Target Details
| UniProt AC | P22894 |
|---|---|
| Gene Symbol | MMP8 |
| Protein Name | Neutrophil collagenase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 934
- Clinical molecules 624
- Avg pChEMBL 7.65
Active Molecules (934)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RCXJWFMVFQBLSC
|
8.6 | IC50 | 8 | Yes | |
BZVYQWLRCHLAGK
|
8.5 | IC50 | 4 | — | |
FFXPIMSNULYFOV
|
8.5 | IC50 | 6 | Yes | |
GKHRDWHFKKUYAX
|
8.5 | IC50 | 8 | Yes | |
GKHRDWHFKKUYAX
|
8.5 | IC50 | 9 | — | |
GSLSWNSJTMLFSO
|
8.5 | IC50 | 3 | Yes | |
GWEITLSXCOXESW
|
8.5 | IC50 | 7 | Yes | |
HJNKYGBTSGQBDU
|
8.5 | Ki | 10 | — | |
HRTBORRCNRXWRR
|
8.5 | IC50 | 3 | Yes | |
ICFOTHUAZLHTNP
|
8.5 | IC50 | 7 | Yes | |
IRBWGGQXMBAYQL
|
8.5 | IC50 | 7 | Yes | |
JZHHNBACJYFNCE
|
8.5 | IC50 | 4 | — | |
KJOVWWTWOVUHSB
|
8.5 | IC50 | 5 | Yes | |
KVMNMFKBWZIOKY
|
8.5 | IC50 | 3 | Yes | |
LFOGEPKUSWRLCL
|
8.5 | IC50 | 7 | Yes | |
PBJWRLBRUGJQMR
|
8.5 | IC50 | 3 | Yes | |
PUHDBKGWNNZTBP
|
8.5 | Ki | 8 | Yes | |
RSWUWSKXIDLCIR
|
8.5 | IC50 | 4 | Yes | |
UIMOJSHBVUUXAE
|
8.5 | Ki | 3 | — | |
APXZBXMVEOBZDS
|
8.5 | IC50 | 2 | — | |
BLYHHTXBRXLLOI
|
8.5 | IC50 | 7 | Yes | |
CDVYEYANHXGLCX
|
8.5 | Ki | 10 | Yes | |
ULPVLGUDYQAPPV
|
8.5 | Ki | 7 | Yes | |
VSLVJIBOSDQNRC
|
8.5 | Ki | 2 | — | |
XDYZXHJJAIXYOR
|
8.5 | IC50 | 8 | Yes | |
YUWSFQQPCKKPJG
|
8.5 | IC50 | 9 | Yes | |
LFIZWBFUWVSLOR
|
8.5 | Ki | 5 | — | |
MERYKHOGOUEPIA
|
8.5 | Ki | 4 | Yes | |
YDYDCNNQCGFQDL
|
8.5 | Ki | 5 | — | |
IOANZCGEYMTXEK
|
8.4 | IC50 | 7 | Yes | |
LWHRQCDZIRQSAN
|
8.4 | Ki | 3 | Yes | |
GPENKXZRTRUYOG
|
8.4 | IC50 | 4 | Yes | |
HTNLSTWGHBHDPS
|
8.4 | IC50 | 8 | Yes | |
MYGNBBVBBNZVCZ
|
8.4 | Ki | 4 | Yes | |
ZRAUMSIZBNBIFE
|
8.4 | IC50 | 8 | Yes | |
FMEMUXYNXWETSE
|
8.4 | IC50 | 6 | — | |
ACSSJLXQNWFMSO
|
8.4 | Ki | 7 | Yes | |
BDPAGEAOFNRCNJ
|
8.4 | IC50 | 4 | — | |
BEQXRWLSEUIFKP
|
8.4 | Ki | 5 | — | |
BLXHYKZAZZIQOC
|
8.4 | Ki | 3 | — | |
CTVWOVYWOFCAMW
|
8.4 | IC50 | 5 | Yes | |
FCGVXISUYVDDPU
|
8.4 | IC50 | 7 | Yes | |
GFUITADOEPNRML
|
8.4 | Ki | 6 | — | |
GFUITADOEPNRML
|
8.4 | Ki | 11 | Yes | |
HCELOWJRPJWTPO
|
8.4 | Ki | 5 | Yes | |
LXQUQEBAZBLBEJ
|
8.4 | IC50 | 5 | Yes | |
OKYUILRERWOFCH
|
8.4 | IC50 | 7 | Yes | |
PPELJLBDXLMTEW
|
8.4 | IC50 | 3 | Yes | |
RDFQXFRQTOWZEQ
|
8.4 | IC50 | 8 | Yes | |
UDNLRUDZHBXCON
|
8.4 | Ki | 7 | Yes |