Target Details
| UniProt AC | P23443 |
|---|---|
| Gene Symbol | RPS6KB1 |
| Protein Name | Ribosomal protein S6 kinase beta-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 1,180
- Clinical molecules 27
- Avg pChEMBL 7.62
KEGG Pathways (31)
- AMPK signaling pathway
- Acute myeloid leukemia
- Apelin signaling pathway
- Autophagy - animal
- Breast cancer
- Chemical carcinogenesis - receptor activation
- Choline metabolism in cancer
- Colorectal cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocrine resistance
- ErbB signaling pathway
- Fc gamma R-mediated phagocytosis
- Gastric cancer
- HIF-1 signaling pathway
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human immunodeficiency virus 1 infection
- Human papillomavirus infection
- Insulin resistance
- Insulin signaling pathway
- Longevity regulating pathway
- Longevity regulating pathway - multiple species
- PD-L1 expression and PD-1 checkpoint pathway in cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Proteoglycans in cancer
- Shigellosis
- TGF-beta signaling pathway
- Thermogenesis
- mTOR signaling pathway
Active Molecules (1,180)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SKFWPKNHRNPQQX
|
10.2 | IC50 | 2 | — | |
LCTSWTGAHKAMHA
|
10.0 | IC50 | 2 | — | |
XHEDMNVAFNSTPV
|
10.0 | IC50 | 2 | — | |
UVOCNINDPZNPIC
|
9.9 | IC50 | 2 | — | |
ZJDZJPZEQDNRHD
|
9.8 | IC50 | 2 | — | |
FCRMIQHGMSYNNQ
|
9.7 | IC50 | 2 | — | |
LIHXUIBRFWFAPL
|
9.7 | IC50 | 2 | — | |
KVMVAUMDSYMRST
|
9.6 | IC50 | 2 | — | |
RWOKWMSYJITVKH
|
9.6 | IC50 | 2 | — | |
BYUUFRNHCFTPTI
|
9.4 | IC50 | 2 | — | |
HNAFGFOVDGEYQN
|
9.4 | IC50 | 2 | — | |
XPDILXVPINMDCE
|
9.4 | IC50 | 2 | — | |
FIZSPRJMYGKSMB
|
9.4 | IC50 | 2 | — | |
XQZHZCUJORPEOS
|
9.4 | IC50 | 2 | — | |
RGZTUPDJESIZJE
|
9.4 | IC50 | 2 | — | |
FVVVHVQIBBDHNP
|
9.3 | IC50 | 2 | — | |
IKONXWFEIGCAGN
|
9.3 | IC50 | 2 | — | |
PANNEFPLJLKPJS
|
9.3 | IC50 | 2 | — | |
UALHJBCHHRMERK
|
9.3 | IC50 | 2 | — | |
XCVFPZYBAGFIKJ
|
9.3 | IC50 | 2 | — | |
RXAZPQCDGXHCAO
|
9.3 | IC50 | 2 | — | |
HAWOAWLBNXPWTR
|
9.2 | IC50 | 2 | — | |
ARGMPCCCUNPEOG
|
9.2 | IC50 | 4 | — | |
AWDSGNQQQIADCU
|
9.2 | IC50 | 2 | — | |
OHPGVBAFZWTDHG
|
9.2 | IC50 | 2 | — | |
QVHGKNYBLQTWEC
|
9.2 | IC50 | 2 | — | |
QWYFZEWKZWQGDU
|
9.2 | IC50 | 2 | — | |
RBMOLIOJAWRTIV
|
9.2 | IC50 | 4 | — | |
UFMCGKYLIYMLOY
|
9.2 | IC50 | 3 | — | |
RHWHWWRJINHZQN
|
9.2 | IC50 | 2 | — | |
YRQSEFHVBKRZFV
|
9.2 | IC50 | 2 | — | |
LAJUPICIRDRINN
|
9.2 | IC50 | 2 | — | |
VWYGEDAFWDXUMQ
|
9.2 | IC50 | 3 | — | |
XQZHZCUJORPEOS
|
9.2 | IC50 | 2 | — | |
CEOCDNNZGIOOGD
|
9.2 | IC50 | 2 | — | |
GIMRLCRHTAIQJM
|
9.2 | IC50 | 2 | — | |
XDCFPLHPOOPKGK
|
9.2 | IC50 | 2 | — | |
KTEVQEUEMLYYMP
|
9.1 | IC50 | 2 | — | |
NUPWMMJWFAYJED
|
9.1 | IC50 | 2 | — | |
XLYVQVWMTOLDNL
|
9.1 | IC50 | 21 | — | |
XLYVQVWMTOLDNL
|
9.1 | IC50 | 21 | — | |
AGDQZNITYJKXQO
|
9.1 | IC50 | 2 | — | |
BQJKHAVFMIHHLG
|
9.1 | IC50 | 2 | — | |
DLFSJMCJAANTKH
|
9.1 | IC50 | 2 | — | |
IDVXLGVNCNGJLE
|
9.1 | IC50 | 2 | — | |
JKACOTYFJGVPGL
|
9.1 | IC50 | 2 | — | |
KVGXNQBHBACSGG
|
9.1 | IC50 | 2 | — | |
NCEITWUOOXWJSM
|
9.1 | IC50 | 2 | — | |
POQNJRCZSQACTE
|
9.1 | IC50 | 2 | — | |
WJQJOCPGZFNQLW
|
9.1 | IC50 | 2 | — |