Target Details
| UniProt AC | P22894 |
|---|---|
| Gene Symbol | MMP8 |
| Protein Name | Neutrophil collagenase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 934
- Clinical molecules 624
- Avg pChEMBL 7.65
Active Molecules (934)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZXGBSFAKYZEOPJ
|
9.3 | IC50 | 4 | — | |
OKGPERFMUXABQD
|
9.3 | Ki | 4 | Yes | |
URVVMIUWONGKFU
|
9.3 | Ki | 4 | Yes | |
YKPYIPVDTNNYCN
|
9.3 | IC50 | 11 | Yes | |
NNCVCMDUQDAWGY
|
9.2 | IC50 | 4 | — | |
VAQVSMUJBPTVIS
|
9.2 | IC50 | 7 | Yes | |
VXXBOZLJRUCYLE
|
9.2 | Ki | 3 | Yes | |
YUPQCEGDWHZIJW
|
9.2 | Ki | 4 | Yes | |
AKNDZTHCJLFZCF
|
9.2 | IC50 | 9 | Yes | |
IXVDOEAUVAJHER
|
9.2 | IC50 | 7 | Yes | |
PRJCFROAJDAXAD
|
9.2 | Ki | 8 | Yes | |
RAPHEYPJGISJNU
|
9.2 | Ki | 10 | Yes | |
SNMQJFHUOZBSDS
|
9.2 | Ki | 5 | — | |
UIHJPRDGPQZWAH
|
9.2 | Ki | 3 | Yes | |
CJQLPOBRKZCBHK
|
9.2 | Ki | 4 | Yes | |
FYGGOGPIPBSHEF
|
9.2 | Ki | 4 | Yes | |
UTMWGWRRRXPAQY
|
9.2 | Ki | 3 | Yes | |
CMKYCYOBCXIZPF
|
9.2 | IC50 | 4 | — | |
DRZSKJBSLSLPQN
|
9.2 | Ki | 4 | Yes | |
FEWWJFPIJXNCFE
|
9.2 | Ki | 7 | Yes | |
KKRBZYCHOUTMBU
|
9.2 | Ki | 4 | Yes | |
LCYYUMHWMVOGPC
|
9.2 | IC50 | 8 | Yes | |
QYZPDCGWIJYZMN
|
9.2 | Ki | 8 | Yes | |
SPBFQBQZZSCDQE
|
9.2 | Ki | 2 | — | |
UGBFTDFVLBACAS
|
9.2 | Ki | 7 | Yes | |
ULILDPSFFUSXJH
|
9.2 | IC50 | 9 | Yes | |
ULILDPSFFUSXJH
|
9.2 | IC50 | 7 | — | |
ZBOSPOSQGJWURE
|
9.2 | Ki | 5 | — | |
HFLSBITWFGZVGL
|
9.1 | IC50 | 11 | Yes | |
QUSCQVGYLGWIJY
|
9.1 | Ki | 4 | Yes | |
UTSFQPTVPZNJJH
|
9.1 | IC50 | 7 | Yes | |
BUKCBCDGRPOFJP
|
9.1 | IC50 | 9 | Yes | |
IWQSGINKBSWILJ
|
9.1 | IC50 | 10 | — | |
MOPRTFSMCQNUCT
|
9.1 | Ki | 4 | Yes | |
QYCUMAKSYBUWER
|
9.1 | Ki | 6 | — | |
BUEVFADAMKTXGD
|
9.1 | IC50 | 5 | Yes | |
QLTNWLFWQKKDEO
|
9.1 | IC50 | 7 | Yes | |
XMVQXBAGOTVZDD
|
9.1 | IC50 | 4 | — | |
BZVYQWLRCHLAGK
|
9.0 | IC50 | 10 | Yes | |
FFEXFXFAIZBMGO
|
9.0 | Ki | 3 | Yes | |
BCORPMHFJPQWGD
|
9.0 | Ki | 3 | Yes | |
CSPDSJARPZQPMQ
|
9.0 | Ki | 7 | Yes | |
FDELEKDMYZLVHP
|
9.0 | IC50 | 3 | Yes | |
IMKDKHQDFFLOKK
|
9.0 | IC50 | 13 | Yes | |
KXYFKTLZKSANJT
|
9.0 | Ki | 4 | Yes | |
LTRQYQYXWUQKJZ
|
9.0 | IC50 | 3 | Yes | |
LTTRJMCJTUBEGF
|
9.0 | IC50 | 4 | — | |
LTVIJEFEZVFIST
|
9.0 | IC50 | 14 | Yes | |
OLEYZXUQGOKVKT
|
9.0 | IC50 | 7 | Yes | |
PECBDMOWKLTTSB
|
9.0 | IC50 | 4 | — |