Target Details
| UniProt AC | P23443 |
|---|---|
| Gene Symbol | RPS6KB1 |
| Protein Name | Ribosomal protein S6 kinase beta-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 1,180
- Clinical molecules 27
- Avg pChEMBL 7.62
KEGG Pathways (31)
- AMPK signaling pathway
- Acute myeloid leukemia
- Apelin signaling pathway
- Autophagy - animal
- Breast cancer
- Chemical carcinogenesis - receptor activation
- Choline metabolism in cancer
- Colorectal cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocrine resistance
- ErbB signaling pathway
- Fc gamma R-mediated phagocytosis
- Gastric cancer
- HIF-1 signaling pathway
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human immunodeficiency virus 1 infection
- Human papillomavirus infection
- Insulin resistance
- Insulin signaling pathway
- Longevity regulating pathway
- Longevity regulating pathway - multiple species
- PD-L1 expression and PD-1 checkpoint pathway in cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Proteoglycans in cancer
- Shigellosis
- TGF-beta signaling pathway
- Thermogenesis
- mTOR signaling pathway
Active Molecules (1,180)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IVUDZHTWTDSSEV
|
8.4 | IC50 | 2 | — | |
SYDBWNWRQBYWOH
|
8.4 | IC50 | 2 | — | |
FKRLYOFLOQRBNO
|
8.4 | IC50 | 2 | — | |
LTLAIOBQBYOIBO
|
8.4 | IC50 | 2 | — | |
PPACVGVOVMKIML
|
8.4 | IC50 | 2 | — | |
SCJPEHNHLXDUFG
|
8.4 | IC50 | 2 | — | |
KGAVPNAQEZTLRD
|
8.3 | IC50 | 2 | — | |
SKTCDUXPKLCJIP
|
8.3 | IC50 | 3 | — | |
FTCVWEWECUNCTD
|
8.3 | IC50 | 2 | — | |
KFYULJIROFVBPN
|
8.3 | IC50 | 2 | — | |
MDBLXTCBPCQULU
|
8.3 | IC50 | 2 | — | |
QXYORZQKCYQMNP
|
8.3 | IC50 | 2 | — | |
RLUCUWZCWXANSZ
|
8.3 | IC50 | 2 | — | |
JBXFRDRWIIKKEZ
|
8.3 | IC50 | 2 | — | |
FSQLPFIYROJSSI
|
8.3 | IC50 | 2 | — | |
KWBXLLQBOZJIAV
|
8.3 | IC50 | 2 | — | |
PJVIGFLRGLEWPN
|
8.3 | IC50 | 2 | — | |
GFWUCLLYVKRKSO
|
8.3 | IC50 | 2 | — | |
GHPKEUAQEZZNIT
|
8.3 | IC50 | 2 | — | |
OPYPJZSJHHSMJL
|
8.3 | IC50 | 2 | — | |
FTLGJGCPUAMLIH
|
8.3 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
8.3 | Ki | 118 | — | |
OTXCECJXPQIXAF
|
8.3 | IC50 | 2 | — | |
PELODSQJHQJMMD
|
8.3 | IC50 | 2 | — | |
UREVFJWGXHMNOI
|
8.3 | IC50 | 2 | — | |
YGQJBWJOHRVWHU
|
8.3 | IC50 | 3 | — | |
AKLMWTZNFKEMQK
|
8.3 | IC50 | 2 | — | |
ALXARYSWRHEWCG
|
8.3 | IC50 | 2 | — | |
TZUSMCMWLCUCGL
|
8.3 | IC50 | 2 | — | |
WHMIUKFQZDKPNG
|
8.3 | IC50 | 2 | — | |
XYZFWUNBADWKLH
|
8.3 | IC50 | 2 | — | |
AUWAFCLIMMJGIZ
|
8.3 | IC50 | 2 | — | |
AVMOOTKRYPDMNB
|
8.3 | IC50 | 2 | — | |
BPJUPXXKAPKTBS
|
8.3 | IC50 | 2 | — | |
COUYLVUYFPDVOO
|
8.3 | IC50 | 2 | — | |
CVDCAMRBGDHTGD
|
8.3 | IC50 | 2 | — | |
DCGFVBYKXGOXIU
|
8.3 | IC50 | 2 | — | |
DPTJVGTULVNDHT
|
8.3 | IC50 | 2 | — | |
FVBJUIPMIDIVCZ
|
8.3 | IC50 | 2 | — | |
GGAFUEXMMLDLSP
|
8.3 | IC50 | 2 | — | |
GHRNTQYBWZUASM
|
8.3 | IC50 | 2 | — | |
GTSLYQNOEMZGNU
|
8.3 | IC50 | 2 | — | |
HDCBQKJBEKMFAM
|
8.3 | IC50 | 2 | — | |
HEIGJIKPAPHGIP
|
8.3 | IC50 | 2 | — | |
HTWLRLMWASQHEU
|
8.3 | IC50 | 2 | — | |
IHXIXEFPEXLJCZ
|
8.3 | IC50 | 2 | — | |
JGYPQUJMROMGBO
|
8.3 | IC50 | 2 | — | |
KZLHWAOADZPQDT
|
8.3 | IC50 | 2 | — | |
LJKNFVAAARXIMN
|
8.3 | IC50 | 2 | — | |
LJKNFVAAARXIMN
|
8.3 | IC50 | 2 | — |