Target Details
UniProt ACP23415
Gene SymbolGLRA1
Protein NameGlycine receptor subunit alpha-1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 20
  • Clinical molecules 0
  • Avg pChEMBL 6.56
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (20)
InChIKey pChEMBL Type Targets Clinical
RETKEJUHMKGUFW 7.3 IC50 2
NRGHCWQGTHPFTE 7.1 IC50 2
WOHVJFQJNVSXAC 7.0 IC50 2
CMOAVMXESDVBSR 7.0 IC50 2
JIEFHNBYMOMHOJ 7.0 IC50 2
AXMKQFHQYPQAND 6.9 IC50 2
QMGVPVSNSZLJIA 6.9 IC50 2
ZYQOFJMYFTVXSE 6.8 IC50 2
SRSRXUGMICPDQE 6.6 IC50 2
DAIFFNCOIUBILX 6.5 IC50 2
ZKLHAXAVCMWFHX 6.4 IC50 2
IAAAVXPESPTBDM 6.4 IC50 2
WAPQUQFEOPBULC 6.3 IC50 2
BNLMIPXTXOQLRY 6.3 IC50 2
PLFAVVBJYCHLRJ 6.2 IC50 2
SITBEFQCWFXBGL 6.2 IC50 2
AOUHSICIWMGARK 6.1 IC50 2
NCZVCWOBWGTWOF 6.1 IC50 2
UIFKYMJUYHLRDT 6.1 IC50 2
VHGCDTVCOLNTBX 6.0 Ki 19
2D structure