Target Details
| UniProt AC | P22894 |
|---|---|
| Gene Symbol | MMP8 |
| Protein Name | Neutrophil collagenase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 934
- Clinical molecules 624
- Avg pChEMBL 7.65
Active Molecules (934)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ORSWNUGKUNQTLF
|
8.7 | IC50 | 7 | Yes | |
QJNGNVJSSUXWBO
|
8.7 | IC50 | 8 | Yes | |
TVNINFNNQVBJHI
|
8.7 | IC50 | 8 | Yes | |
WMYJDFANEQLDGP
|
8.7 | IC50 | 6 | — | |
BYJSIHNQXBCYBX
|
8.7 | IC50 | 3 | Yes | |
DHXMAFQQCCOWGL
|
8.7 | IC50 | 3 | Yes | |
DZCGIZPIPKWUIX
|
8.7 | IC50 | 7 | Yes | |
FNUQESAUEFWUCJ
|
8.7 | IC50 | 3 | Yes | |
GEPDPACRTHVSTD
|
8.7 | IC50 | 2 | Yes | |
GEPDPACRTHVSTD
|
8.7 | IC50 | 3 | Yes | |
HTKNWYDCBWYORK
|
8.7 | IC50 | 3 | Yes | |
JNFMXXAZBVSNRC
|
8.7 | Ki | 4 | Yes | |
JXSWSZIEDSTKDW
|
8.7 | IC50 | 3 | Yes | |
MOPRTFSMCQNUCT
|
8.7 | Ki | 9 | Yes | |
NOYXCNRQZBBVGT
|
8.7 | Ki | 7 | Yes | |
NSDMBIOAMTZMED
|
8.7 | IC50 | 5 | Yes | |
OCSMOTCMPXTDND
|
8.7 | IC50 | 8 | Yes | |
OCSMOTCMPXTDND
|
8.7 | IC50 | 14 | Yes | |
OGWVESDVKZYNCK
|
8.7 | IC50 | 3 | Yes | |
PNICWAPKRSLYIU
|
8.7 | IC50 | 3 | Yes | |
PUBARVPHTAEUJQ
|
8.7 | IC50 | 5 | Yes | |
QSONFBZTWRVCKO
|
8.7 | Ki | 5 | Yes | |
RNWNGVUCFRPGIO
|
8.7 | IC50 | 3 | Yes | |
ROVRDWIOAVCKAV
|
8.7 | IC50 | 2 | Yes | |
ROVRDWIOAVCKAV
|
8.7 | IC50 | 3 | Yes | |
UCWSKTMFEWSSSI
|
8.7 | IC50 | 4 | — | |
VPDOXKSDXTZFIX
|
8.7 | IC50 | 4 | — | |
VZEDRBAGPXKVHL
|
8.7 | IC50 | 3 | Yes | |
YJKSIUVAMOZWEF
|
8.7 | IC50 | 3 | Yes | |
ZRDGYJAMDSHROJ
|
8.7 | IC50 | 7 | Yes | |
SKADGQGCAOBKKC
|
8.7 | Ki | 7 | Yes | |
WFQFQAQNCYHBTC
|
8.7 | IC50 | 8 | Yes | |
UGZOJBSDACNWAB
|
8.6 | Ki | 7 | Yes | |
CQRAUIRVDKNRIO
|
8.6 | IC50 | 9 | Yes | |
IIBGHLQTRXDEKI
|
8.6 | IC50 | 7 | Yes | |
KNFQAZOHJDVGHS
|
8.6 | Ki | 5 | — | |
NZKKRYAESABOSS
|
8.6 | IC50 | 8 | Yes | |
RCGPSTRFXVIUQB
|
8.6 | Ki | 7 | Yes | |
SPEYRVQKGFNUCY
|
8.6 | IC50 | 8 | Yes | |
SYYRIPAKWJBIOW
|
8.6 | IC50 | 8 | Yes | |
UGMRVUAZVAXFHK
|
8.6 | Ki | 8 | Yes | |
VGXYGECPCDQSNI
|
8.6 | IC50 | 6 | Yes | |
VZUMDYFAZYINJW
|
8.6 | Ki | 4 | Yes | |
LHVGXRIIQBVWQU
|
8.6 | Ki | 5 | — | |
SFORRVNMTYAPLQ
|
8.6 | Ki | 4 | Yes | |
YQEMFOGNUTYMTJ
|
8.6 | Ki | 4 | Yes | |
YQEMFOGNUTYMTJ
|
8.6 | IC50 | 5 | — | |
YQEMFOGNUTYMTJ
|
8.6 | IC50 | 5 | Yes | |
WWNOVCQMRIZSRV
|
8.6 | IC50 | 8 | Yes | |
ILTCMGUVAAYHSE
|
8.6 | IC50 | 7 | Yes |