Target Details
| UniProt AC | P22894 |
|---|---|
| Gene Symbol | MMP8 |
| Protein Name | Neutrophil collagenase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 934
- Clinical molecules 624
- Avg pChEMBL 7.65
Active Molecules (934)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ROMGJVVZNVJOPW
|
9.0 | Ki | 10 | Yes | |
XFNJKSWXHKYCFN
|
9.0 | Ki | 10 | Yes | |
CNZGQRARNYMASL
|
9.0 | Ki | 7 | Yes | |
DONMTDNLNMLOIC
|
9.0 | Ki | 13 | Yes | |
HNXQLWUITFQYPE
|
9.0 | Ki | 10 | Yes | |
SNYKGOMEURTYMK
|
9.0 | Ki | 10 | Yes | |
VWKXFDZWHLCIIU
|
9.0 | IC50 | 9 | Yes | |
YXXIQAWIZFAIOP
|
9.0 | Ki | 9 | Yes | |
BDONYXHHXNTUSW
|
8.9 | IC50 | 8 | Yes | |
BWPZARSJOUWFCK
|
8.9 | Ki | 4 | Yes | |
HBYRXCFAHCMHAA
|
8.9 | IC50 | 9 | Yes | |
JGWTVBVOISUVJD
|
8.9 | IC50 | 9 | — | |
LFOGEPKUSWRLCL
|
8.9 | IC50 | 7 | Yes | |
MHGISLAIZQKUNW
|
8.9 | Ki | 7 | Yes | |
NBRBWZJMBITNBC
|
8.9 | IC50 | 8 | Yes | |
AOPZFYOXZYZEAC
|
8.9 | IC50 | 7 | Yes | |
BGBWSADVPWNBME
|
8.9 | IC50 | 9 | Yes | |
GHHVNOZFZMDYFQ
|
8.9 | Ki | 7 | Yes | |
HGCCQMHYESJBML
|
8.9 | Ki | 7 | Yes | |
HXZPYZWICHZKRL
|
8.9 | IC50 | 10 | — | |
LMIHEFSBOIGKDH
|
8.9 | IC50 | 8 | Yes | |
USFNQSYWKLKGHX
|
8.9 | Ki | 4 | Yes | |
VDDKIBQLKXMKIW
|
8.9 | Ki | 7 | Yes | |
CYYCSKFJEOSZTF
|
8.8 | IC50 | 9 | Yes | |
JKRVXAWKSWVVCV
|
8.8 | IC50 | 7 | Yes | |
LTCNKRUYOJZZJO
|
8.8 | IC50 | 7 | Yes | |
XCCIACQOXSWRJQ
|
8.8 | Ki | 7 | Yes | |
ZBRHTUMWSDPCMI
|
8.8 | IC50 | 10 | Yes | |
GETQXLAMYOMSJS
|
8.8 | IC50 | 8 | Yes | |
HGCZRPPCNXJXAB
|
8.8 | IC50 | 7 | Yes | |
JATUSZYMCBLDQS
|
8.8 | IC50 | 8 | Yes | |
LFOGEPKUSWRLCL
|
8.8 | IC50 | 7 | Yes | |
MOHDKNTXJIGORP
|
8.8 | Ki | 7 | Yes | |
RFNUTMXSNZMOSL
|
8.8 | Ki | 7 | Yes | |
VAQNHYAKIUNIKM
|
8.8 | IC50 | 8 | Yes | |
VKFNDAOTTJONML
|
8.8 | IC50 | 9 | Yes | |
VURZBHKGMIEEFK
|
8.8 | Ki | 7 | Yes | |
XFBRPTYLOIFAQR
|
8.8 | IC50 | 8 | Yes | |
AOPYXKATLYBNDC
|
8.8 | Ki | 4 | Yes | |
DGZZVIWCMGVHGV
|
8.8 | IC50 | 11 | Yes | |
QDGVTWBFTFHWOG
|
8.8 | IC50 | 8 | Yes | |
SIEIWCDBNIGNIG
|
8.8 | IC50 | 7 | Yes | |
SLZZXDGACSPBLI
|
8.8 | Ki | 4 | Yes | |
LICFKTFLYQYXDH
|
8.8 | Ki | 4 | Yes | |
NXUHVWMBPOFLMA
|
8.8 | IC50 | 6 | Yes | |
FNURWSLLBXZLRC
|
8.7 | IC50 | 7 | Yes | |
KKVTZTBYJGHGCO
|
8.7 | IC50 | 8 | Yes | |
KOPIIXVBCHXDHO
|
8.7 | IC50 | 8 | Yes | |
SXSIQUOYBXOPSS
|
8.7 | IC50 | 7 | Yes | |
WXNWNNKHEJMQOM
|
8.7 | IC50 | 8 | Yes |