Target Details
| UniProt AC | P23443 |
|---|---|
| Gene Symbol | RPS6KB1 |
| Protein Name | Ribosomal protein S6 kinase beta-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 1,180
- Clinical molecules 27
- Avg pChEMBL 7.62
KEGG Pathways (31)
- AMPK signaling pathway
- Acute myeloid leukemia
- Apelin signaling pathway
- Autophagy - animal
- Breast cancer
- Chemical carcinogenesis - receptor activation
- Choline metabolism in cancer
- Colorectal cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocrine resistance
- ErbB signaling pathway
- Fc gamma R-mediated phagocytosis
- Gastric cancer
- HIF-1 signaling pathway
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human immunodeficiency virus 1 infection
- Human papillomavirus infection
- Insulin resistance
- Insulin signaling pathway
- Longevity regulating pathway
- Longevity regulating pathway - multiple species
- PD-L1 expression and PD-1 checkpoint pathway in cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Proteoglycans in cancer
- Shigellosis
- TGF-beta signaling pathway
- Thermogenesis
- mTOR signaling pathway
Active Molecules (1,180)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PDWXUDFNTMNSTQ
|
7.9 | IC50 | 2 | — | |
VHQHJGLYTLVYKC
|
7.9 | Ki | 4 | — | |
WARQMCTXKWMOOS
|
7.9 | IC50 | 2 | — | |
FCWOKBAQNTUHOR
|
7.9 | IC50 | 2 | — | |
WMHVRDMXMXGXEQ
|
7.9 | IC50 | 2 | — | |
VCQOVNIEIZUWRP
|
7.9 | IC50 | 2 | — | |
CSWJHPQUGVGBIV
|
7.8 | IC50 | 2 | — | |
OFGXCCDXYUXZLX
|
7.8 | IC50 | 2 | — | |
QYGYKSCXWILKPY
|
7.8 | IC50 | 2 | — | |
SWEZOINTKPVMEG
|
7.8 | IC50 | 3 | — | |
UHKHLFSIUKCZQE
|
7.8 | IC50 | 2 | — | |
WBXAZIHUNVIWMP
|
7.8 | IC50 | 2 | — | |
AKPRVQKEQOLLND
|
7.8 | IC50 | 3 | — | |
BXOCOVVDMXWPQN
|
7.8 | IC50 | 3 | — | |
RKSDWJBFBPKMFN
|
7.8 | IC50 | 3 | — | |
DSXXEELGXBCYNQ
|
7.8 | IC50 | 28 | Yes | |
JPXOUJDDCUAQFV
|
7.8 | IC50 | 2 | — | |
REICLTJSLHAADW
|
7.8 | IC50 | 2 | — | |
RFRCSMPUQCLUQP
|
7.8 | IC50 | 2 | — | |
RKZPJUYYKFXMLU
|
7.8 | IC50 | 3 | — | |
SFVVRJCZCCKAKZ
|
7.8 | IC50 | 2 | — | |
SZCJQZJURBSEEN
|
7.8 | IC50 | 2 | — | |
UGSMZLIUJPNNFB
|
7.8 | IC50 | 2 | — | |
BGCQKRIZWQNGJK
|
7.8 | IC50 | 2 | — | |
FJMQHAKZJZXKED
|
7.8 | IC50 | 2 | — | |
FKGMUZBYHNMNSM
|
7.8 | IC50 | 2 | — | |
FWCNPQPYGXFFSI
|
7.8 | IC50 | 3 | — | |
KRUKDVBCEQTOCL
|
7.8 | IC50 | 3 | — | |
MTYMWGNJKDHWGN
|
7.8 | Ki | 18 | — | |
NRBGHJOLFXFDFP
|
7.8 | IC50 | 3 | — | |
NSTHHWXJQFPGNS
|
7.8 | IC50 | 2 | — | |
OPOGDZANLATWGS
|
7.8 | Ki | 9 | — | |
RLEBVXHKDJKLHD
|
7.8 | IC50 | 2 | — | |
SPCDTNUNXCPQPQ
|
7.8 | IC50 | 2 | — | |
VYWFLGVPKXPOKG
|
7.8 | IC50 | 2 | — | |
WYIHYHHXTNJQBE
|
7.8 | IC50 | 2 | — | |
XYXLUJQBBIBJFV
|
7.8 | Ki | 36 | — | |
ZKZXNDJNWUTGDK
|
7.8 | Ki | 14 | — | |
CBIORNCAYCELBK
|
7.8 | IC50 | 2 | — | |
LDFNTCCSAZUOGI
|
7.8 | IC50 | 2 | — | |
PSYMLFSTUXAGFZ
|
7.8 | IC50 | 3 | — | |
YJOVRFFTOQUZOT
|
7.8 | IC50 | 2 | — | |
WLLLTIDXGZYUPF
|
7.8 | IC50 | 2 | — | |
DEJZGAXRKVTAOI
|
7.7 | IC50 | 2 | — | |
DUXGYYIANJMODE
|
7.7 | IC50 | 4 | — | |
IJCVUIACMPFTBC
|
7.7 | IC50 | 2 | — | |
IWGIUZSSSYNTCU
|
7.7 | IC50 | 2 | — | |
NCAWHBLWUZPAJV
|
7.7 | IC50 | 2 | — | |
YERVWHTZAGNUEL
|
7.7 | IC50 | 2 | — | |
ZMIIFFANXFZVIP
|
7.7 | IC50 | 2 | — |