Target Details
| UniProt AC | P23443 |
|---|---|
| Gene Symbol | RPS6KB1 |
| Protein Name | Ribosomal protein S6 kinase beta-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 1,180
- Clinical molecules 27
- Avg pChEMBL 7.62
KEGG Pathways (31)
- AMPK signaling pathway
- Acute myeloid leukemia
- Apelin signaling pathway
- Autophagy - animal
- Breast cancer
- Chemical carcinogenesis - receptor activation
- Choline metabolism in cancer
- Colorectal cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocrine resistance
- ErbB signaling pathway
- Fc gamma R-mediated phagocytosis
- Gastric cancer
- HIF-1 signaling pathway
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human immunodeficiency virus 1 infection
- Human papillomavirus infection
- Insulin resistance
- Insulin signaling pathway
- Longevity regulating pathway
- Longevity regulating pathway - multiple species
- PD-L1 expression and PD-1 checkpoint pathway in cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Proteoglycans in cancer
- Shigellosis
- TGF-beta signaling pathway
- Thermogenesis
- mTOR signaling pathway
Active Molecules (1,180)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WRWWQYDXUXWNBS
|
9.1 | IC50 | 2 | — | |
HZCSYARAUKXOFF
|
9.1 | IC50 | 2 | — | |
NERGHRXOVVUXNP
|
9.1 | IC50 | 2 | — | |
JKUFJTIKVQADGJ
|
9.1 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
9.1 | IC50 | 408 | — | |
AJHYNXPIENOPCI
|
9.1 | IC50 | 2 | — | |
DCGJPYQDBNQMHR
|
9.1 | IC50 | 2 | — | |
LDOJECIQNJBVHE
|
9.1 | IC50 | 2 | — | |
MOQRMWMUHUDDJL
|
9.1 | IC50 | 2 | — | |
QZMSENZZQWAYFQ
|
9.1 | IC50 | 2 | — | |
SKBGXGJACXJIHW
|
9.1 | IC50 | 2 | — | |
USJIOUUNHSENIY
|
9.1 | IC50 | 2 | — | |
WMGWBZXIQPUBFV
|
9.1 | IC50 | 2 | — | |
XCTRDYNPZXNINO
|
9.1 | IC50 | 2 | — | |
RBMOLIOJAWRTIV
|
9.0 | IC50 | 5 | — | |
AOMMHIPSMLPJKQ
|
9.0 | IC50 | 4 | — | |
DHEDUDJQNPBXHX
|
9.0 | IC50 | 2 | — | |
FECIECQDFIPTFY
|
9.0 | IC50 | 2 | — | |
FJZFOTKMZCYJDF
|
9.0 | IC50 | 4 | — | |
HJFIIHVQWRUIBJ
|
9.0 | IC50 | 2 | — | |
JNORLXPNXUUQIG
|
9.0 | IC50 | 2 | — | |
KIOZCJFPASJAIE
|
9.0 | IC50 | 2 | — | |
KMAREWFGYUHLEK
|
9.0 | IC50 | 2 | — | |
TYXBLVVBDICGSW
|
9.0 | IC50 | 2 | — | |
UUQUQPUHXKTHDD
|
9.0 | IC50 | 2 | — | |
YFTUDCDZHZYZAB
|
9.0 | IC50 | 2 | — | |
AESKEMGHXXMKDS
|
9.0 | IC50 | 2 | — | |
BBTVEWXIIOMQJE
|
9.0 | IC50 | 2 | — | |
CDOPSCORKPCGMU
|
9.0 | IC50 | 2 | — | |
CNFJGGPOIJUVKL
|
9.0 | IC50 | 2 | — | |
DCRRXSUQGXVDLQ
|
9.0 | IC50 | 2 | — | |
HXAUJHZZPCBFPN
|
9.0 | IC50 | 4 | — | |
MERNKFHEABWVHR
|
9.0 | IC50 | 2 | — | |
ODIBHBBABRKJIO
|
9.0 | IC50 | 2 | — | |
RGACXOZZMADIOP
|
9.0 | IC50 | 2 | — | |
SXNSPDSUPXINEH
|
9.0 | IC50 | 2 | — | |
YOXMBPVKSDWRAV
|
9.0 | IC50 | 2 | — | |
BVYUJCVPGYLIMY
|
8.9 | IC50 | 5 | — | |
BXSXPCFESWIUHR
|
8.9 | IC50 | 3 | — | |
YFPFHMOVBQYQHX
|
8.9 | IC50 | 2 | — | |
AUVWKQGXLMJMFV
|
8.9 | IC50 | 2 | — | |
BMPTUVXOIJURIA
|
8.9 | IC50 | 2 | — | |
CGTSDPKWWBJGPO
|
8.9 | IC50 | 2 | — | |
CIVKYRVMDOHDLK
|
8.9 | IC50 | 2 | — | |
GOPVGMUVSGFICI
|
8.9 | IC50 | 2 | — | |
GXYOPEGHNADCQI
|
8.9 | IC50 | 2 | — | |
HQPYWCQKQNPHGR
|
8.9 | IC50 | 2 | — | |
IUEUJHZZCUYXKU
|
8.9 | IC50 | 2 | — | |
SIRZTYWYVGTPEV
|
8.9 | IC50 | 4 | — | |
UPNXCPZAHNPTHY
|
8.9 | IC50 | 2 | — |