Target Details
| UniProt AC | P22894 |
|---|---|
| Gene Symbol | MMP8 |
| Protein Name | Neutrophil collagenase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 934
- Clinical molecules 624
- Avg pChEMBL 7.65
Active Molecules (934)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DBYYJEGRUPLGLD
|
7.8 | Ki | 7 | Yes | |
HMXFQXRHTFBPFX
|
7.8 | IC50 | 4 | — | |
JZIODDCGNMBMLB
|
7.8 | IC50 | 5 | Yes | |
LTRFXCQZLSSSPG
|
7.8 | IC50 | 3 | Yes | |
RSMQCSLXBNSQJJ
|
7.8 | Ki | 7 | Yes | |
SJEBBPDOLJCLQH
|
7.8 | IC50 | 4 | Yes | |
SYAAEFMNVNGONW
|
7.8 | IC50 | 5 | Yes | |
ZGBAPSHWPBXEKN
|
7.8 | IC50 | 10 | — | |
IVFPKTAJBISJDW
|
7.8 | Ki | 4 | Yes | |
JPTZDOYPNCQOTF
|
7.8 | Ki | 4 | Yes | |
MXPPQWXYSRGIMR
|
7.8 | Ki | 4 | Yes | |
NSZHVJWSFHBPMB
|
7.8 | Ki | 3 | Yes | |
NSZHVJWSFHBPMB
|
7.8 | Ki | 4 | Yes | |
QVKJHTQSZHYYSV
|
7.8 | IC50 | 3 | — | |
YMYDSTVSNKTLJM
|
7.8 | Ki | 7 | Yes | |
YZDALJROFHNCEI
|
7.8 | Ki | 3 | Yes | |
DDIJQZRWMIFTHG
|
7.8 | IC50 | 3 | — | |
NPTUUUXCZCQNQS
|
7.8 | IC50 | 4 | — | |
PHBHELQPDZPJEY
|
7.8 | IC50 | 3 | — | |
ZSZOBVLJWIXXND
|
7.8 | IC50 | 5 | Yes | |
AQKDLUIAUGFUEC
|
7.7 | Ki | 7 | Yes | |
DUPWUQYVKWCUOG
|
7.7 | Ki | 7 | — | |
HLJHTDAQDAFOFS
|
7.7 | Ki | 7 | Yes | |
YVCXCHMORKNFGU
|
7.7 | IC50 | 5 | Yes | |
BRKOQUQULDVEDN
|
7.7 | Ki | 4 | Yes | |
CWYHAUKCGMBLAH
|
7.7 | Ki | 2 | — | |
DKPAZQOKVRHHON
|
7.7 | IC50 | 4 | Yes | |
JRCGNOYYZQLNTH
|
7.7 | Ki | 11 | Yes | |
JVBPIOHSXSYBRG
|
7.7 | Ki | 7 | Yes | |
RWOLXJOULAGHOB
|
7.7 | IC50 | 5 | Yes | |
VKESMHHXVWGWQQ
|
7.7 | IC50 | 2 | — | |
XVUIGVGFVWRFJO
|
7.7 | Ki | 8 | Yes | |
ALUHGPANWKZMAA
|
7.7 | IC50 | 3 | Yes | |
AMUGNOPZMAZKFD
|
7.7 | Ki | 4 | Yes | |
AQWIHDVVCANJLS
|
7.7 | Ki | 3 | — | |
HCCYYUWFQWPMDZ
|
7.7 | Ki | 4 | Yes | |
HRMWQQBRFJMAPM
|
7.7 | IC50 | 3 | Yes | |
JGRIYRSQHHLUHI
|
7.7 | IC50 | 7 | Yes | |
JNBNCWQZPZWAOV
|
7.7 | IC50 | 2 | — | |
JXGACOLDOLFHQF
|
7.7 | IC50 | 4 | Yes | |
LKNQKZXVRWZYQR
|
7.7 | IC50 | 3 | Yes | |
MVEPSFJZKBVDHV
|
7.7 | IC50 | 7 | Yes | |
OEPLGUBYTRYCJX
|
7.7 | IC50 | 7 | Yes | |
QXLMMZHXXOWCDY
|
7.7 | IC50 | 4 | Yes | |
SFWRCXWXHAIKBP
|
7.7 | IC50 | 5 | Yes | |
UJACCCBUXXMATQ
|
7.7 | IC50 | 3 | Yes | |
WYVILPRSBDCCKY
|
7.7 | Ki | 7 | Yes | |
WYWULSIANADMTA
|
7.7 | IC50 | 2 | Yes | |
XTRJAENNSAJIAU
|
7.7 | IC50 | 3 | Yes | |
XVUIGVGFVWRFJO
|
7.7 | Ki | 4 | — |