Target Details
| UniProt AC | P22894 |
|---|---|
| Gene Symbol | MMP8 |
| Protein Name | Neutrophil collagenase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 934
- Clinical molecules 624
- Avg pChEMBL 7.65
Active Molecules (934)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HSJPSXSXQYYJSY
|
8.0 | Ki | 7 | Yes | |
IGRVUOPMHNISAV
|
8.0 | IC50 | 3 | Yes | |
LRVIJTRFTUQDKW
|
8.0 | IC50 | 7 | Yes | |
OHZMUNMVWGUMMY
|
8.0 | IC50 | 6 | Yes | |
OTJGAHJWYSLTDB
|
8.0 | IC50 | 3 | Yes | |
PMVTXYIJWIAFKQ
|
8.0 | Ki | 4 | Yes | |
RSWUWSKXIDLCIR
|
8.0 | IC50 | 4 | Yes | |
UKBWLBZDMUKXSY
|
8.0 | IC50 | 3 | Yes | |
WPXAJFJACNOICK
|
8.0 | Ki | 7 | Yes | |
WVDBZKCLVKPIHE
|
8.0 | IC50 | 3 | Yes | |
WVJHDQDLYDFIKS
|
8.0 | IC50 | 3 | Yes | |
XNKSQYFVFJZMOA
|
8.0 | IC50 | 7 | Yes | |
YLYMDJMYRSEUOA
|
8.0 | IC50 | 7 | Yes | |
YMPRSEQZGBKKAZ
|
8.0 | IC50 | 3 | Yes | |
YNIHTMMJQXUNPE
|
8.0 | Ki | 7 | Yes | |
ZVAKMIZOMSWYGQ
|
8.0 | IC50 | 7 | Yes | |
KEHDBOGRIVHUBV
|
8.0 | Ki | 6 | — | |
MDWFJTBWOFNAQX
|
8.0 | IC50 | 7 | Yes | |
BEKYMPWGANBKBK
|
8.0 | Ki | 7 | Yes | |
UFKJDXKTPYNZRZ
|
8.0 | IC50 | 4 | — | |
NKHJMAWHLPBSOA
|
7.9 | Ki | 5 | — | |
FGEXLQKMIJWUIY
|
7.9 | IC50 | 5 | Yes | |
FPIZTGFSDBBQIE
|
7.9 | Ki | 4 | Yes | |
GTZKIGXVCZWIAR
|
7.9 | IC50 | 4 | — | |
JMWYGNIQHYKDCH
|
7.9 | Ki | 7 | Yes | |
NEUXHEKNAOUEQU
|
7.9 | Ki | 7 | Yes | |
ROFAQOFULLWONA
|
7.9 | IC50 | 5 | Yes | |
UHJDYMMCTFTTSW
|
7.9 | Ki | 4 | Yes | |
YLRBOIVJMWEGGX
|
7.9 | Ki | 6 | — | |
UILNVWQPBYOCJX
|
7.9 | IC50 | 2 | Yes | |
BITXXJKMASUYME
|
7.9 | Ki | 7 | Yes | |
DEDGVHPWRWYTIC
|
7.9 | Ki | 4 | Yes | |
IVGHGMHNUBCTDC
|
7.9 | Ki | 6 | Yes | |
KOFNJKLYWDTWHZ
|
7.9 | Ki | 7 | Yes | |
MZISFPSOTJFTTJ
|
7.9 | Ki | 7 | Yes | |
OUMHWPMKRPJGKY
|
7.9 | Ki | 4 | Yes | |
PYHVMKLBOIYJOG
|
7.9 | Ki | 5 | Yes | |
WKYYIJNBJSICFM
|
7.9 | IC50 | 5 | — | |
XJBCYCWPLLYLPI
|
7.9 | Ki | 2 | — | |
XYXRFODFDUOQKS
|
7.9 | Ki | 3 | — | |
ZGSTVUAZFACDLH
|
7.9 | Ki | 4 | — | |
AKWKBACKRMYPRV
|
7.8 | Ki | 6 | Yes | |
CXNJLMYOAJTOHP
|
7.8 | IC50 | 4 | Yes | |
FWNRCECLAVXIOV
|
7.8 | Ki | 4 | Yes | |
JLXRKMSJFVPFIG
|
7.8 | IC50 | 4 | — | |
LMKSZZKXCRCXFM
|
7.8 | Ki | 3 | — | |
NEPHXSICDJEKLG
|
7.8 | IC50 | 6 | — | |
YJBLORWBSQLNFW
|
7.8 | IC50 | 4 | Yes | |
ZGSTVUAZFACDLH
|
7.8 | Ki | 8 | Yes | |
BCOFTFDFNHXYGF
|
7.8 | IC50 | 5 | Yes |