Target Details
| UniProt AC | P23443 |
|---|---|
| Gene Symbol | RPS6KB1 |
| Protein Name | Ribosomal protein S6 kinase beta-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 1,180
- Clinical molecules 27
- Avg pChEMBL 7.62
KEGG Pathways (31)
- AMPK signaling pathway
- Acute myeloid leukemia
- Apelin signaling pathway
- Autophagy - animal
- Breast cancer
- Chemical carcinogenesis - receptor activation
- Choline metabolism in cancer
- Colorectal cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocrine resistance
- ErbB signaling pathway
- Fc gamma R-mediated phagocytosis
- Gastric cancer
- HIF-1 signaling pathway
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human immunodeficiency virus 1 infection
- Human papillomavirus infection
- Insulin resistance
- Insulin signaling pathway
- Longevity regulating pathway
- Longevity regulating pathway - multiple species
- PD-L1 expression and PD-1 checkpoint pathway in cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Proteoglycans in cancer
- Shigellosis
- TGF-beta signaling pathway
- Thermogenesis
- mTOR signaling pathway
Active Molecules (1,180)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NVNKWJJSRWQTOL
|
8.6 | IC50 | 2 | — | |
RBBGFPFJXKWNLT
|
8.6 | IC50 | 2 | — | |
WUMMWDXRTHGRCO
|
8.6 | IC50 | 2 | — | |
GBOPQOSLCOHLCP
|
8.6 | IC50 | 4 | — | |
JBVURKUJSPOJSL
|
8.6 | IC50 | 2 | — | |
PNRZJJLWTXOCFE
|
8.6 | IC50 | 2 | — | |
QABWGDMMZLJSRS
|
8.6 | IC50 | 4 | — | |
RBIOEFDNYQWSEM
|
8.6 | IC50 | 2 | — | |
RWBMPHFTXFAKIZ
|
8.6 | IC50 | 2 | — | |
WQRREPRLHYMJEK
|
8.6 | IC50 | 2 | — | |
XBOMQGBNZCOWGB
|
8.6 | IC50 | 2 | — | |
ZHWCYSIHEZKFKK
|
8.6 | IC50 | 2 | — | |
AHFPBQFTVHYBMP
|
8.6 | IC50 | 2 | — | |
BBZZGHQVCVQLBB
|
8.6 | IC50 | 2 | — | |
BFLHCYRERXMTKZ
|
8.6 | IC50 | 2 | — | |
DZNGHHAQHVFGAF
|
8.6 | IC50 | 2 | — | |
GNOBRAMAIHJFOP
|
8.6 | IC50 | 2 | — | |
PTOIXCNADVPLTL
|
8.6 | IC50 | 2 | — | |
URIUMRYBFCLNMT
|
8.6 | IC50 | 2 | — | |
VUVBORUFCYIRBE
|
8.6 | IC50 | 2 | — | |
WZYKPNJEZBIZHP
|
8.6 | IC50 | 2 | — | |
XAVPWAIYBBCDNE
|
8.6 | IC50 | 2 | — | |
CBBZXHUFHIEZHP
|
8.5 | IC50 | 4 | — | |
FCMPFDJGJGIJNQ
|
8.5 | IC50 | 2 | — | |
FVGWPRCBTOEKKZ
|
8.5 | IC50 | 2 | — | |
MNAVNDWRKFKOGX
|
8.5 | IC50 | 2 | — | |
SDKIMOPCSMIIJC
|
8.5 | IC50 | 2 | — | |
INFMNFLDNVYAMO
|
8.5 | IC50 | 2 | — | |
LLIYOFOBWKBOEE
|
8.5 | IC50 | 2 | — | |
WGAZQGSVJXMVOV
|
8.5 | IC50 | 2 | — | |
YFRKDKXIBIGAAM
|
8.5 | IC50 | 2 | — | |
DKRZLTGERJSUDX
|
8.5 | IC50 | 2 | — | |
HZQDPLPFNYFLTM
|
8.5 | IC50 | 2 | — | |
ITZVXMVPGXCHHN
|
8.5 | IC50 | 2 | — | |
QNTRMTAUUIEBHU
|
8.5 | IC50 | 2 | — | |
QWDUSFJGONFTMI
|
8.5 | IC50 | 2 | — | |
VPNSTYRFYMPBQK
|
8.5 | IC50 | 2 | — | |
YOVNFNXUCOWYSG
|
8.5 | Ki | 33 | Yes | |
GIAKGRDDSYYQQS
|
8.5 | IC50 | 5 | — | |
JQTUGUXQKTXVPW
|
8.5 | IC50 | 2 | — | |
NXVPWAJSJJLIEJ
|
8.5 | IC50 | 2 | — | |
WIHRPNRYTMAFLK
|
8.5 | IC50 | 2 | — | |
GTUAZZUFAUMXII
|
8.5 | IC50 | 2 | — | |
PIVDYIBVDVOUTC
|
8.5 | IC50 | 2 | — | |
YNPQIFHMRSVLHW
|
8.5 | IC50 | 3 | — | |
ZWIYTRXREXLLRD
|
8.5 | IC50 | 2 | — | |
BGUOWQGLKCCWAA
|
8.5 | IC50 | 2 | — | |
BZOAWHFCLQZEIR
|
8.5 | IC50 | 2 | — | |
FJOQZMMQNNGPJK
|
8.5 | IC50 | 2 | — | |
NTSTWVKDSHLTLO
|
8.5 | IC50 | 2 | — |