Target Details
| UniProt AC | P23443 |
|---|---|
| Gene Symbol | RPS6KB1 |
| Protein Name | Ribosomal protein S6 kinase beta-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 1,180
- Clinical molecules 27
- Avg pChEMBL 7.62
KEGG Pathways (31)
- AMPK signaling pathway
- Acute myeloid leukemia
- Apelin signaling pathway
- Autophagy - animal
- Breast cancer
- Chemical carcinogenesis - receptor activation
- Choline metabolism in cancer
- Colorectal cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocrine resistance
- ErbB signaling pathway
- Fc gamma R-mediated phagocytosis
- Gastric cancer
- HIF-1 signaling pathway
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human immunodeficiency virus 1 infection
- Human papillomavirus infection
- Insulin resistance
- Insulin signaling pathway
- Longevity regulating pathway
- Longevity regulating pathway - multiple species
- PD-L1 expression and PD-1 checkpoint pathway in cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Proteoglycans in cancer
- Shigellosis
- TGF-beta signaling pathway
- Thermogenesis
- mTOR signaling pathway
Active Molecules (1,180)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MPLYXIRRQBHUMZ
|
7.7 | IC50 | 2 | — | |
UNRMMILBIIITEU
|
7.7 | IC50 | 3 | — | |
UUQADGWFQPYANC
|
7.7 | IC50 | 3 | — | |
XOKVRHIXBOTBIS
|
7.7 | IC50 | 2 | — | |
XOLMMSRNKAXJNW
|
7.7 | IC50 | 2 | — | |
DZSUJUOJJJCWGG
|
7.7 | Ki | 55 | Yes | |
GTTSANJRVQIGFM
|
7.7 | IC50 | 3 | — | |
HNGORDVZNLENER
|
7.7 | IC50 | 2 | — | |
JWSHIVZYYNSBPC
|
7.7 | IC50 | 3 | — | |
MQRDVGBWWVWMEN
|
7.7 | Ki | 47 | — | |
NDBVBSHGQOHFEG
|
7.7 | IC50 | 2 | — | |
RQAXQHGKLHCEHQ
|
7.7 | IC50 | 2 | — | |
SFPWNTQWFFNJIH
|
7.7 | Ki | 48 | — | |
AFNBZIQKVHCFIT
|
7.7 | IC50 | 2 | — | |
CIGYNACQDYSRCK
|
7.7 | IC50 | 2 | — | |
COANUJWURZDRKT
|
7.7 | IC50 | 3 | — | |
GSWYQMZWPSIFDH
|
7.7 | IC50 | 3 | — | |
LCJCTWAUTPNXKH
|
7.7 | IC50 | 2 | — | |
LCTWFROMTHUGEH
|
7.7 | IC50 | 2 | — | |
NZSCAAFVISAPPF
|
7.7 | IC50 | 2 | — | |
OBAJYVJLNXGBOG
|
7.7 | IC50 | 3 | — | |
OKNLBGPUZXUDJN
|
7.7 | IC50 | 2 | — | |
OPLIFFRWVGVBNQ
|
7.7 | IC50 | 2 | — | |
OZLZGTRWERFWLS
|
7.7 | IC50 | 2 | — | |
PDULEZONFAQVLI
|
7.7 | IC50 | 3 | — | |
QCETXMLIFLYKQH
|
7.7 | IC50 | 3 | — | |
QTAJBRBSORWZDL
|
7.7 | IC50 | 2 | — | |
UUVFRMLWZBOAOM
|
7.7 | IC50 | 3 | — | |
WVHAMWAJDWCCNB
|
7.7 | IC50 | 2 | — | |
XGXROOYTEGFACC
|
7.7 | IC50 | 3 | — | |
BTWIQOVBQBEGSN
|
7.7 | IC50 | 2 | — | |
DHNFKQPWVFBZIL
|
7.7 | IC50 | 3 | — | |
NYUVVVDGKCTKKF
|
7.7 | Ki | 3 | — | |
PLSBOWQASGBKLJ
|
7.7 | IC50 | 2 | — | |
RWTOHSIAYKNWEG
|
7.7 | IC50 | 2 | — | |
ULUQVPIBCGQLRE
|
7.7 | IC50 | 2 | — | |
KTBJSZWXMIFTCA
|
7.6 | IC50 | 2 | — | |
ORMLOSONIQIDBI
|
7.6 | IC50 | 3 | — | |
OUIQTZMFLWJZDO
|
7.6 | IC50 | 2 | — | |
PZRFGYNACSHNJL
|
7.6 | IC50 | 2 | — | |
UEJXELMBDCXXAQ
|
7.6 | IC50 | 9 | — | |
YOZQOXRJRWBJBE
|
7.6 | IC50 | 2 | — | |
ZSRJHGJCRGZJNH
|
7.6 | IC50 | 2 | — | |
BIKYYRLGHVJTHO
|
7.6 | IC50 | 2 | — | |
GJOLOIJGOFZXST
|
7.6 | IC50 | 3 | — | |
JPUOKUGRWCCCOL
|
7.6 | IC50 | 2 | — | |
NCPSMNWGGLQFPN
|
7.6 | IC50 | 2 | — | |
URYOYOMAOIZWMC
|
7.6 | IC50 | 2 | — | |
VSIZGIFPGSTFOV
|
7.6 | IC50 | 3 | — | |
CHTMRWQLNNRRFJ
|
7.6 | Ki | 70 | — |