Target Details
| UniProt AC | P23443 |
|---|---|
| Gene Symbol | RPS6KB1 |
| Protein Name | Ribosomal protein S6 kinase beta-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 1,180
- Clinical molecules 27
- Avg pChEMBL 7.62
KEGG Pathways (31)
- AMPK signaling pathway
- Acute myeloid leukemia
- Apelin signaling pathway
- Autophagy - animal
- Breast cancer
- Chemical carcinogenesis - receptor activation
- Choline metabolism in cancer
- Colorectal cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocrine resistance
- ErbB signaling pathway
- Fc gamma R-mediated phagocytosis
- Gastric cancer
- HIF-1 signaling pathway
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human immunodeficiency virus 1 infection
- Human papillomavirus infection
- Insulin resistance
- Insulin signaling pathway
- Longevity regulating pathway
- Longevity regulating pathway - multiple species
- PD-L1 expression and PD-1 checkpoint pathway in cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Proteoglycans in cancer
- Shigellosis
- TGF-beta signaling pathway
- Thermogenesis
- mTOR signaling pathway
Active Molecules (1,180)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VSYXMJKNSDTUDZ
|
8.9 | IC50 | 2 | — | |
UUKGDBLVFLHJLM
|
8.9 | IC50 | 2 | — | |
BZNBRLIMNHJECW
|
8.8 | IC50 | 2 | — | |
CJAKBHSFDAWLEM
|
8.8 | IC50 | 2 | — | |
DCCVOYXJENYWAN
|
8.8 | IC50 | 2 | — | |
FPTITAKKUXPEEF
|
8.8 | IC50 | 2 | — | |
HIIWAIXZTVGCMF
|
8.8 | IC50 | 2 | — | |
KRASTSBCSPTMCM
|
8.8 | IC50 | 2 | — | |
OIPUWMRXDFZHSB
|
8.8 | IC50 | 2 | — | |
OSJZAAQNTQOLFR
|
8.8 | IC50 | 4 | — | |
WTXODCJICMVXLA
|
8.8 | IC50 | 2 | — | |
YFBSBJBNKSZCLY
|
8.8 | IC50 | 4 | — | |
ZJYLBZWVQNQDEG
|
8.8 | IC50 | 2 | — | |
ZRGLOCZGYSBBDT
|
8.8 | IC50 | 2 | — | |
BDNUCRITDDPHCE
|
8.8 | IC50 | 2 | — | |
DHPPYCQBIXXVFM
|
8.8 | IC50 | 2 | — | |
DYERZMIJULWDJN
|
8.8 | IC50 | 2 | — | |
LPZBVVARVJQTAW
|
8.8 | IC50 | 4 | — | |
QMDGKERTSOLCLO
|
8.8 | IC50 | 2 | — | |
SPGIFTJYQFCUFV
|
8.8 | IC50 | 2 | — | |
BAOLTBUSJGESBU
|
8.8 | IC50 | 2 | — | |
IAQPRHKDYNIJFN
|
8.8 | IC50 | 2 | — | |
OPMLKXQPQMIRGC
|
8.8 | IC50 | 2 | — | |
XMZNZUXMEXIQDA
|
8.8 | IC50 | 2 | — | |
YMZVKOCKXHQABC
|
8.8 | IC50 | 2 | — | |
CEEYIVGYAJJUTB
|
8.8 | IC50 | 2 | — | |
GAYRMKRSQCSTHF
|
8.8 | IC50 | 2 | — | |
IZYOAMDRLUYOEU
|
8.8 | IC50 | 2 | — | |
PFBFGTPOSIOVBG
|
8.8 | IC50 | 2 | — | |
POWWZDRBSXYCHK
|
8.8 | IC50 | 2 | — | |
TZUSMCMWLCUCGL
|
8.8 | IC50 | 2 | — | |
XZEFTYTUTILRTG
|
8.8 | IC50 | 3 | — | |
BKWJTVGUNLNJRS
|
8.7 | IC50 | 2 | — | |
FVZJYBLPVJFOIE
|
8.7 | IC50 | 2 | — | |
HNNYZFMEBYIBQI
|
8.7 | IC50 | 2 | — | |
LYVAUQAZKOULMJ
|
8.7 | IC50 | 2 | — | |
WCBMSENIXPZAJT
|
8.7 | IC50 | 4 | — | |
CLVJQNXBLQVWOL
|
8.7 | IC50 | 2 | — | |
FMBXWBOUJFSHEK
|
8.7 | IC50 | 2 | — | |
GVXVELAMVOVTAS
|
8.7 | IC50 | 2 | — | |
IKNUWQGXRGMLOY
|
8.7 | IC50 | 2 | — | |
RELZDYOQGLSASS
|
8.7 | IC50 | 2 | — | |
RUZSLLVTXSZYLX
|
8.7 | IC50 | 2 | — | |
AWCXGXCOCLVOSP
|
8.7 | IC50 | 2 | — | |
DSLKQMBMFBKGRK
|
8.7 | IC50 | 4 | — | |
FLGUGRAWIWHCJF
|
8.7 | IC50 | 4 | — | |
JNWSILMDEXPLAM
|
8.7 | IC50 | 2 | — | |
KLIDFKYRDXZCOP
|
8.7 | IC50 | 4 | — | |
OVSZEAIKKSSNTM
|
8.7 | IC50 | 2 | — | |
PANRGGPPMYRRKF
|
8.7 | IC50 | 2 | — |