Target Details
| UniProt AC | P23443 |
|---|---|
| Gene Symbol | RPS6KB1 |
| Protein Name | Ribosomal protein S6 kinase beta-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 1,180
- Clinical molecules 27
- Avg pChEMBL 7.62
KEGG Pathways (31)
- AMPK signaling pathway
- Acute myeloid leukemia
- Apelin signaling pathway
- Autophagy - animal
- Breast cancer
- Chemical carcinogenesis - receptor activation
- Choline metabolism in cancer
- Colorectal cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocrine resistance
- ErbB signaling pathway
- Fc gamma R-mediated phagocytosis
- Gastric cancer
- HIF-1 signaling pathway
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human immunodeficiency virus 1 infection
- Human papillomavirus infection
- Insulin resistance
- Insulin signaling pathway
- Longevity regulating pathway
- Longevity regulating pathway - multiple species
- PD-L1 expression and PD-1 checkpoint pathway in cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Proteoglycans in cancer
- Shigellosis
- TGF-beta signaling pathway
- Thermogenesis
- mTOR signaling pathway
Active Molecules (1,180)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
STVCAXFLBPJWGX
|
8.7 | IC50 | 2 | — | |
UOFRCDSWOWULBQ
|
8.7 | IC50 | 2 | — | |
WNBFWWDKYZWYOX
|
8.7 | IC50 | 4 | — | |
XMHXPVAYPRDKLU
|
8.7 | IC50 | 2 | — | |
XQARBBFJIGXIQL
|
8.7 | IC50 | 2 | — | |
XYZNKCSDQRKAFR
|
8.7 | Ki | 53 | — | |
DPOINXAMYFWFQQ
|
8.7 | IC50 | 4 | — | |
FFERJDPLOMISPG
|
8.7 | IC50 | 4 | — | |
GYEINYAKLFRDRF
|
8.7 | IC50 | 2 | — | |
ILZXORYWWZNZFW
|
8.7 | IC50 | 4 | — | |
IVOSBLQIUULOJZ
|
8.7 | IC50 | 2 | — | |
MGYJNZHGAIGKBJ
|
8.7 | IC50 | 2 | — | |
ODYFSBTYYQCOOI
|
8.7 | IC50 | 2 | — | |
SARBPKFLMZQUBL
|
8.7 | IC50 | 2 | — | |
SWAZPZDRQOTKRL
|
8.7 | IC50 | 2 | — | |
DEEBDOUWFMNWMC
|
8.7 | IC50 | 2 | — | |
GEVIIBINALZINE
|
8.7 | IC50 | 2 | — | |
IQANLWOGWYDRQM
|
8.7 | IC50 | 2 | — | |
JRKHYWUIWWXMOR
|
8.7 | IC50 | 2 | — | |
LKAJMVXQBAURGH
|
8.7 | IC50 | 2 | — | |
MMMSSXLSEGSDHS
|
8.7 | IC50 | 4 | — | |
MOYOONIFAFLCQH
|
8.7 | IC50 | 2 | — | |
NLKBUXJOZSFKGH
|
8.7 | IC50 | 2 | — | |
UZGVQLRDYZTKCP
|
8.7 | IC50 | 2 | — | |
BBBBDEZZSLFOAB
|
8.6 | IC50 | 2 | — | |
CHNUAVFQDQXIJR
|
8.6 | IC50 | 2 | — | |
DGRRIAPTLIYFBK
|
8.6 | IC50 | 2 | — | |
HOKDRFCPZWCKRR
|
8.6 | IC50 | 2 | — | |
PIVZZRIUTCLWJD
|
8.6 | IC50 | 2 | — | |
PVABXGMHLMUIRO
|
8.6 | IC50 | 2 | — | |
BHCBOHJYGRDABU
|
8.6 | IC50 | 2 | — | |
BIPPZTXGSWIXFV
|
8.6 | IC50 | 4 | — | |
DXXQAWREKCQJCS
|
8.6 | IC50 | 4 | — | |
GEZVKRSPTDGJTN
|
8.6 | IC50 | 2 | — | |
GYYUJPVOODOEGB
|
8.6 | IC50 | 2 | — | |
JHGDIFKUZFGJGH
|
8.6 | IC50 | 2 | — | |
KREFPQLDZVYMGF
|
8.6 | IC50 | 2 | — | |
LYWHOKPGLIJYCR
|
8.6 | IC50 | 2 | — | |
PRCCLLICHPIENY
|
8.6 | IC50 | 2 | — | |
GZCKUAGOLSTPFP
|
8.6 | IC50 | 2 | — | |
IOBVCHJTLVPPBR
|
8.6 | Ki | 39 | — | |
KTJLGJXEMNHTFM
|
8.6 | IC50 | 2 | — | |
MRYHAUHEHQAMRQ
|
8.6 | IC50 | 2 | — | |
OYHQDBOKPCRZLQ
|
8.6 | IC50 | 2 | — | |
YZSOMODRJHNWOR
|
8.6 | IC50 | 3 | — | |
ALUYNNMYLAIVQS
|
8.6 | IC50 | 5 | — | |
DQQHLMXTQBGBKI
|
8.6 | IC50 | 2 | — | |
INWAPLGMARPPCH
|
8.6 | IC50 | 3 | — | |
LYRHYDHWKBCSKX
|
8.6 | IC50 | 2 | — | |
NOEMLPJTVJSKAG
|
8.6 | IC50 | 2 | — |