Target Details
| UniProt AC | P23443 |
|---|---|
| Gene Symbol | RPS6KB1 |
| Protein Name | Ribosomal protein S6 kinase beta-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 1,180
- Clinical molecules 27
- Avg pChEMBL 7.62
KEGG Pathways (31)
- AMPK signaling pathway
- Acute myeloid leukemia
- Apelin signaling pathway
- Autophagy - animal
- Breast cancer
- Chemical carcinogenesis - receptor activation
- Choline metabolism in cancer
- Colorectal cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocrine resistance
- ErbB signaling pathway
- Fc gamma R-mediated phagocytosis
- Gastric cancer
- HIF-1 signaling pathway
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human immunodeficiency virus 1 infection
- Human papillomavirus infection
- Insulin resistance
- Insulin signaling pathway
- Longevity regulating pathway
- Longevity regulating pathway - multiple species
- PD-L1 expression and PD-1 checkpoint pathway in cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Proteoglycans in cancer
- Shigellosis
- TGF-beta signaling pathway
- Thermogenesis
- mTOR signaling pathway
Active Molecules (1,180)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WOVZBZPJTHFHQU
|
8.0 | IC50 | 2 | — | |
CUNFBMBOBMNCLK
|
8.0 | IC50 | 2 | — | |
DDSBMKNXVLTBPK
|
8.0 | IC50 | 3 | — | |
BKVQOYGRGNOWSO
|
8.0 | IC50 | 2 | — | |
CKXDOCDUQDMDLW
|
8.0 | IC50 | 2 | — | |
GGCRTRINBCFKEU
|
8.0 | IC50 | 2 | — | |
JGTLCWBXBNQZGX
|
8.0 | IC50 | 3 | — | |
JMLSGXAFWBMOHG
|
8.0 | IC50 | 2 | — | |
LSOZVYDETZGJRK
|
8.0 | IC50 | 3 | — | |
MCCCQFAOMZMZKE
|
8.0 | Ki | 52 | — | |
NMOBMAXTXLXAEL
|
8.0 | IC50 | 2 | — | |
OQISTSSMSVJSIA
|
8.0 | IC50 | 2 | — | |
VNTBJROWKHAASF
|
8.0 | IC50 | 2 | — | |
WXELJDBMNZEMTI
|
8.0 | IC50 | 2 | — | |
IEQAHFTVGLZUBI
|
8.0 | IC50 | 8 | — | |
NBIUBKUPIRWCOK
|
8.0 | IC50 | 2 | — | |
BTHHPHAIATVJEX
|
8.0 | IC50 | 2 | — | |
HAKWYGIXPYBWTK
|
8.0 | IC50 | 2 | — | |
IZYYQEHJGDFEGP
|
8.0 | IC50 | 2 | — | |
QSSBFEIISOSMHF
|
8.0 | IC50 | 2 | — | |
STKRLXKLVFXNGU
|
8.0 | IC50 | 2 | — | |
SZZYWZLEQNPFSI
|
8.0 | IC50 | 2 | — | |
UUHAJBVAHFVAPV
|
8.0 | IC50 | 2 | — | |
WVWKMLRXXWPJFD
|
8.0 | Kd | 3 | — | |
GHPPBFVKOZAUET
|
8.0 | IC50 | 2 | — | |
IWBOFXHEGIMYAM
|
7.9 | IC50 | 3 | — | |
OVECHGPXFIKXEK
|
7.9 | IC50 | 3 | — | |
VPHVDXANMJOXMQ
|
7.9 | IC50 | 3 | — | |
AUJLKABCXYHSMK
|
7.9 | IC50 | 2 | — | |
AWJSEDIXXHFUSS
|
7.9 | IC50 | 3 | — | |
BCODCVMBVICQAV
|
7.9 | Ki | 4 | — | |
CHCRYENRCVXRJA
|
7.9 | IC50 | 2 | — | |
CQAJURUOVMFONQ
|
7.9 | IC50 | 2 | — | |
IIRWNGPLJQXWFJ
|
7.9 | IC50 | 21 | — | |
JMHMGIHHTONCMK
|
7.9 | IC50 | 3 | — | |
JSWNYZOFSLKPNK
|
7.9 | IC50 | 2 | — | |
JXOFZRFVAKUHDR
|
7.9 | IC50 | 2 | — | |
KCRPTSILJIQNRD
|
7.9 | IC50 | 2 | — | |
LLDVRUBUBPSOMY
|
7.9 | Ki | 4 | — | |
MOZQZSIJFQHRST
|
7.9 | IC50 | 2 | — | |
DKSNLQYRZJKYOC
|
7.9 | Ki | 51 | — | |
UMTWTCVTRDYHQQ
|
7.9 | Ki | 56 | — | |
XCHWBXBDZRJVDP
|
7.9 | Ki | 51 | — | |
BXFVYQXRSWCGMU
|
7.9 | IC50 | 3 | — | |
FWADTUVPBQDECD
|
7.9 | IC50 | 2 | — | |
HGCQHRUBKWVKHA
|
7.9 | IC50 | 2 | — | |
JYHDWNWORMYNHM
|
7.9 | IC50 | 2 | — | |
KXEJAEQUXNWZTK
|
7.9 | IC50 | 2 | — | |
NHNIQMDXSHWKPU
|
7.9 | IC50 | 2 | — | |
OSVUGUHRKMMBSE
|
7.9 | Kd | 170 | — |