Target Details
| UniProt AC | P23443 |
|---|---|
| Gene Symbol | RPS6KB1 |
| Protein Name | Ribosomal protein S6 kinase beta-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 1,180
- Clinical molecules 27
- Avg pChEMBL 7.62
KEGG Pathways (31)
- AMPK signaling pathway
- Acute myeloid leukemia
- Apelin signaling pathway
- Autophagy - animal
- Breast cancer
- Chemical carcinogenesis - receptor activation
- Choline metabolism in cancer
- Colorectal cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocrine resistance
- ErbB signaling pathway
- Fc gamma R-mediated phagocytosis
- Gastric cancer
- HIF-1 signaling pathway
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human immunodeficiency virus 1 infection
- Human papillomavirus infection
- Insulin resistance
- Insulin signaling pathway
- Longevity regulating pathway
- Longevity regulating pathway - multiple species
- PD-L1 expression and PD-1 checkpoint pathway in cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Proteoglycans in cancer
- Shigellosis
- TGF-beta signaling pathway
- Thermogenesis
- mTOR signaling pathway
Active Molecules (1,180)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CJMAJALOUQYWKR
|
7.3 | IC50 | 2 | — | |
KSFGFFQQMLCHJC
|
7.3 | IC50 | 3 | — | |
MAZAMYSGSCRKQA
|
7.3 | IC50 | 3 | — | |
WPDWJWPDAWEUDW
|
7.3 | IC50 | 3 | — | |
QSIHIKQTAYUVBM
|
7.3 | IC50 | 2 | — | |
TXCWDJYJHQBALS
|
7.3 | IC50 | 2 | — | |
DMKGGPGYGHAZLX
|
7.3 | IC50 | 2 | — | |
GQHMZZXJWGPHDA
|
7.3 | Ki | 20 | — | |
GVMDVMPNOAVKJR
|
7.3 | Ki | 26 | Yes | |
HCRQPXYLXXLKPT
|
7.3 | Ki | 5 | — | |
NPLQZQGAZAUUTB
|
7.3 | Ki | 9 | — | |
PYXQMJSGJIJHJT
|
7.3 | Ki | 28 | — | |
RWEHAHIEUDLKGT
|
7.3 | Ki | 33 | — | |
SEVCBWKJSOLMNQ
|
7.3 | Ki | 38 | — | |
VLNRWHJKUQHNER
|
7.3 | IC50 | 2 | — | |
VWVYILCFSYNJHF
|
7.3 | Ki | 49 | — | |
WKWGFJFNCXAUEX
|
7.3 | Ki | 14 | Yes | |
GJTZJJVUDPIOOX
|
7.3 | IC50 | 2 | — | |
HIUMPNPHWNCFBW
|
7.3 | IC50 | 3 | — | |
OIDHYGPWCABWGM
|
7.3 | IC50 | 3 | — | |
OZKLXNJWZUXQAC
|
7.3 | IC50 | 3 | — | |
QXQBUHCSEYQBBD
|
7.3 | IC50 | 2 | — | |
FOUODSJMGGENMN
|
7.3 | IC50 | 2 | — | |
XVNFBGOMJAUCKO
|
7.3 | IC50 | 3 | — | |
ZOAQMCSHCNWYTR
|
7.3 | IC50 | 2 | — | |
GYOJAUPBIHPKFM
|
7.2 | IC50 | 2 | — | |
MYNMWFXSBRRDCA
|
7.2 | IC50 | 3 | — | |
OEFRWUPQSHQOMD
|
7.2 | IC50 | 2 | — | |
CBEVEZTUJLXHCH
|
7.2 | IC50 | 2 | — | |
PNFSXOCCWZKQET
|
7.2 | IC50 | 2 | — | |
RBVRSMCCUMHQRB
|
7.2 | IC50 | 2 | — | |
VXJNQGXNBJPYRH
|
7.2 | IC50 | 2 | — | |
JGFQBBRDUAPPHV
|
7.2 | IC50 | 2 | — | |
AXTAPYRUEKNRBA
|
7.2 | IC50 | 24 | — | |
SZUFVMKRAKNXNR
|
7.2 | IC50 | 2 | — | |
WTZPLLLUSQHZPS
|
7.2 | IC50 | 3 | — | |
ADGNQMNEVYGZMR
|
7.2 | IC50 | 2 | — | |
AMOJCASSAZNSPN
|
7.2 | IC50 | 3 | — | |
CCXAZVAJEKWLBF
|
7.2 | IC50 | 2 | — | |
CJGRHBWUMPISNN
|
7.2 | IC50 | 2 | — | |
CKKONTWSDZZMIN
|
7.2 | IC50 | 2 | — | |
CUBQBLLPFKWXRJ
|
7.2 | IC50 | 2 | — | |
DXIDCSBKUQPZSC
|
7.2 | IC50 | 2 | — | |
GEKRHWYIFQTBAI
|
7.2 | IC50 | 2 | — | |
GXPXLCKCZLZHRD
|
7.2 | IC50 | 2 | — | |
JCZDYEBBWFRSGI
|
7.2 | IC50 | 2 | — | |
KNHGAKWDTPNWIC
|
7.2 | IC50 | 2 | — | |
ORFQXNMTLHYGKN
|
7.2 | IC50 | 2 | — | |
YBAOLDRYZQFNOG
|
7.2 | IC50 | 2 | — | |
YRBXVESCSKRYGH
|
7.2 | IC50 | 2 | — |