clinical molecules 27
- Avg pChEMBL 7.62
KEGG Pathways (31)
- AMPK signaling pathway
- Acute myeloid leukemia
- Apelin signaling pathway
- Autophagy - animal
- Breast cancer
- Chemical carcinogenesis - receptor activation
- Choline metabolism in cancer
- Colorectal cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocrine resistance
- ErbB signaling pathway
- Fc gamma R-mediated phagocytosis
- Gastric cancer
- HIF-1 signaling pathway
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human immunodeficiency virus 1 infection
- Human papillomavirus infection
- Insulin resistance
- Insulin signaling pathway
- Longevity regulating pathway
- Longevity regulating pathway - multiple species
- PD-L1 expression and PD-1 checkpoint pathway in cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Proteoglycans in cancer
- Shigellosis
- TGF-beta signaling pathway
- Thermogenesis
- mTOR signaling pathway
Active Molecules (1,180)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LJXSBCQMIYAMGA
|
8.3 | IC50 | 2 | — | |
LRMSXQHUFDZMGI
|
8.3 | IC50 | 2 | — | |
LVVCVENXRLWTCD
|
8.3 | IC50 | 2 | — | |
MQOJWNUSDMISEA
|
8.3 | IC50 | 2 | — | |
NZRLHDMDWYOVDS
|
8.3 | IC50 | 2 | — | |
OGKDMWHNCKBDCJ
|
8.3 | IC50 | 2 | — | |
OIRFZMZDQYSRGA
|
8.3 | IC50 | 2 | — | |
PMRNETHOPVNITN
|
8.3 | IC50 | 2 | — | |
QAQKEARBBXQETD
|
8.3 | IC50 | 2 | — | |
QDFZHFJIXUUJBE
|
8.3 | IC50 | 2 | — | |
QYOOPWNXGCHVME
|
8.3 | IC50 | 2 | — | |
SOJORSMYDWVCJP
|
8.3 | IC50 | 2 | — | |
UFTVLKDQOGAMAF
|
8.3 | IC50 | 2 | — | |
WSLCBKLAKWPNRS
|
8.3 | IC50 | 2 | — | |
XYYUONVZPWBNMS
|
8.3 | IC50 | 2 | — | |
YAJGIHMFZQZBOI
|
8.3 | IC50 | 2 | — | |
ZBTYTRHPZXUMHE
|
8.3 | IC50 | 2 | — | |
NSSGEOSIDLVXLC
|
8.2 | IC50 | 2 | — | |
BNCDEGOHMGKVSC
|
8.2 | IC50 | 2 | — | |
GIIXJDCFQJQOJU
|
8.2 | IC50 | 2 | — | |
NJIVJKWGLFWRER
|
8.2 | IC50 | 2 | — | |
SSRVZOUCWCJWRF
|
8.2 | IC50 | 2 | — | |
UFLJSDDIILZXQC
|
8.2 | IC50 | 2 | — | |
FWGSFILZFNXMHO
|
8.2 | IC50 | 2 | — | |
PBYZYQNLHOJHBY
|
8.2 | IC50 | 2 | — | |
GOYSUCROGDOVQW
|
8.2 | IC50 | 2 | — | |
HFKGXBIBYCUDKG
|
8.2 | IC50 | 2 | — | |
AXRKLNCGVDURIG
|
8.2 | IC50 | 2 | — | |
GBGCYRWGGGBDRM
|
8.2 | IC50 | 2 | — | |
RECCKGZZXRVOCZ
|
8.2 | IC50 | 2 | — | |
GWJHMRBQEUHFOC
|
8.2 | Ki | 42 | — | |
NXUJCUODKLXIPE
|
8.2 | IC50 | 2 | — | |
QHGSRVBVRLMYKL
|
8.2 | IC50 | 2 | — | |
SRJJNRIRROSSLD
|
8.2 | IC50 | 2 | — | |
TUSAVAMNJRWMLZ
|
8.2 | IC50 | 2 | — | |
VYDMLEVVUWMMDW
|
8.2 | IC50 | 2 | — | |
WUCQKINAICDMQD
|
8.2 | IC50 | 2 | — | |
BBJXVAVUGRNQFP
|
8.2 | IC50 | 5 | — | |
DWZCDSLYZDTWQH
|
8.2 | IC50 | 5 | — | |
GXXQTUGBAPRNKE
|
8.2 | IC50 | 2 | — | |
ITXKGBBXVAPCIH
|
8.2 | IC50 | 2 | — | |
XTVAOEKBSKZYFK
|
8.2 | IC50 | 2 | — | |
AKYGBXZKHJOPDB
|
8.2 | IC50 | 3 | — | |
DLYKSKLOFRPDPD
|
8.2 | IC50 | 2 | — | |
ONDIGGGYJRDIFY
|
8.2 | IC50 | 2 | — | |
SRJJNRIRROSSLD
|
8.2 | IC50 | 3 | — | |
ALLGNFRRMBCRHD
|
8.2 | IC50 | 2 | — | |
IEESPAXLZMRDHR
|
8.2 | IC50 | 2 | — | |
IQJONXIMMCOKLM
|
8.2 | IC50 | 2 | — | |
YHXSFEKLXZCQNP
|
8.2 | IC50 | 2 | — |